AU2001237526A1 - Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof - Google Patents

Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof

Info

Publication number: AU2001237526A1
Authority: AU; Australia
Prior art keywords: derivatives; amino; preparation; pharmaceutical compositions; compositions containing
Prior art date: 2000-03-03
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2001237526A

Other versions

AU2001237526B2 (en

Inventor

Daniel Achard

Herve Bouchard

Jean Bouquerel

Bruno Filoche

Serge Grisoni

Augustin Hittinger

Michael Myers

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Aventis Pharma SA

Original Assignee

Aventis Pharma SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-03-03

Filing date

2001-03-01

Publication date

2001-11-22

2000-03-03 Priority claimed from FR0002777A external-priority patent/FR2805810B1/en

2001-03-01 Application filed by Aventis Pharma SA filed Critical Aventis Pharma SA

2001-11-22 Publication of AU2001237526A1 publication Critical patent/AU2001237526A1/en

2006-01-05 Application granted granted Critical

2006-01-05 Publication of AU2001237526B2 publication Critical patent/AU2001237526B2/en

2021-03-01 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
FR0002777		2000-03-03
FR0002777A FR2805810B1 (en)	2000-03-03	2000-03-03	PHARMACEUTICAL COMPOSITIONS CONTAINING 3- AMINO-AZETIDINE DERIVATIVES, THE NEW DERIVATIVES AND THEIR PREPARATION
PCT/FR2001/000601 WO2001064633A1 (en)	2000-03-03	2001-03-01	Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof

Publications (2)

Publication Number	Publication Date
AU2001237526A1 true AU2001237526A1 (en)	2001-11-22
AU2001237526B2 AU2001237526B2 (en)	2006-01-05

Family

ID=8847707

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AU3752601A Pending AU3752601A (en)	2000-03-03	2001-03-01	Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
AU2001237526A Ceased AU2001237526B2 (en)	2000-03-03	2001-03-01	Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
AU3752601A Pending AU3752601A (en)	2000-03-03	2001-03-01	Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof

Country Status (35)

Country	Link
EP (1)	EP1263721B1 (en)
JP (1)	JP2003525269A (en)
KR (1)	KR100813740B1 (en)
CN (1)	CN1187325C (en)
AR (1)	AR034405A1 (en)
AT (1)	ATE478840T1 (en)
AU (2)	AU3752601A (en)
BG (1)	BG107057A (en)
BR (1)	BR0108894A (en)
CA (1)	CA2400138A1 (en)
CY (1)	CY1111075T1 (en)
DE (1)	DE60142890D1 (en)
DK (1)	DK1263721T3 (en)
DZ (1)	DZ3311A1 (en)
EA (1)	EA004649B1 (en)
EE (1)	EE05081B1 (en)
ES (1)	ES2351183T3 (en)
FR (1)	FR2805810B1 (en)
HR (1)	HRP20020710A2 (en)
HU (1)	HUP0300350A2 (en)
IL (2)	IL151209A0 (en)
MA (1)	MA26879A1 (en)
MX (1)	MXPA02008346A (en)
NO (1)	NO324523B1 (en)
NZ (1)	NZ521076A (en)
OA (1)	OA12221A (en)
PL (1)	PL365007A1 (en)
PT (1)	PT1263721E (en)
SI (1)	SI1263721T1 (en)
SK (1)	SK12442002A3 (en)
TW (1)	TWI294420B (en)
UA (1)	UA72319C2 (en)
WO (1)	WO2001064633A1 (en)
YU (1)	YU65902A (en)
ZA (1)	ZA200206916B (en)

Families Citing this family (85)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU2001288972A1 (en)	2000-09-11	2002-03-26	Sepracor, Inc.	Antipsychotic sulfonamide-heterocycles, and methods of use thereof
FR2814678B1 (en) *	2000-10-04	2002-12-20	Aventis Pharma Sa	COMBINATION OF AN ANTAGONIST OF THE CB1 RECEPTOR AND SIBUTRAMINE, THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE FOR THE TREATMENT OF OBESITY
WO2003007887A2 (en)	2001-07-20	2003-01-30	Merck & Co., Inc.	Substituted imidazoles as cannabinoid receptor modulators
FR2833842B1 (en) *	2001-12-21	2004-02-13	Aventis Pharma Sa	PHARMACEUTICAL COMPOSITIONS BASED ON AZETIDINE DERIVATIVES
EP1487436A4 (en)	2002-03-08	2009-06-03	Signal Pharm Inc	Combination therapy for treating, preventing or managing proliferative disorders and cancers
CA2478183C (en)	2002-03-12	2010-02-16	Merck & Co. Inc.	Substituted amides
FR2837706A1 (en) *	2002-03-28	2003-10-03	Sanofi Synthelabo	USE OF A CB1 CANNABINOID RECEPTOR ANTAGONIST FOR THE PREPARATION OF MEDICINES USEFUL FOR THE TREATMENT OF SEXUAL DYSFUNCTION AND / OR IMPROVING SEXUAL PERFORMANCE
US7105526B2 (en)	2002-06-28	2006-09-12	Banyu Pharmaceuticals Co., Ltd.	Benzimidazole derivatives
EP1532132B1 (en)	2002-07-29	2008-03-19	F.Hoffmann-La Roche Ag	Novel benzodioxoles
BR0317926A (en)	2003-01-02	2005-11-29	Hoffmann La Roche	Compounds, process for their manufacture, pharmaceutical compositions comprising them, method for the treatment and / or prophylaxis of diseases that are associated with modulation of cb1 receptors and their use
CN100360527C (en)	2003-01-02	2008-01-09	霍夫曼-拉罗奇有限公司	CB 1 receptor inverse agonists
US7772188B2 (en)	2003-01-28	2010-08-10	Ironwood Pharmaceuticals, Inc.	Methods and compositions for the treatment of gastrointestinal disorders
CN1780615A (en) *	2003-05-01	2006-05-31	弗奈利斯研究有限公司	Use of azetidinecarboxamide derivatives in therapy
MXPA05013583A (en)	2003-06-11	2006-03-09	Merck & Co Inc	Substituted 3-alkyl and 3-alkenyl azetidine derivatives.
JP2007506654A (en)	2003-06-20	2007-03-22	エフ．ホフマン−ラ　ロシュ　アーゲー	2-Aminobenzothiazoles as CB1 receptor inverse agonists
JP4765627B2 (en)	2003-09-22	2011-09-07	Ｍｓｄ株式会社	Novel piperidine derivatives
AU2004299198A1 (en)	2003-12-08	2005-06-30	F. Hoffmann-La Roche Ag	Novel thiazole derivates
BRPI0507120A (en)	2004-01-28	2007-06-19	Hoffmann La Roche	compounds, process for the manufacture thereof, pharmaceutical compositions comprising them, method for treating and / or prophylaxis of diseases that are associated with cb1 receptor modulation and their use
RU2006133258A (en) *	2004-02-17	2008-04-10	Лабораториос Дель Др. Эстеве С.А. (Es)	SUBSTITUTED AZETIDINE DERIVATIVES, THEIR PRODUCTION AND APPLICATION AS MEDICINES
EP1574211A1 (en)	2004-03-09	2005-09-14	Inserm	Use of antagonists of the CB1 receptor for the manufacture of a composition useful for the treatment of hepatic diseases
EP1734963A4 (en)	2004-04-02	2008-06-18	Merck & Co Inc	Method of treating men with metabolic and anthropometric disorders
CA2564986A1 (en)	2004-05-10	2005-11-17	F. Hoffmann-La Roche Ag	Pyrrole or imidazole amides for treating obesity
JP2008517959A (en)	2004-10-27	2008-05-29	エフ．ホフマン−ラロシュアーゲー	Novel indole or benzimidazole derivatives
KR100896353B1 (en)	2004-11-09	2009-05-08	에프. 호프만-라 로슈 아게	Dibenzosuberone derivatives
DE602006007563D1 (en)	2005-04-06	2009-08-13	Hoffmann La Roche	AGONIST
EP1892241B1 (en)	2005-05-30	2016-03-30	Msd K.K.	Novel piperidine derivative
WO2006129178A1 (en)	2005-06-02	2006-12-07	Glenmark Pharmaceuticals S.A.	Novel cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation
US7923465B2 (en)	2005-06-02	2011-04-12	Glenmark Pharmaceuticals S.A.	Cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation
EP1916239A4 (en)	2005-08-10	2009-10-21	Banyu Pharma Co Ltd	Pyridone compound
KR101440409B1 (en) *	2005-08-18	2014-09-15	닛산 가가쿠 고교 가부시키 가이샤	Thiophene compound having sulfonyl group and process for producing the same
JPWO2007024004A1 (en)	2005-08-24	2009-03-05	萬有製薬株式会社	Phenylpyridone derivatives
US20090264426A1 (en)	2005-09-07	2009-10-22	Shunji Sakuraba	Bicyclic aromatic substituted pyridone derivative
CN101277960A (en)	2005-09-29	2008-10-01	默克公司	Acylated spiropiperidine derivatives as melanocortin-4 receptor modulators
AU2006307046A1 (en)	2005-10-27	2007-05-03	Msd K.K.	Novel benzoxathiin derivative
RU2428423C2 (en)	2005-11-10	2011-09-10	Баниу Фармасьютикал Ко., Лтд.	Aza-substituted spiro-derivatives
AR058199A1 (en) *	2005-11-28	2008-01-23	Merck & Co Inc	DERIVATIVES OF 3- RENTED ALQUILAZETIDINA WITH HETEROCICLOS
US7906652B2 (en)	2005-11-28	2011-03-15	Merck Sharp & Dohme Corp.	Heterocycle-substituted 3-alkyl azetidine derivatives
US7629346B2 (en)	2006-06-19	2009-12-08	Hoffmann-La Roche Inc.	Pyrazinecarboxamide derivatives as CB1 antagonists
CA2666193A1 (en)	2006-08-08	2008-02-14	Sanofi-Aventis	Arylaminoaryl-alkyl-substituted imidazolidine-2,4-diones, process for preparing them, medicaments comprising these compounds, and their use
US7781593B2 (en)	2006-09-14	2010-08-24	Hoffmann-La Roche Inc.	5-phenyl-nicotinamide derivatives
EP2083831B1 (en)	2006-09-22	2013-12-25	Merck Sharp & Dohme Corp.	Method of treatment using fatty acid synthesis inhibitors
AU2007301126A1 (en)	2006-09-28	2008-04-03	Banyu Pharmaceutical Co., Ltd.	Diaryl ketimine derivative
WO2008120653A1 (en)	2007-04-02	2008-10-09	Banyu Pharmaceutical Co., Ltd.	Indoledione derivative
ES2559319T3 (en)	2007-06-04	2016-02-11	Synergy Pharmaceuticals Inc.	Guanylate cliclas agonists useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
US8969514B2 (en)	2007-06-04	2015-03-03	Synergy Pharmaceuticals, Inc.	Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
EP2264026A4 (en)	2008-03-06	2012-03-28	Msd Kk	Alkylaminopyridine derivative
CA2717384A1 (en)	2008-03-28	2009-10-01	Banyu Pharmaceutical Co., Ltd.	Diarylmethylamide derivative having melanin-concentrating hormone receptor antagonism
JP2011522828A (en)	2008-06-04	2011-08-04	シナジーファーマシューティカルズインコーポレイテッド	Guanylate cyclase agonists useful for the treatment of gastrointestinal disorders, inflammation, cancer, and other disorders
US20110071129A1 (en)	2008-06-19	2011-03-24	Makoto Ando	Spirodiamine-diaryl ketoxime derivative
WO2010009319A2 (en)	2008-07-16	2010-01-21	Synergy Pharmaceuticals Inc.	Agonists of guanylate cyclase useful for the treatment of gastrointestinal, inflammation, cancer and other disorders
CA2731358A1 (en)	2008-07-30	2010-02-04	Banyu Pharmaceutical Co., Ltd.	5/5-or 5/6-membered condensed ring cycloalkylamine derivative
CA2741125A1 (en)	2008-10-22	2010-04-29	Merck Sharp & Dohme Corp.	Novel cyclic benzimidazole derivatives useful anti-diabetic agents
AU2009308980B2 (en)	2008-10-30	2013-02-28	Merck Sharp & Dohme Corp.	Isonicotinamide orexin receptor antagonists
JP5557845B2 (en)	2008-10-31	2014-07-23	メルク・シャープ・アンド・ドーム・コーポレーション	Novel cyclic benzimidazole derivatives useful as antidiabetic agents
US8759539B2 (en)	2008-11-17	2014-06-24	Merck Sharp & Dohme Corp.	Substituted bicyclic amines for the treatment of diabetes
WO2011011506A1 (en)	2009-07-23	2011-01-27	Schering Corporation	Spirocyclic oxazepine compounds as stearoyl-coenzyme a delta-9 desaturase inhibitors
US20120220567A1 (en)	2009-07-23	2012-08-30	Shipps Jr Gerald W	Benzo-fused oxazepine compounds as stearoyl-coenzyme a delta-9 desaturase inhibitors
AU2011218830B2 (en)	2010-02-25	2014-07-24	Merck Sharp & Dohme Corp.	Novel cyclic benzimidazole derivatives useful anti-diabetic agents
EP2563764B1 (en)	2010-04-26	2015-02-25	Merck Sharp & Dohme Corp.	Novel spiropiperidine prolylcarboxypeptidase inhibitors
WO2011143057A1 (en)	2010-05-11	2011-11-17	Merck Sharp & Dohme Corp.	Novel prolylcarboxypeptidase inhibitors
WO2011156246A1 (en)	2010-06-11	2011-12-15	Merck Sharp & Dohme Corp.	Novel prolylcarboxypeptidase inhibitors
US9616097B2 (en)	2010-09-15	2017-04-11	Synergy Pharmaceuticals, Inc.	Formulations of guanylate cyclase C agonists and methods of use
US8410107B2 (en)	2010-10-15	2013-04-02	Hoffmann-La Roche Inc.	N-pyridin-3-yl or N-pyrazin-2-yl carboxamides
JP2013540160A (en) *	2010-10-22	2013-10-31	ヤンセンファーマシューティカエヌ．ベー．	Amino-pyrrolidine-azetidine diamide as monoacylglycerol lipase inhibitor
US8669254B2 (en)	2010-12-15	2014-03-11	Hoffman-La Roche Inc.	Pyridine, pyridazine, pyrimidine or pyrazine carboxamides as HDL-cholesterol raising agents
EA201690035A1 (en)	2011-02-25	2016-05-31	Мерк Шарп Энд Домэ Корп.	NEW CYCLIC DERIVATIVES OF AZABENZIMIDAZOLE, USED AS ANTI-DIABETIC AGENTS
WO2012120051A1 (en)	2011-03-08	2012-09-13	Sanofi	Benzyl-oxathiazine derivates substituted with adamantane or noradamantane, medicaments containing said compounds and use thereof
EP2683703B1 (en)	2011-03-08	2015-05-27	Sanofi	Novel substituted phenyl-oxathiazine derivatives, method for producing them, drugs containing said compounds and the use thereof
WO2012120050A1 (en)	2011-03-08	2012-09-13	Sanofi	Novel substituted phenyl-oxathiazine derivatives, method for producing them, drugs containing said compounds and the use thereof
US8846666B2 (en)	2011-03-08	2014-09-30	Sanofi	Oxathiazine derivatives which are substituted with benzyl or heteromethylene groups, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
AR088352A1 (en)	2011-10-19	2014-05-28	Merck Sharp & Dohme	ANTAGONISTS OF THE RECEIVER OF 2-PIRIDILOXI-4-NITRILE OREXINE
AU2013296470B2 (en)	2012-08-02	2016-03-17	Merck Sharp & Dohme Corp.	Antidiabetic tricyclic compounds
CN104994848A (en)	2013-02-22	2015-10-21	默沙东公司	Antidiabetic bicyclic compounds
EP2970119B1 (en)	2013-03-14	2021-11-03	Merck Sharp & Dohme Corp.	Novel indole derivatives useful as anti-diabetic agents
EP2968439A2 (en)	2013-03-15	2016-01-20	Synergy Pharmaceuticals Inc.	Compositions useful for the treatment of gastrointestinal disorders
US9708367B2 (en)	2013-03-15	2017-07-18	Synergy Pharmaceuticals, Inc.	Agonists of guanylate cyclase and their uses
PT3004138T (en)	2013-06-05	2024-06-18	Bausch Health Ireland Ltd	Ultra-pure agonists of guanylate cyclase c, method of making and using same
WO2015051496A1 (en)	2013-10-08	2015-04-16	Merck Sharp & Dohme Corp.	Antidiabetic tricyclic compounds
RU2021109549A (en)	2014-08-29	2021-05-13	Тес Фарма С.Р.Л.	Α-AMINO-β-CARBOXYMUCONATE INHIBITORS of ε-SEMIALDEHYDE-DECARBOXYLASE
WO2018069532A1 (en)	2016-10-14	2018-04-19	Tes Pharma S.R.L.	Inhibitors of alpha-amino-beta-carboxymuconic acid semialdehyde decarboxylase
US11072602B2 (en)	2016-12-06	2021-07-27	Merck Sharp & Dohme Corp.	Antidiabetic heterocyclic compounds
CN113302189A (en)	2018-11-20	2021-08-24	Tes制药有限责任公司	Inhibitors of alpha-amino-beta-carboxyadipimic acid semialdehyde decarboxylating enzyme
WO2020167706A1 (en)	2019-02-13	2020-08-20	Merck Sharp & Dohme Corp.	5-alkyl pyrrolidine orexin receptor agonists
US20230018413A1 (en)	2019-08-08	2023-01-19	Merck Sharp & Dohme Corp.	Heteroaryl pyrrolidine and piperidine orexin receptor agonists
JP7443625B2 (en)	2020-08-18	2024-03-05	メルク・シャープ・アンド・ドーム・エルエルシー	Bicycloheptane pyrrolidine orexin receptor agonist

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4242261A (en) *	1979-07-19	1980-12-30	A. H. Robins Company, Inc.	Production of methylene-cycloamines
FR2649100B1 (en) *	1989-06-29	1994-03-04	Laboratorios Dr Esteve Sa	NOVEL AZETIDINES, THEIR PREPARATION AND THEIR APPLICATION AS INTERMEDIATES FOR THE PREPARATION OF COMPOUNDS WITH ANTIMICROBIAL ACTIVITY
JPH05201971A (en) *	1992-01-28	1993-08-10	Hokuriku Seiyaku Co Ltd	Benzenesulfonamide derivative containing cyclic amine
EP0842172A1 (en) *	1995-06-29	1998-05-20	Novo Nordisk A/S	Novel substituted azacyclic or azabicyclic compounds
GB9714129D0 (en) *	1997-07-04	1997-09-10	Pfizer Ltd	Azetidines

2000
- 2000-03-03 FR FR0002777A patent/FR2805810B1/en not_active Expired - Fee Related
2001
- 2001-01-03 UA UA2002097700A patent/UA72319C2/en unknown
- 2001-02-23 TW TW090104188A patent/TWI294420B/en not_active IP Right Cessation
- 2001-03-01 EA EA200200942A patent/EA004649B1/en not_active IP Right Cessation
- 2001-03-01 SK SK1244-2002A patent/SK12442002A3/en unknown
- 2001-03-01 PT PT01909938T patent/PT1263721E/en unknown
- 2001-03-01 IL IL15120901A patent/IL151209A0/en unknown
- 2001-03-01 NZ NZ521076A patent/NZ521076A/en unknown
- 2001-03-01 SI SI200130980T patent/SI1263721T1/en unknown
- 2001-03-01 ES ES01909938T patent/ES2351183T3/en not_active Expired - Lifetime
- 2001-03-01 CN CNB018060269A patent/CN1187325C/en not_active Expired - Fee Related
- 2001-03-01 MX MXPA02008346A patent/MXPA02008346A/en active IP Right Grant
- 2001-03-01 EP EP01909938A patent/EP1263721B1/en not_active Expired - Lifetime
- 2001-03-01 KR KR1020027011516A patent/KR100813740B1/en not_active IP Right Cessation
- 2001-03-01 DE DE60142890T patent/DE60142890D1/en not_active Expired - Lifetime
- 2001-03-01 AT AT01909938T patent/ATE478840T1/en active
- 2001-03-01 AU AU3752601A patent/AU3752601A/en active Pending
- 2001-03-01 WO PCT/FR2001/000601 patent/WO2001064633A1/en active IP Right Grant
- 2001-03-01 EE EEP200200486A patent/EE05081B1/en not_active IP Right Cessation
- 2001-03-01 BR BR0108894-7A patent/BR0108894A/en not_active Application Discontinuation
- 2001-03-01 YU YU65902A patent/YU65902A/en unknown
- 2001-03-01 AU AU2001237526A patent/AU2001237526B2/en not_active Ceased
- 2001-03-01 HU HU0300350A patent/HUP0300350A2/en unknown
- 2001-03-01 OA OA1200200269A patent/OA12221A/en unknown
- 2001-03-01 PL PL01365007A patent/PL365007A1/en not_active IP Right Cessation
- 2001-03-01 JP JP2001563476A patent/JP2003525269A/en not_active Ceased
- 2001-03-01 CA CA002400138A patent/CA2400138A1/en not_active Abandoned
- 2001-03-01 DK DK01909938.1T patent/DK1263721T3/en active
- 2001-03-02 AR ARP010101025A patent/AR034405A1/en unknown
- 2001-09-07 DZ DZ013311A patent/DZ3311A1/en active
2002
- 2002-08-12 IL IL151209A patent/IL151209A/en not_active IP Right Cessation
- 2002-08-28 ZA ZA200206916A patent/ZA200206916B/en unknown
- 2002-08-28 MA MA26793A patent/MA26879A1/en unknown
- 2002-08-29 HR HR20020710A patent/HRP20020710A2/en not_active Application Discontinuation
- 2002-09-02 NO NO20024176A patent/NO324523B1/en not_active IP Right Cessation
- 2002-09-03 BG BG107057A patent/BG107057A/en unknown
2010
- 2010-10-29 CY CY20101100983T patent/CY1111075T1/en unknown

Publication	Publication Date	Title
AU2001237526A1 (en)	2001-11-22	Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
DZ3311A1 (en)	2001-09-07	Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
AU2001237525A1 (en)	2001-11-22	Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same
DZ3313A1 (en)	2001-09-07	Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same
HUP0400636A3 (en)	2004-09-28	Pharmaceutical compositions containing azetidine derivatives, novel azetidine derivatives and preparation thereof
HUP0204242A3 (en)	2004-05-28	Novel 1,3-dihydro-2h-indol-2-one derivatives, their preparation and pharmaceutical compositions compositions containing them
IL154965A0 (en)	2003-10-31	Sulfonamide derivatives, their preparation and pharmaceutical compositions containing them
HUP0300207A3 (en)	2005-07-28	1,2,3,4-tetrahydroisquinoline derivatives, pharmaceutical compositions containing them and their preparation processes
HUP0400837A3 (en)	2007-11-28	2-phenyl-thiazole derivatives, their use and pharmaceutical compositions containing them
HUP0204474A3 (en)	2004-07-28	1h-imidazopyridine derivatives, pharmaceutical compositions containing them and their use
AU2001250420A1 (en)	2001-10-23	Pharmaceutical compositions
HUP0400551A2 (en)	2006-02-28	Piperazine derivatives, their preparation and pharmaceutical compositions containing them
AU2001235737A1 (en)	2001-09-12	Novel 1,3-dihydro-2h-indol-2-one, preparation method and pharmaceutical compositions containing same
IL151912A0 (en)	2003-04-10	Pyrolidine derivatives, their preparation and pharmaceutical compositions containing them
AU2001292331A1 (en)	2002-06-27	5-amidino-2-hydroxybenzenesulfonamide derivatives, pharmaceutical compositions containing the same and intermediates for their preparation
AU2001292331A2 (en)	2003-07-24	5-amidino-2-hydroxybenzenesulfonamide derivatives, pharmaceutical compositions containing the same and intermediates for their preparation
AU2001273919A1 (en)	2001-10-23	Pharmaceutical compositions
IL154966A0 (en)	2003-10-31	Sulfonamide derivatives, their preparation and pharmaceutical compositions containing them
AU3560601A (en)	2001-08-07	Novel isoquinoline derivatives, preparation method and pharmaceutical compositions containing them
AU2002360117A1 (en)	2003-07-03	Aralkyl-tetrahydro-pyridines, their preparation and pharmaceutical compositions containing same
HUP0401713A3 (en)	2012-08-28	Aralkyl-tetrahydro-pyridines, their preparation and pharmaceutical compositions containing same
HUP0300330A3 (en)	2003-09-29	Oligosaccharides, pharmaceutical compositions containing them and preparation thereof
IL154986A0 (en)	2003-10-31	Triazolo-epothilone derivatives, pharmaceutical compositions containing the same and methods for the preparation thereof
AU2001274171A1 (en)	2001-12-11	Aminothiolester compounds, pharmaceutical and cosmetic compositions containing same and uses thereof
AU4884701A (en)	2001-11-20	Malonanilic acid derivatives, medicinal compositions containing the same and usethereof