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CY1117583T1 - Στερεες μορφες περιλαμβανοντας ν-(5-τριτοταγες-βουτυλ-ισοξαζολ-3-υλ)-ν΄-{4-[7-(2-μορφολιν-4-υλ-αιθοξυ)ιμιδαζο[2,1-β][1,3]βενζοθειαζολ-2-υλ]φαινυλ}ουρια,συνθεσεις εξ΄ αυτης, και χρησεις μετ΄ αυτης - Google Patents

Στερεες μορφες περιλαμβανοντας ν-(5-τριτοταγες-βουτυλ-ισοξαζολ-3-υλ)-ν΄-{4-[7-(2-μορφολιν-4-υλ-αιθοξυ)ιμιδαζο[2,1-β][1,3]βενζοθειαζολ-2-υλ]φαινυλ}ουρια,συνθεσεις εξ΄ αυτης, και χρησεις μετ΄ αυτης

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Publication number
CY1117583T1
CY1117583T1 CY20161100450T CY161100450T CY1117583T1 CY 1117583 T1 CY1117583 T1 CY 1117583T1 CY 20161100450 T CY20161100450 T CY 20161100450T CY 161100450 T CY161100450 T CY 161100450T CY 1117583 T1 CY1117583 T1 CY 1117583T1
Authority
CY
Cyprus
Prior art keywords
solid forms
isoxazol
morpholin
imidazo
ethoxy
Prior art date
Application number
CY20161100450T
Other languages
English (en)
Inventor
Shripad Bhagwat
Wei Lai
Stephan D Parent
Melanie J Roe
Alan Schwartz
Valeriya N Smolenskaya
Original Assignee
Ambit Biosciences Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ambit Biosciences Corporation filed Critical Ambit Biosciences Corporation
Publication of CY1117583T1 publication Critical patent/CY1117583T1/el

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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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Abstract

Στερεές μορφές περιλαμβάνοντας Ν-(5-τριτοταγές-βουτυλ-ισοξαζολ-3-υλ)-Ν'-{4-[7-(2-μορφολιν-4-υλ-αιθοξυ)ιμιδαζο[2,1-b][1,3]βενζοθειαζολ-2-υλ]φαινυλ}ουρία, συνθέσεις περιλαμβάνοντας τις στερεές μορφές, μέθοδοι παρασκευής των στερεών μορφών και μέθοδοι της χρήσης αυτών για την αγωγή διαφόρων παθήσεων και/ή διαταραχών αποκαλύπτονται.
CY20161100450T 2007-09-19 2016-05-24 Στερεες μορφες περιλαμβανοντας ν-(5-τριτοταγες-βουτυλ-ισοξαζολ-3-υλ)-ν΄-{4-[7-(2-μορφολιν-4-υλ-αιθοξυ)ιμιδαζο[2,1-β][1,3]βενζοθειαζολ-2-υλ]φαινυλ}ουρια,συνθεσεις εξ΄ αυτης, και χρησεις μετ΄ αυτης CY1117583T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US99463507P 2007-09-19 2007-09-19
EP08832577.4A EP2201018B1 (en) 2007-09-19 2008-09-19 Solid forms comprising n-(5-tert-butyl-isoxazol-3-yl)-n'-{4-ý7-(2-morpholin-4-yl-ethoxy)imidazoý2,1-b¨ý1,3¨benzothiazol-2-yl¨phenyl}urea, compositions thereof, and uses therewith

Publications (1)

Publication Number Publication Date
CY1117583T1 true CY1117583T1 (el) 2017-04-26

Family

ID=40468693

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20161100450T CY1117583T1 (el) 2007-09-19 2016-05-24 Στερεες μορφες περιλαμβανοντας ν-(5-τριτοταγες-βουτυλ-ισοξαζολ-3-υλ)-ν΄-{4-[7-(2-μορφολιν-4-υλ-αιθοξυ)ιμιδαζο[2,1-β][1,3]βενζοθειαζολ-2-υλ]φαινυλ}ουρια,συνθεσεις εξ΄ αυτης, και χρησεις μετ΄ αυτης

Country Status (20)

Country Link
US (2) US8883783B2 (el)
EP (1) EP2201018B1 (el)
JP (1) JP5462168B2 (el)
KR (2) KR20150104231A (el)
CN (1) CN101868465B (el)
AR (1) AR068528A1 (el)
AU (1) AU2008302744B2 (el)
BR (1) BRPI0816904B8 (el)
CA (1) CA2696776C (el)
CY (1) CY1117583T1 (el)
DK (1) DK2201018T3 (el)
ES (1) ES2573292T3 (el)
HR (1) HRP20160520T1 (el)
HU (1) HUE027982T2 (el)
IL (1) IL203926A (el)
MX (1) MX2010002295A (el)
PL (1) PL2201018T3 (el)
SI (1) SI2201018T1 (el)
TW (1) TWI437988B (el)
WO (1) WO2009038757A2 (el)

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