NO20050088L - Kationisk substituerte difenylazefidinoner, fremgangsmate for deres fremstilling, medikamenter inneholdende nevnte forbindelser og anvendelse derav - Google Patents
Kationisk substituerte difenylazefidinoner, fremgangsmate for deres fremstilling, medikamenter inneholdende nevnte forbindelser og anvendelse deravInfo
- Publication number
- NO20050088L NO20050088L NO20050088A NO20050088A NO20050088L NO 20050088 L NO20050088 L NO 20050088L NO 20050088 A NO20050088 A NO 20050088A NO 20050088 A NO20050088 A NO 20050088A NO 20050088 L NO20050088 L NO 20050088L
- Authority
- NO
- Norway
- Prior art keywords
- compounds
- diphenylazofidinones
- processes
- preparation
- medicaments containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
Det er beskrevet forbindelser med formel I, hvori RI, R2, R3, R4, R5 og R6 har de angitte betydningene, samt deres fysiologisk godtagbare salter. Forbindelsene egner seg for eksempel som hypolipidemika.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10227507A DE10227507A1 (de) | 2002-06-19 | 2002-06-19 | Kationisch substituierte Diphenylazetidinone, Verfahren zu deren Herstellung, diese Verbindungen enthaltende Arzneimittel und deren Verwendung |
PCT/EP2003/005814 WO2004000803A1 (de) | 2002-06-19 | 2003-06-04 | Kationisch substituierte diphenylazetidinone, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20050088L true NO20050088L (no) | 2005-01-06 |
Family
ID=29719282
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20050088A NO20050088L (no) | 2002-06-19 | 2005-01-06 | Kationisk substituerte difenylazefidinoner, fremgangsmate for deres fremstilling, medikamenter inneholdende nevnte forbindelser og anvendelse derav |
Country Status (26)
Country | Link |
---|---|
EP (1) | EP1517890B1 (no) |
JP (1) | JP2005533071A (no) |
KR (1) | KR20050010061A (no) |
CN (1) | CN1662494A (no) |
AT (1) | ATE401304T1 (no) |
AU (1) | AU2003238209B2 (no) |
BR (1) | BR0311984A (no) |
CA (1) | CA2490108A1 (no) |
DE (2) | DE10227507A1 (no) |
DK (1) | DK1517890T3 (no) |
ES (1) | ES2310662T3 (no) |
HR (1) | HRP20041202A2 (no) |
IL (1) | IL165790A (no) |
MA (1) | MA27251A1 (no) |
MX (1) | MXPA04012308A (no) |
NO (1) | NO20050088L (no) |
PA (1) | PA8575601A1 (no) |
PL (1) | PL372660A1 (no) |
PT (1) | PT1517890E (no) |
RS (1) | RS108604A (no) |
RU (1) | RU2315753C2 (no) |
SV (1) | SV2004001555A (no) |
TW (1) | TW200406380A (no) |
UY (1) | UY27852A1 (no) |
WO (1) | WO2004000803A1 (no) |
ZA (1) | ZA200409379B (no) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0215579D0 (en) | 2002-07-05 | 2002-08-14 | Astrazeneca Ab | Chemical compounds |
JP4688819B2 (ja) | 2003-12-23 | 2011-05-25 | アストラゼネカ アクチボラグ | コレステロール吸収阻害活性を有するジフェニルアゼチジノン誘導体 |
KR101351209B1 (ko) | 2004-12-03 | 2014-02-06 | 머크 샤프 앤드 돔 코포레이션 | Cb1 길항제로서 치환된 피페라진 |
BRPI0609614A2 (pt) * | 2005-04-04 | 2010-04-20 | Univ Pontificia Catolica Chile | uso de ezetimiba na prevenção e tratamento de litìases de colesterol na árvore biliar |
TW200738676A (en) | 2005-06-20 | 2007-10-16 | Schering Corp | Heteroatom-linked substituted piperidines and derivatives thereof useful as histamine H3 antagonists |
SA06270191B1 (ar) | 2005-06-22 | 2010-03-29 | استرازينيكا ايه بي | مشتقات من 2- أزيتيدينون جديدة باعتبارها مثبطات لامتصاص الكوليسترول لعلاج حالات فرط نسبة الدهون في الدم |
AR060623A1 (es) | 2006-04-27 | 2008-07-02 | Astrazeneca Ab | Compuestos derivados de 2-azetidinona y un metodo de preparacion |
MX2009001043A (es) | 2006-08-08 | 2009-02-06 | Sanofi Aventis | Imidazolidina-2,4-dionas sustituidas con arilaminoarilalquilo, procedimiento para preparalas, medicamentos que comprenden estos compuestos y su uso. |
DE102007002260A1 (de) | 2007-01-16 | 2008-07-31 | Sanofi-Aventis | Verwendung von substituierten Pyranonsäurederivaten zur Herstellung von Medikamenten zur Behandlung des Metabolischen Syndroms |
EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
DE102007063671A1 (de) | 2007-11-13 | 2009-06-25 | Sanofi-Aventis Deutschland Gmbh | Neue kristalline Diphenylazetidinonhydrate, diese Verbindungen enthaltende Arzneimittel und deren Verwendung |
WO2010003624A2 (en) | 2008-07-09 | 2010-01-14 | Sanofi-Aventis | Heterocyclic compounds, processes for their preparation, medicaments comprising these compounds, and the use thereof |
WO2010068601A1 (en) | 2008-12-08 | 2010-06-17 | Sanofi-Aventis | A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof |
US9212175B2 (en) | 2009-03-06 | 2015-12-15 | Lipideon Biotechnology Ag | Pharmaceutical hypocholesterolemic compositions |
CN101993403B (zh) | 2009-08-11 | 2012-07-11 | 浙江海正药业股份有限公司 | 氮杂环丁酮类化合物及医药应用 |
SG178880A1 (en) | 2009-08-26 | 2012-04-27 | Sanofi Sa | Novel crystalline heteroaromatic fluoroglycoside hydrates, pharmaceuticals comprising these compounds and their use |
US8933024B2 (en) | 2010-06-18 | 2015-01-13 | Sanofi | Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases |
US8710050B2 (en) | 2011-03-08 | 2014-04-29 | Sanofi | Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof |
US8901114B2 (en) | 2011-03-08 | 2014-12-02 | Sanofi | Oxathiazine derivatives substituted with carbocycles or heterocycles, method for producing same, drugs containing said compounds, and use thereof |
WO2012120056A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
US8828994B2 (en) | 2011-03-08 | 2014-09-09 | Sanofi | Di- and tri-substituted oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof |
WO2012120053A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
EP2567959B1 (en) | 2011-09-12 | 2014-04-16 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10042447A1 (de) * | 2000-08-29 | 2002-03-28 | Aventis Pharma Gmbh | Protein aus dem Darm von Wirbeltieren, welches Cholesterin absorbiert, sowie Verwendung dieses Proteins zur Identifizierung von Inhibitoren des intestinalen Cholesterintransports |
IL156552A0 (en) * | 2000-12-21 | 2004-01-04 | Aventis Pharma Gmbh | Diphenyl azetidinone derivatives, method for the production thereof, medicaments containing these compounds, and their use |
AU1609702A (en) * | 2000-12-21 | 2002-07-01 | Aventis Pharma Gmbh | Novel 1,2-diphenzylazetidinones, method for producing the same, medicaments containing said compounds, and the use thereof for treating disorders of the lipid metabolism |
PL362512A1 (en) * | 2000-12-21 | 2004-11-02 | Avantis Pharma Deutschland Gmbh | Diphenyl azetidinone derivatives, method for the production thereof, medicaments containing these compounds, and their use |
-
2002
- 2002-06-19 DE DE10227507A patent/DE10227507A1/de not_active Withdrawn
-
2003
- 2003-06-04 DE DE50310161T patent/DE50310161D1/de not_active Expired - Lifetime
- 2003-06-04 AT AT03735534T patent/ATE401304T1/de not_active IP Right Cessation
- 2003-06-04 PT PT03735534T patent/PT1517890E/pt unknown
- 2003-06-04 BR BR0311984-0A patent/BR0311984A/pt not_active IP Right Cessation
- 2003-06-04 MX MXPA04012308A patent/MXPA04012308A/es active IP Right Grant
- 2003-06-04 DK DK03735534T patent/DK1517890T3/da active
- 2003-06-04 JP JP2004514659A patent/JP2005533071A/ja not_active Abandoned
- 2003-06-04 KR KR10-2004-7020518A patent/KR20050010061A/ko not_active Application Discontinuation
- 2003-06-04 PL PL03372660A patent/PL372660A1/xx not_active Application Discontinuation
- 2003-06-04 ES ES03735534T patent/ES2310662T3/es not_active Expired - Lifetime
- 2003-06-04 WO PCT/EP2003/005814 patent/WO2004000803A1/de active IP Right Grant
- 2003-06-04 CN CN038140934A patent/CN1662494A/zh active Pending
- 2003-06-04 CA CA002490108A patent/CA2490108A1/en not_active Abandoned
- 2003-06-04 RS YUP-1086/04A patent/RS108604A/sr unknown
- 2003-06-04 RU RU2005101088/04A patent/RU2315753C2/ru not_active IP Right Cessation
- 2003-06-04 EP EP03735534A patent/EP1517890B1/de not_active Expired - Lifetime
- 2003-06-04 AU AU2003238209A patent/AU2003238209B2/en not_active Ceased
- 2003-06-13 PA PA20038575601A patent/PA8575601A1/es unknown
- 2003-06-16 UY UY27852A patent/UY27852A1/es unknown
- 2003-06-16 SV SV2003001555A patent/SV2004001555A/es unknown
- 2003-06-17 TW TW092116320A patent/TW200406380A/zh unknown
-
2004
- 2004-11-22 ZA ZA200409379A patent/ZA200409379B/xx unknown
- 2004-12-08 MA MA27989A patent/MA27251A1/fr unknown
- 2004-12-15 IL IL165790A patent/IL165790A/en not_active IP Right Cessation
- 2004-12-17 HR HR20041202A patent/HRP20041202A2/xx not_active Application Discontinuation
-
2005
- 2005-01-06 NO NO20050088A patent/NO20050088L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
PT1517890E (pt) | 2008-10-14 |
EP1517890A1 (de) | 2005-03-30 |
KR20050010061A (ko) | 2005-01-26 |
RS108604A (en) | 2007-02-05 |
PA8575601A1 (es) | 2004-02-07 |
CA2490108A1 (en) | 2003-12-31 |
IL165790A (en) | 2010-04-15 |
TW200406380A (en) | 2004-05-01 |
AU2003238209B2 (en) | 2009-01-22 |
DE10227507A1 (de) | 2004-01-08 |
DK1517890T3 (da) | 2008-11-10 |
AU2003238209A1 (en) | 2004-01-06 |
UY27852A1 (es) | 2003-12-31 |
JP2005533071A (ja) | 2005-11-04 |
ATE401304T1 (de) | 2008-08-15 |
RU2005101088A (ru) | 2005-06-27 |
WO2004000803A1 (de) | 2003-12-31 |
SV2004001555A (es) | 2004-03-19 |
EP1517890B1 (de) | 2008-07-16 |
RU2315753C2 (ru) | 2008-01-27 |
ZA200409379B (en) | 2006-05-31 |
MXPA04012308A (es) | 2005-02-25 |
BR0311984A (pt) | 2005-04-26 |
HRP20041202A2 (en) | 2005-06-30 |
IL165790A0 (en) | 2006-01-15 |
CN1662494A (zh) | 2005-08-31 |
ES2310662T3 (es) | 2009-01-16 |
PL372660A1 (en) | 2005-07-25 |
MA27251A1 (fr) | 2005-03-01 |
DE50310161D1 (de) | 2008-08-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |