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DE69736711D1 - Substituierte 6,5-heterobicyclische-derivate - Google Patents

Substituierte 6,5-heterobicyclische-derivate

Info

Publication number
DE69736711D1
DE69736711D1 DE69736711T DE69736711T DE69736711D1 DE 69736711 D1 DE69736711 D1 DE 69736711D1 DE 69736711 T DE69736711 T DE 69736711T DE 69736711 T DE69736711 T DE 69736711T DE 69736711 D1 DE69736711 D1 DE 69736711D1
Authority
DE
Germany
Prior art keywords
substituted
heterobicyclic derivatives
heterobicyclic
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69736711T
Other languages
English (en)
Other versions
DE69736711T2 (de
Inventor
Liang Chen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21823717&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE69736711(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc filed Critical Pfizer Inc
Application granted granted Critical
Publication of DE69736711D1 publication Critical patent/DE69736711D1/de
Publication of DE69736711T2 publication Critical patent/DE69736711T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
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    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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    • AHUMAN NECESSITIES
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    • A61P5/42Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of mineralocorticosteroids
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    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Addiction (AREA)
  • Endocrinology (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Communicable Diseases (AREA)
  • Gynecology & Obstetrics (AREA)
  • Hospice & Palliative Care (AREA)
  • Virology (AREA)
  • Dermatology (AREA)
DE69736711T 1996-08-28 1997-07-25 Substituierte 6,5-heterobicyclische-derivate Expired - Fee Related DE69736711T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US2503996P 1996-08-28 1996-08-28
US25039P 1996-08-28
PCT/IB1997/000922 WO1998008847A1 (en) 1996-08-28 1997-07-25 Substituted 6,5-hetero-bicyclic derivatives

Publications (2)

Publication Number Publication Date
DE69736711D1 true DE69736711D1 (de) 2006-11-02
DE69736711T2 DE69736711T2 (de) 2007-09-20

Family

ID=21823717

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69736711T Expired - Fee Related DE69736711T2 (de) 1996-08-28 1997-07-25 Substituierte 6,5-heterobicyclische-derivate

Country Status (36)

Country Link
EP (1) EP0923582B1 (de)
JP (2) JP3621706B2 (de)
KR (1) KR20000035934A (de)
CN (1) CN1227554A (de)
AP (1) AP762A (de)
AR (1) AR015103A1 (de)
AT (1) ATE340176T1 (de)
AU (1) AU735401B2 (de)
BG (1) BG103189A (de)
BR (1) BR9711970A (de)
CA (1) CA2263566C (de)
CO (1) CO4600634A1 (de)
CZ (1) CZ68199A3 (de)
DE (1) DE69736711T2 (de)
DZ (1) DZ2300A1 (de)
EA (1) EA002769B1 (de)
ES (1) ES2273369T3 (de)
GT (1) GT199700095A (de)
HR (1) HRP970454B1 (de)
HU (1) HUP9903965A3 (de)
ID (1) ID18249A (de)
IL (1) IL127566A0 (de)
IS (1) IS4963A (de)
MA (1) MA26438A1 (de)
NO (1) NO313636B1 (de)
NZ (1) NZ333302A (de)
OA (1) OA10977A (de)
PA (1) PA8436201A1 (de)
PE (1) PE108898A1 (de)
PL (1) PL332040A1 (de)
SK (1) SK23399A3 (de)
TN (1) TNSN97145A1 (de)
TR (1) TR199900389T2 (de)
TW (1) TW575573B (de)
WO (1) WO1998008847A1 (de)
ZA (1) ZA977687B (de)

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DE69603240T2 (de) 1995-05-12 2000-01-05 Neurogen Corp., Branford Neue deazapurinderivate; eine neue klasse von crf1-spezifischen liganden
US7094782B1 (en) 1996-07-24 2006-08-22 Bristol-Myers Squibb Company Azolo triazines and pyrimidines
US6060478A (en) * 1996-07-24 2000-05-09 Dupont Pharmaceuticals Azolo triazines and pyrimidines
US6191131B1 (en) 1997-07-23 2001-02-20 Dupont Pharmaceuticals Company Azolo triazines and pyrimidines
US6124289A (en) * 1996-07-24 2000-09-26 Dupont Pharmaceuticals Co. Azolo triazines and pyrimidines
US6313124B1 (en) 1997-07-23 2001-11-06 Dupont Pharmaceuticals Company Tetrazine bicyclic compounds
WO1998035967A2 (en) * 1997-02-18 1998-08-20 Neurocrine Biosciences, Inc. Biazacyclic crf antagonists
NZ335823A (en) * 1997-04-22 2001-06-29 Neurocrine Biosciences Inc Thiophenopyridines, preparation as CRF receptor antagonists
CA2294117A1 (en) 1997-07-03 1999-01-14 Dupont Pharmaceuticals Company Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders
DK1049699T3 (da) * 1998-01-28 2004-07-05 Bristol Myers Squibb Pharma Co Pyrazolotriaziner som CRF-antagonister
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
US6472402B1 (en) 1998-04-02 2002-10-29 Neurogen Corporation Aminoalkyl substituted 5,6,7,8-Tetrahydro-9H-Pyridino [2,3-B]indole derivatives
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