WO2006105127A8 - Inhibiteurs de l'hydroxysteroide deshydrogenase - Google Patents
Inhibiteurs de l'hydroxysteroide deshydrogenase Download PDFInfo
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- WO2006105127A8 WO2006105127A8 PCT/US2006/011347 US2006011347W WO2006105127A8 WO 2006105127 A8 WO2006105127 A8 WO 2006105127A8 US 2006011347 W US2006011347 W US 2006011347W WO 2006105127 A8 WO2006105127 A8 WO 2006105127A8
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- hydroxysteroid dehydrogenase
- dehydrogenase inhibitors
- inhibitors
- hydroxysteroid
- kits
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- C07D241/38—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
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- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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Abstract
L'invention concerne des composés, des compositions pharmaceutiques, des trousses et des procédés s'utilisant avec des hydroxystéroïde déshydrogénases et qui comprennent un composé sélectionné dans le groupe des composés représentés par la formule (I), les variables de celle-ci étant définies dans le descriptif.
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP06748832A EP1866298A2 (fr) | 2005-03-31 | 2006-03-28 | Inhibiteurs de l'hydroxysteroide deshydrogenase |
JP2008504269A JP5140577B2 (ja) | 2005-03-31 | 2006-03-28 | ヒドロキシステロイドデヒドロゲナーゼ阻害剤 |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US66729705P | 2005-03-31 | 2005-03-31 | |
US60/667,297 | 2005-03-31 |
Publications (3)
Publication Number | Publication Date |
---|---|
WO2006105127A2 WO2006105127A2 (fr) | 2006-10-05 |
WO2006105127A3 WO2006105127A3 (fr) | 2007-03-22 |
WO2006105127A8 true WO2006105127A8 (fr) | 2017-02-09 |
Family
ID=36616791
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2006/011347 WO2006105127A2 (fr) | 2005-03-31 | 2006-03-28 | Inhibiteurs de l'hydroxysteroide deshydrogenase |
Country Status (4)
Country | Link |
---|---|
US (1) | US7759339B2 (fr) |
EP (1) | EP1866298A2 (fr) |
JP (2) | JP5140577B2 (fr) |
WO (1) | WO2006105127A2 (fr) |
Families Citing this family (45)
Publication number | Priority date | Publication date | Assignee | Title |
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TW200630337A (en) | 2004-10-14 | 2006-09-01 | Euro Celtique Sa | Piperidinyl compounds and the use thereof |
JP5140577B2 (ja) * | 2005-03-31 | 2013-02-06 | タケダ カリフォルニア インコーポレイテッド | ヒドロキシステロイドデヒドロゲナーゼ阻害剤 |
EP2527337A1 (fr) * | 2005-04-14 | 2012-11-28 | Bristol-Myers Squibb Company | Inhibiteurs de la 11-bêta hydroxystéroïde déshydrogénase de type I |
BRPI0614974A2 (pt) * | 2005-08-30 | 2010-12-14 | Asahi Kasei Pharma Corp | composto, medicamento, inibidor da fosforilaÇço da cadeia leve regulatària da miosina, inibidor da via rho/rho quinase, e, mÉtodo para tratamento terapÊutico e/ou profilÁtico de glaucoma |
BRPI0616574A2 (pt) | 2005-09-27 | 2009-11-24 | Shionogi & Co | derivado de sulfonamida tendo atividade antagonìstica de receptor de pgd2 |
EP1968962A2 (fr) | 2005-12-14 | 2008-09-17 | Amgen Inc. | Derives diaza heterocycliques de sulfonamide et leurs utilisations |
WO2007092435A2 (fr) * | 2006-02-07 | 2007-08-16 | Wyeth | Inhibiteurs 11-beta hsd1 |
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WO2007110449A1 (fr) * | 2006-03-29 | 2007-10-04 | Euro-Celtique S.A. | Composés de benzènesulfonamide et utilisation de ceux-ci |
US8937181B2 (en) | 2006-04-13 | 2015-01-20 | Purdue Pharma L.P. | Benzenesulfonamide compounds and the use thereof |
WO2007118853A1 (fr) | 2006-04-13 | 2007-10-25 | Euro-Celtique S.A. | Benzènesulfonamides et leur emploi en tant qu'agents bloquants des canaux calcium |
PE20110235A1 (es) | 2006-05-04 | 2011-04-14 | Boehringer Ingelheim Int | Combinaciones farmaceuticas que comprenden linagliptina y metmorfina |
CA2655282A1 (fr) * | 2006-06-16 | 2007-12-21 | High Point Pharmaceuticals, Llc | Utilisation pharmaceutique de carboxamides de piperidine substitues |
TW200811158A (en) * | 2006-06-27 | 2008-03-01 | Sanofi Aventis | Piperidine or pyrrolidine urea derivatives, their preparation and their therapeutic application |
FR2902790A1 (fr) * | 2006-06-27 | 2007-12-28 | Sanofi Aventis Sa | Derives d'urees de piperidine ou pyrrolidine,leur preparation et leur application en therapeutique |
PE20080344A1 (es) | 2006-06-27 | 2008-06-09 | Sanofi Aventis | Compuestos 8-azabiciclo[3.2.1]oct-8-il-1,2,3,4-tetrahidroquinolina sustituidos como inhibidores 11b-hsd1 |
US8415372B2 (en) * | 2007-02-27 | 2013-04-09 | Asahi Kasei Pharma Corporation | Sulfonamide compound |
CN101622243B (zh) * | 2007-02-28 | 2013-12-04 | 旭化成制药株式会社 | 磺酰胺衍生物 |
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US8399486B2 (en) | 2007-04-09 | 2013-03-19 | Purdue Pharma L.P. | Benzenesulfonyl compounds and the use thereof |
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2006
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- 2006-03-28 EP EP06748832A patent/EP1866298A2/fr not_active Withdrawn
- 2006-03-28 WO PCT/US2006/011347 patent/WO2006105127A2/fr active Application Filing
- 2006-03-28 US US11/392,297 patent/US7759339B2/en not_active Expired - Fee Related
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2012
- 2012-08-03 JP JP2012173398A patent/JP2012255004A/ja active Pending
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WO2006105127A3 (fr) | 2007-03-22 |
JP2012255004A (ja) | 2012-12-27 |
JP5140577B2 (ja) | 2013-02-06 |
US20060223829A1 (en) | 2006-10-05 |
US7759339B2 (en) | 2010-07-20 |
JP2008534600A (ja) | 2008-08-28 |
WO2006105127A2 (fr) | 2006-10-05 |
EP1866298A2 (fr) | 2007-12-19 |
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