ZA200303794B - Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same. - Google Patents

Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same.

Info

Publication number: ZA200303794B
Authority: ZA; South Africa
Prior art keywords: preparation; compositions containing; containing same; piperidine derivatives; heterocyclylalkyl piperidine
Prior art date: 2000-11-15

Application number

ZA200303794A

Inventor

Eric Bacque

Youssef El-Ahmad

Philippe Hubert

Serge Mignani

Michel Tabart

Jean-Christophe Carry

Michel Evers

Jean-Luc Malleron

Guy Pantel

Fabrice Viviani

Original Assignee

Aventis Pharma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-15

Filing date

2003-05-15

Publication date

2004-06-29

2003-05-15 Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa

2004-06-29 Publication of ZA200303794B publication Critical patent/ZA200303794B/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)

ZA200303794A 2000-11-15 2003-05-15 Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same. ZA200303794B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0014738A FR2816618B1 (en)	2000-11-15	2000-11-15	HETEROCYCLYLALCOYL PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THE COMPOSITIONS CONTAINING THEM

Publications (1)

Publication Number	Publication Date
ZA200303794B true ZA200303794B (en)	2004-06-29

Family

ID=8856503

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200303794A ZA200303794B (en)	2000-11-15	2003-05-15	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same.

Country Status (28)

Country	Link
EP (2)	EP1337529B1 (en)
JP (1)	JP2004514661A (en)
KR (1)	KR100849608B1 (en)
CN (1)	CN1483031A (en)
AR (1)	AR034006A1 (en)
AT (1)	ATE337311T1 (en)
AU (2)	AU2002218365B2 (en)
BG (1)	BG107793A (en)
BR (1)	BR0115312A (en)
CA (1)	CA2429311A1 (en)
CZ (1)	CZ20031316A3 (en)
DE (1)	DE60122567T2 (en)
DK (1)	DK1337529T3 (en)
EA (1)	EA200300568A1 (en)
EE (1)	EE200300207A (en)
ES (1)	ES2271119T3 (en)
FR (1)	FR2816618B1 (en)
HR (1)	HRP20030379A2 (en)
HU (1)	HUP0303758A3 (en)
IL (1)	IL155841A0 (en)
NO (2)	NO20032187L (en)
PL (1)	PL363004A1 (en)
PT (1)	PT1337529E (en)
SK (1)	SK5822003A3 (en)
TN (1)	TNSN01160A1 (en)
WO (1)	WO2002040474A2 (en)
YU (1)	YU46803A (en)
ZA (1)	ZA200303794B (en)

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EP1305308B1 (en)	2000-07-26	2006-12-20	Smithkline Beecham Plc	Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity
GB0101577D0 (en)	2001-01-22	2001-03-07	Smithkline Beecham Plc	Compounds
GB0112836D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0112834D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0118238D0 (en) *	2001-07-26	2001-09-19	Smithkline Beecham Plc	Medicaments
AU2003239302A1 (en)	2002-01-29	2003-09-02	Glaxo Group Limited	Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them
JP4445753B2 (en)	2002-01-29	2010-04-07	グラクソグループリミテッド	Aminopiperidine derivatives
AR040335A1 (en)	2002-06-26	2005-03-30	Glaxo Group Ltd	CYCLLOHEXAN OR CYCLHEXENE COMPOUND, USE OF THE SAME TO PREPARE A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT, PROCEDURE AND INTERMEDIATE COMPOUNDS OF UTILITY TO PREPARE SUCH COMPOUND
AR040336A1 (en)	2002-06-26	2005-03-30	Glaxo Group Ltd	PIPERIDINE COMPOUND, USE OF THE SAME FOR THE MANUFACTURE OF A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND PROCEDURE TO PREPARE SUCH COMPOUND
FR2842807A1 (en) *	2002-07-23	2004-01-30	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESS AND PREPARATION INTERMEDIATES AND COMPOSITIONS COMPRISING THE SAME
GB0217294D0 (en) *	2002-07-25	2002-09-04	Glaxo Group Ltd	Medicaments
FR2844270B1 (en) *	2002-09-11	2006-05-19	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, THEIR PROCESS AND PREPARATION INTERMEDIATES AND THE COMPOSITIONS CONTAINING THEM
FR2844268B1 (en) *	2002-09-11	2004-10-22	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION, AND COMPOSITIONS CONTAINING THEM
DE10256405A1 (en) *	2002-12-02	2004-06-17	Morphochem Aktiengesellschaft für kombinatorische Chemie	New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
EP1560821B8 (en)	2002-11-05	2010-05-19	Glaxo Group Limited	Antibacterial agents
US7491714B2 (en)	2002-12-04	2009-02-17	Glaxo Group Limited	Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
FR2852954B1 (en) *	2003-03-28	2006-07-14	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
US7232833B2 (en)	2003-03-28	2007-06-19	Novexel	4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
FR2862301B1 (en) *	2003-11-17	2007-12-21	Aventis Pharma Sa	NEW PROCESS FOR THE PREPARATION OF 3-FLUORINATED QUINOLINES
FR2867472B1 (en) *	2004-03-12	2008-07-18	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
US7709472B2 (en)	2005-01-25	2010-05-04	Glaxo Group Limited	Antibacterial agents
WO2006081264A1 (en)	2005-01-25	2006-08-03	Glaxo Group Limited	Antibacterial agents
WO2006081178A2 (en)	2005-01-25	2006-08-03	Glaxo Group Limited	Antibacterial agents
US7592334B2 (en)	2005-01-25	2009-09-22	Glaxo Group Limited	Antibacterial agents
JP2008531709A (en)	2005-03-01	2008-08-14	ワイス	Cinnoline compounds and their use as liver X receptor modulators
MY150958A (en)	2005-06-16	2014-03-31	Astrazeneca Ab	Compounds for the treatment of multi-drug resistant bacterial infections
ATE536351T1 (en)	2006-01-26	2011-12-15	Actelion Pharmaceuticals Ltd	TETRAHYDROPYRAN ANTIBIOTICS
ATE481406T1 (en)	2006-04-06	2010-10-15	Glaxo Group Ltd	PYRROLOQUINOXALINONE DERIVATIVES AS ANTIBACTERIAL AGENTS
EP1992628A1 (en)	2007-05-18	2008-11-19	Glaxo Group Limited	Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
US8193179B2 (en)	2007-06-15	2012-06-05	Actelion Pharmaceuticals, Ltd	3-amino-6-(1-amino-ethyl)-tetrahydropyran derivatives
EP2080761A1 (en)	2008-01-18	2009-07-22	Glaxo Group Limited	Compounds
JP2012505866A (en)	2008-10-17	2012-03-08	グラクソグループリミテッド	Tricyclic nitrogen compounds used as antibacterial agents
US8318940B2 (en)	2009-01-15	2012-11-27	Glaxo Group Limited	Naphthyridin-2 (1 H)-one compounds useful as antibacterials
BR112015003101B1 (en) *	2012-08-15	2022-06-14	Glaxo Group Limited	PROCESS FOR PREPARING A COMPOUND
PE20170501A1 (en)	2014-08-22	2017-04-27	Glaxosmithkline Ip Dev Ltd	A PROCEDURE INVOLVING COMPOUNDS ADMINISTERING TO A SUBJECT INFECTED WITH NEISSERIA GONORRHOEAE
WO2016138988A1 (en) *	2015-03-02	2016-09-09	University Of Copenhagen	Piperazine inhibitors of bacterial gyrase and topoisomerase iv
TW201722965A (en)	2015-08-16	2017-07-01	葛蘭素史密斯克藍智慧財產發展有限公司	Compounds for use in antibacterial applications

Family Cites Families (6)

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Publication number	Priority date	Publication date	Assignee	Title
NL7908031A (en)	1979-11-01	1981-06-01	Acf Chemiefarma Nv	NEW QUINOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING SUCH A COMPOUND AND METHOD FOR PREPARING THESE COMPOUNDS.
JPH0239546A (en)	1988-07-29	1990-02-08	Origin Electric Co Ltd	Manufacture of hybrid integrated circuit
NZ232091A (en)	1989-01-16	1990-12-21	Bellon Labor Sa Roger	7-fluoro-8-(piperazin-1-yl)-4-oxo-1,4-dihydro-benzo(b)(1,8)naphthyridine-3-carboxylic acid derivatives, preparation and pharmaceutical compositions thereof
DE69908555T2 (en) *	1998-01-26	2004-05-06	Smithkline Beecham P.L.C., Brentford	CHINOLINE DERIVATIVES AS AN ANTIBACTERIAL MEDICINAL PRODUCT
JP2002535323A (en) *	1999-01-20	2002-10-22	スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー	Piperidinylquinoline as a protein kinase inhibitor
FR2852954B1 (en) *	2003-03-28	2006-07-14	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

2000
- 2000-11-15 FR FR0014738A patent/FR2816618B1/en not_active Expired - Fee Related
2001
- 2001-11-13 AR ARP010105289A patent/AR034006A1/en unknown
- 2001-11-14 BR BR0115312-9A patent/BR0115312A/en not_active Application Discontinuation
- 2001-11-14 CN CNA018210996A patent/CN1483031A/en active Pending
- 2001-11-14 EE EEP200300207A patent/EE200300207A/en unknown
- 2001-11-14 JP JP2002543484A patent/JP2004514661A/en active Pending
- 2001-11-14 KR KR1020037006600A patent/KR100849608B1/en not_active IP Right Cessation
- 2001-11-14 PT PT01996538T patent/PT1337529E/en unknown
- 2001-11-14 DE DE60122567T patent/DE60122567T2/en not_active Expired - Fee Related
- 2001-11-14 EP EP01996538A patent/EP1337529B1/en not_active Expired - Lifetime
- 2001-11-14 ES ES01996538T patent/ES2271119T3/en not_active Expired - Lifetime
- 2001-11-14 HU HU0303758A patent/HUP0303758A3/en unknown
- 2001-11-14 IL IL15584101A patent/IL155841A0/en unknown
- 2001-11-14 AU AU2002218365A patent/AU2002218365B2/en not_active Ceased
- 2001-11-14 YU YU46803A patent/YU46803A/en unknown
- 2001-11-14 PL PL01363004A patent/PL363004A1/en not_active Application Discontinuation
- 2001-11-14 SK SK582-2003A patent/SK5822003A3/en unknown
- 2001-11-14 CZ CZ20031316A patent/CZ20031316A3/en unknown
- 2001-11-14 AU AU1836502A patent/AU1836502A/en active Pending
- 2001-11-14 CA CA002429311A patent/CA2429311A1/en not_active Abandoned
- 2001-11-14 AT AT01996538T patent/ATE337311T1/en not_active IP Right Cessation
- 2001-11-14 TN TNTNSN01160A patent/TNSN01160A1/en unknown
- 2001-11-14 EP EP06010725A patent/EP1695964A1/en not_active Withdrawn
- 2001-11-14 EA EA200300568A patent/EA200300568A1/en unknown
- 2001-11-14 DK DK01996538T patent/DK1337529T3/en active
- 2001-11-14 WO PCT/FR2001/003559 patent/WO2002040474A2/en active IP Right Grant
2003
- 2003-05-09 BG BG107793A patent/BG107793A/en unknown
- 2003-05-13 HR HR20030379A patent/HRP20030379A2/en not_active Application Discontinuation
- 2003-05-14 NO NO20032187A patent/NO20032187L/en unknown
- 2003-05-15 ZA ZA200303794A patent/ZA200303794B/en unknown
2007
- 2007-04-25 NO NO20072142A patent/NO20072142L/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
NO20032187L (en)	2003-06-26
ATE337311T1 (en)	2006-09-15
YU46803A (en)	2006-05-25
HRP20030379A2 (en)	2005-04-30
EP1337529B1 (en)	2006-08-23
AU1836502A (en)	2002-05-27
EP1695964A1 (en)	2006-08-30
BR0115312A (en)	2003-09-23
HUP0303758A2 (en)	2004-03-01
KR20030060934A (en)	2003-07-16
EP1337529A2 (en)	2003-08-27
WO2002040474A2 (en)	2002-05-23
CN1483031A (en)	2004-03-17
DE60122567D1 (en)	2006-10-05
AU2002218365B2 (en)	2007-07-05
FR2816618A1 (en)	2002-05-17
FR2816618B1 (en)	2002-12-27
DK1337529T3 (en)	2006-12-18
IL155841A0 (en)	2003-12-23
EE200300207A (en)	2003-08-15
SK5822003A3 (en)	2004-06-08
NO20072142L (en)	2007-04-25
ES2271119T3 (en)	2007-04-16
HUP0303758A3 (en)	2009-08-28
CA2429311A1 (en)	2002-05-23
BG107793A (en)	2004-08-31
JP2004514661A (en)	2004-05-20
WO2002040474A3 (en)	2002-10-31
KR100849608B1 (en)	2008-07-31
DE60122567T2 (en)	2007-08-23
CZ20031316A3 (en)	2003-10-15
PL363004A1 (en)	2004-11-15
EA200300568A1 (en)	2003-12-25
AR034006A1 (en)	2004-01-21
PT1337529E (en)	2006-12-29
NO20032187D0 (en)	2003-05-14
TNSN01160A1 (en)	2005-11-10

Publication	Publication Date	Title
ZA200303794B (en)	2004-06-29	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same.
ZA200206905B (en)	2003-08-26	Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same.
IL151209A0 (en)	2003-04-10	Pharmaceutical compositions containing 3-aminoazetidine derivatives, novel derivatives and their preparation
HUP0303835A3 (en)	2009-08-28	Anti-allergic piperidine compounds, their use and pharmaceutical compositions containing them
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HUP0204514A3 (en)	2004-07-28	Pyridinylimidazoles, pharmaceutical compositions containing them and their use
AU2001237526A1 (en)	2001-11-22	Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
MXPA03000771A (en)	2003-06-04	New pharmaceutical composition.
AU2001237525A1 (en)	2001-11-22	Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same
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AU2002253219A1 (en)	2003-03-20	Quinolyl propyl piperidine derivatives, the preparation thereof and compositions containing same
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