DK1337529T3 - Heterocyclylalkylpiperidine derivatives, their preparation and preparations containing them - Google Patents

Heterocyclylalkylpiperidine derivatives, their preparation and preparations containing them

Info

Publication number: DK1337529T3
Authority: DK; Denmark
Prior art keywords: preparation; preparations containing; heterocyclylalkylpiperidine derivatives; heterocyclylalkylpiperidine; derivatives
Prior art date: 2000-11-15

Application number

DK01996538T

Other languages

Danish (da)

Inventor

Philippe Hubert

Eric Bacqu

Jean-Christophe Carry

Youssef El-Ahmad

Michel Evers

Jean-Luc Malleron

Serge Mignani

Guy Pantel

Michel Tabart

Fabrice Viviani

Original Assignee

Novexel

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-15

Filing date

2001-11-14

Publication date

2006-12-18

2001-11-14 Application filed by Novexel filed Critical Novexel

2006-12-18 Application granted granted Critical

2006-12-18 Publication of DK1337529T3 publication Critical patent/DK1337529T3/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)

DK01996538T 2000-11-15 2001-11-14 Heterocyclylalkylpiperidine derivatives, their preparation and preparations containing them DK1337529T3 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0014738A FR2816618B1 (en)	2000-11-15	2000-11-15	HETEROCYCLYLALCOYL PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THE COMPOSITIONS CONTAINING THEM

Publications (1)

Publication Number	Publication Date
DK1337529T3 true DK1337529T3 (en)	2006-12-18

Family

ID=8856503

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK01996538T DK1337529T3 (en)	2000-11-15	2001-11-14	Heterocyclylalkylpiperidine derivatives, their preparation and preparations containing them

Country Status (28)

Country	Link
EP (2)	EP1337529B1 (en)
JP (1)	JP2004514661A (en)
KR (1)	KR100849608B1 (en)
CN (1)	CN1483031A (en)
AR (1)	AR034006A1 (en)
AT (1)	ATE337311T1 (en)
AU (2)	AU2002218365B2 (en)
BG (1)	BG107793A (en)
BR (1)	BR0115312A (en)
CA (1)	CA2429311A1 (en)
CZ (1)	CZ20031316A3 (en)
DE (1)	DE60122567T2 (en)
DK (1)	DK1337529T3 (en)
EA (1)	EA200300568A1 (en)
EE (1)	EE200300207A (en)
ES (1)	ES2271119T3 (en)
FR (1)	FR2816618B1 (en)
HR (1)	HRP20030379A2 (en)
HU (1)	HUP0303758A3 (en)
IL (1)	IL155841A0 (en)
NO (2)	NO20032187L (en)
PL (1)	PL363004A1 (en)
PT (1)	PT1337529E (en)
SK (1)	SK5822003A3 (en)
TN (1)	TNSN01160A1 (en)
WO (1)	WO2002040474A2 (en)
YU (1)	YU46803A (en)
ZA (1)	ZA200303794B (en)

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NZ523749A (en)	2000-07-26	2005-03-24	Smithkline Beecham P	Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity
GB0101577D0 (en)	2001-01-22	2001-03-07	Smithkline Beecham Plc	Compounds
GB0112836D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0112834D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0118238D0 (en) *	2001-07-26	2001-09-19	Smithkline Beecham Plc	Medicaments
EP1470131A2 (en)	2002-01-29	2004-10-27	Glaxo Group Limited	Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them
AR038240A1 (en)	2002-01-29	2005-01-05	Glaxo Group Ltd	PIPERIDINE COMPOUND, USE OF THE SAME FOR THE MANUFACTURE OF A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND PROCEDURE FOR PREPARATION
AR040335A1 (en)	2002-06-26	2005-03-30	Glaxo Group Ltd	CYCLLOHEXAN OR CYCLHEXENE COMPOUND, USE OF THE SAME TO PREPARE A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT, PROCEDURE AND INTERMEDIATE COMPOUNDS OF UTILITY TO PREPARE SUCH COMPOUND
TW200409637A (en)	2002-06-26	2004-06-16	Glaxo Group Ltd	Compounds
FR2842807A1 (en) *	2002-07-23	2004-01-30	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESS AND PREPARATION INTERMEDIATES AND COMPOSITIONS COMPRISING THE SAME
GB0217294D0 (en) *	2002-07-25	2002-09-04	Glaxo Group Ltd	Medicaments
FR2844270B1 (en) *	2002-09-11	2006-05-19	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, THEIR PROCESS AND PREPARATION INTERMEDIATES AND THE COMPOSITIONS CONTAINING THEM
FR2844268B1 (en)	2002-09-11	2004-10-22	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION, AND COMPOSITIONS CONTAINING THEM
DE10256405A1 (en) *	2002-12-02	2004-06-17	Morphochem Aktiengesellschaft für kombinatorische Chemie	New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
ATE461928T1 (en)	2002-11-05	2010-04-15	Glaxosmithkline Llc	ANTIBACTERIAL ACTIVE INGREDIENTS
EP1567520B1 (en)	2002-12-04	2008-10-15	Glaxo Group Limited	Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
FR2852954B1 (en) *	2003-03-28	2006-07-14	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
US7232833B2 (en)	2003-03-28	2007-06-19	Novexel	4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
FR2862301B1 (en) *	2003-11-17	2007-12-21	Aventis Pharma Sa	NEW PROCESS FOR THE PREPARATION OF 3-FLUORINATED QUINOLINES
FR2867472B1 (en) *	2004-03-12	2008-07-18	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
EP1846418A4 (en)	2005-01-25	2009-12-23	Glaxo Group Ltd	Antibacterial agents
JP2008528586A (en)	2005-01-25	2008-07-31	グラクソグループリミテッド	Antibacterial agent
JP2008528598A (en)	2005-01-25	2008-07-31	グラクソグループリミテッド	Antibacterial agent
US7709472B2 (en)	2005-01-25	2010-05-04	Glaxo Group Limited	Antibacterial agents
RU2007131400A (en)	2005-03-01	2009-04-10	Вайет (Us)	COMPOUNDS OF CINNOLINE AND THEIR APPLICATION AS MODULATORS OF LIVER X-RECEPTORS
MY150958A (en) *	2005-06-16	2014-03-31	Astrazeneca Ab	Compounds for the treatment of multi-drug resistant bacterial infections
EP1981881B1 (en)	2006-01-26	2011-12-07	Actelion Pharmaceuticals Ltd.	Tetrahydropyrane antibiotics
ATE481406T1 (en)	2006-04-06	2010-10-15	Glaxo Group Ltd	PYRROLOQUINOXALINONE DERIVATIVES AS ANTIBACTERIAL AGENTS
EP1992628A1 (en)	2007-05-18	2008-11-19	Glaxo Group Limited	Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
AU2008263397B2 (en)	2007-06-15	2013-12-05	Idorsia Pharmaceuticals Ltd	3-amino-6-(1-amino-ethyl)-tetrahydropyran derivatives
EP2080761A1 (en)	2008-01-18	2009-07-22	Glaxo Group Limited	Compounds
WO2010043714A1 (en)	2008-10-17	2010-04-22	Glaxo Group Limited	Tricyclic nitrogen compounds used as antibacterials
ES2561631T3 (en)	2009-01-15	2016-02-29	Glaxo Group Limited	Naphthyridine-2 (1H) -one compounds useful as antibacterial agents
CA2881935A1 (en) *	2012-08-15	2014-02-20	Glaxo Group Limited	Process for preparing a 1-(2-haolethyl)-4-piperidine carboxylate intermediate useful in the synthesis of umeclidinium bromide
EP3639824A1 (en)	2014-08-22	2020-04-22	GlaxoSmithKline Intellectual Property Development Limited	Tricyclic nitrogen containing compounds for treating neisseria gonorrhoea infection
WO2016138988A1 (en) *	2015-03-02	2016-09-09	University Of Copenhagen	Piperazine inhibitors of bacterial gyrase and topoisomerase iv
TW201722965A (en)	2015-08-16	2017-07-01	葛蘭素史密斯克藍智慧財產發展有限公司	Compounds for use in antibacterial applications

Family Cites Families (6)

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Publication number	Priority date	Publication date	Assignee	Title
NL7908031A (en)	1979-11-01	1981-06-01	Acf Chemiefarma Nv	NEW QUINOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING SUCH A COMPOUND AND METHOD FOR PREPARING THESE COMPOUNDS.
JPH0239546A (en)	1988-07-29	1990-02-08	Origin Electric Co Ltd	Manufacture of hybrid integrated circuit
NZ232091A (en)	1989-01-16	1990-12-21	Bellon Labor Sa Roger	7-fluoro-8-(piperazin-1-yl)-4-oxo-1,4-dihydro-benzo(b)(1,8)naphthyridine-3-carboxylic acid derivatives, preparation and pharmaceutical compositions thereof
EP1051413B1 (en) *	1998-01-26	2003-06-04	SmithKline Beecham plc	Quinoline derivatives as antibacterials
WO2000043383A1 (en) *	1999-01-20	2000-07-27	Smithkline Beecham P.L.C.	Piperidinylquinolines as protein tyrosine kinase inhibitors
FR2852954B1 (en) *	2003-03-28	2006-07-14	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

2000
- 2000-11-15 FR FR0014738A patent/FR2816618B1/en not_active Expired - Fee Related
2001
- 2001-11-13 AR ARP010105289A patent/AR034006A1/en unknown
- 2001-11-14 WO PCT/FR2001/003559 patent/WO2002040474A2/en active IP Right Grant
- 2001-11-14 JP JP2002543484A patent/JP2004514661A/en active Pending
- 2001-11-14 TN TNTNSN01160A patent/TNSN01160A1/en unknown
- 2001-11-14 HU HU0303758A patent/HUP0303758A3/en unknown
- 2001-11-14 AT AT01996538T patent/ATE337311T1/en not_active IP Right Cessation
- 2001-11-14 DE DE60122567T patent/DE60122567T2/en not_active Expired - Fee Related
- 2001-11-14 BR BR0115312-9A patent/BR0115312A/en not_active Application Discontinuation
- 2001-11-14 YU YU46803A patent/YU46803A/en unknown
- 2001-11-14 PL PL01363004A patent/PL363004A1/en not_active Application Discontinuation
- 2001-11-14 AU AU2002218365A patent/AU2002218365B2/en not_active Ceased
- 2001-11-14 PT PT01996538T patent/PT1337529E/en unknown
- 2001-11-14 DK DK01996538T patent/DK1337529T3/en active
- 2001-11-14 KR KR1020037006600A patent/KR100849608B1/en not_active IP Right Cessation
- 2001-11-14 CZ CZ20031316A patent/CZ20031316A3/en unknown
- 2001-11-14 AU AU1836502A patent/AU1836502A/en active Pending
- 2001-11-14 CN CNA018210996A patent/CN1483031A/en active Pending
- 2001-11-14 CA CA002429311A patent/CA2429311A1/en not_active Abandoned
- 2001-11-14 EP EP01996538A patent/EP1337529B1/en not_active Expired - Lifetime
- 2001-11-14 IL IL15584101A patent/IL155841A0/en unknown
- 2001-11-14 EA EA200300568A patent/EA200300568A1/en unknown
- 2001-11-14 EE EEP200300207A patent/EE200300207A/en unknown
- 2001-11-14 SK SK582-2003A patent/SK5822003A3/en unknown
- 2001-11-14 EP EP06010725A patent/EP1695964A1/en not_active Withdrawn
- 2001-11-14 ES ES01996538T patent/ES2271119T3/en not_active Expired - Lifetime
2003
- 2003-05-09 BG BG107793A patent/BG107793A/en unknown
- 2003-05-13 HR HR20030379A patent/HRP20030379A2/en not_active Application Discontinuation
- 2003-05-14 NO NO20032187A patent/NO20032187L/en unknown
- 2003-05-15 ZA ZA200303794A patent/ZA200303794B/en unknown
2007
- 2007-04-25 NO NO20072142A patent/NO20072142L/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
CA2429311A1 (en)	2002-05-23
CZ20031316A3 (en)	2003-10-15
NO20032187D0 (en)	2003-05-14
SK5822003A3 (en)	2004-06-08
EP1695964A1 (en)	2006-08-30
DE60122567D1 (en)	2006-10-05
DE60122567T2 (en)	2007-08-23
EP1337529B1 (en)	2006-08-23
ZA200303794B (en)	2004-06-29
HUP0303758A3 (en)	2009-08-28
FR2816618A1 (en)	2002-05-17
KR20030060934A (en)	2003-07-16
JP2004514661A (en)	2004-05-20
EP1337529A2 (en)	2003-08-27
WO2002040474A2 (en)	2002-05-23
FR2816618B1 (en)	2002-12-27
ATE337311T1 (en)	2006-09-15
BR0115312A (en)	2003-09-23
PT1337529E (en)	2006-12-29
IL155841A0 (en)	2003-12-23
ES2271119T3 (en)	2007-04-16
AU2002218365B2 (en)	2007-07-05
AR034006A1 (en)	2004-01-21
NO20032187L (en)	2003-06-26
YU46803A (en)	2006-05-25
NO20072142L (en)	2007-04-25
EE200300207A (en)	2003-08-15
HRP20030379A2 (en)	2005-04-30
WO2002040474A3 (en)	2002-10-31
EA200300568A1 (en)	2003-12-25
AU1836502A (en)	2002-05-27
HUP0303758A2 (en)	2004-03-01
BG107793A (en)	2004-08-31
CN1483031A (en)	2004-03-17
PL363004A1 (en)	2004-11-15
KR100849608B1 (en)	2008-07-31
TNSN01160A1 (en)	2005-11-10

Publication	Publication Date	Title
DK1337529T3 (en)	2006-12-18	Heterocyclylalkylpiperidine derivatives, their preparation and preparations containing them
DK1370550T3 (en)	2007-09-03	Quinolylpropylpiperidine derivatives, their preparation and preparations containing them
NO20024175D0 (en)	2002-09-02	Acetidine derivatives, their preparation and pharmaceutical compounds containing the same
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NO20014603D0 (en)	2001-09-21	Tienopyrimidine Compounds, Their Preparation and Use
DK1112251T3 (en)	2003-09-01	Acetidine derivatives, their preparation and drugs containing these derivatives
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