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IL114142A - Amidino sulphone derivatives their preparation pharmaceutical compositions containing them and their use - Google Patents

Amidino sulphone derivatives their preparation pharmaceutical compositions containing them and their use

Info

Publication number
IL114142A
IL114142A IL11414295A IL11414295A IL114142A IL 114142 A IL114142 A IL 114142A IL 11414295 A IL11414295 A IL 11414295A IL 11414295 A IL11414295 A IL 11414295A IL 114142 A IL114142 A IL 114142A
Authority
IL
Israel
Prior art keywords
amidino
pharmaceutical compositions
compositions containing
preparation pharmaceutical
sulphone derivatives
Prior art date
Application number
IL11414295A
Other languages
English (en)
Other versions
IL114142A0 (en
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9509774.7A external-priority patent/GB9509774D0/en
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of IL114142A0 publication Critical patent/IL114142A0/xx
Priority to IL12871799A priority Critical patent/IL128717A0/xx
Publication of IL114142A publication Critical patent/IL114142A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • C07C317/48—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Immobilizing And Processing Of Enzymes And Microorganisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Steroid Compounds (AREA)
IL11414295A 1994-06-15 1995-06-14 Amidino sulphone derivatives their preparation pharmaceutical compositions containing them and their use IL114142A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IL12871799A IL128717A0 (en) 1994-06-15 1999-02-25 Amino sulphone derivatives

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP94304314 1994-06-15
GBGB9509774.7A GB9509774D0 (en) 1995-05-15 1995-05-15 Enzyme inhibitors

Publications (2)

Publication Number Publication Date
IL114142A0 IL114142A0 (en) 1995-10-31
IL114142A true IL114142A (en) 2000-02-17

Family

ID=26137155

Family Applications (2)

Application Number Title Priority Date Filing Date
IL11414295A IL114142A (en) 1994-06-15 1995-06-14 Amidino sulphone derivatives their preparation pharmaceutical compositions containing them and their use
IL12871799A IL128717A0 (en) 1994-06-15 1999-02-25 Amino sulphone derivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL12871799A IL128717A0 (en) 1994-06-15 1999-02-25 Amino sulphone derivatives

Country Status (29)

Country Link
US (2) USRE39576E1 (da)
EP (2) EP0765308B1 (da)
JP (2) JP2989010B2 (da)
KR (1) KR100430207B1 (da)
CN (1) CN1070849C (da)
AT (2) ATE191470T1 (da)
AU (1) AU692892B2 (da)
BR (1) BR9507995A (da)
CA (1) CA2192668A1 (da)
CY (2) CY2238B1 (da)
DE (2) DE69529101T2 (da)
DK (2) DK0957087T3 (da)
ES (2) ES2189322T3 (da)
FI (1) FI965019A (da)
GR (1) GR3033746T3 (da)
HK (1) HK1003935A1 (da)
HU (1) HUT77407A (da)
IL (2) IL114142A (da)
IS (1) IS4384A (da)
MX (1) MX9606136A (da)
MY (1) MY115437A (da)
NO (1) NO308655B1 (da)
NZ (1) NZ289157A (da)
PT (2) PT765308E (da)
RU (1) RU2162841C2 (da)
SI (2) SI0765308T1 (da)
TW (1) TW442453B (da)
WO (1) WO1995034534A1 (da)
ZA (1) ZA954940B (da)

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JP6517319B2 (ja) 2014-03-28 2019-05-22 キャリター・サイエンシーズ・リミテッド・ライアビリティ・カンパニーＣａｌｉｔｏｒ Ｓｃｉｅｎｃｅｓ， Ｌｌｃ 置換されたヘテロアリール化合物および使用方法
TW201625247A (zh) 2014-05-12 2016-07-16 葛蘭素史密斯克藍智慧財產權有限公司 用於治療傳染性疾病之醫藥組合物
GB201512635D0 (en) 2015-07-17 2015-08-26 Ucl Business Plc Uses of therapeutic compounds
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JP7254076B2 (ja) 2017-11-19 2023-04-07 サンシャイン・レイク・ファーマ・カンパニー・リミテッド 置換ヘテロアリール化合物及び使用方法
KR20200112900A (ko) 2018-01-20 2020-10-05 선샤인 레이크 파르마 컴퍼니 리미티드 치환된 아미노피리미딘 화합물 및 이의 사용 방법
CN116194114A (zh) 2020-03-26 2023-05-30 葛兰素史密斯克莱知识产权发展有限公司 用于防止或治疗病毒感染的组织蛋白酶抑制剂

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Also Published As

Publication number Publication date
HU9603454D0 (en) 1997-02-28
AU692892B2 (en) 1998-06-18
EP0765308A1 (en) 1997-04-02
NO965379D0 (no) 1996-12-13
DE69529101D1 (de) 2003-01-16
DE69516141T2 (de) 2000-10-19
FI965019A0 (fi) 1996-12-13
JP2989010B2 (ja) 1999-12-13
EP0765308B1 (en) 2000-04-05
IL128717A0 (en) 2000-01-31
ES2145282T3 (es) 2000-07-01
ATE191470T1 (de) 2000-04-15
HK1003935A1 (en) 1998-11-13
ES2189322T3 (es) 2003-07-01
NZ289157A (en) 1998-03-25
MY115437A (en) 2003-06-30
CA2192668A1 (en) 1995-12-21
USRE39576E1 (en) 2007-04-17
SI0765308T1 (en) 2000-08-31
EP0957087A2 (en) 1999-11-17
TW442453B (en) 2001-06-23
EP0957087A3 (en) 2000-12-20
NO965379L (no) 1996-12-13
EP0957087B1 (en) 2002-12-04
DK0765308T3 (da) 2000-09-11
SI0957087T1 (en) 2003-04-30
CN1155276A (zh) 1997-07-23
ATE229001T1 (de) 2002-12-15
FI965019A (fi) 1996-12-13
CN1070849C (zh) 2001-09-12
AU2891795A (en) 1996-01-05
NO308655B1 (no) 2000-10-09
ZA954940B (en) 1996-12-17
DE69529101T2 (de) 2003-11-13
JPH10506371A (ja) 1998-06-23
IS4384A (is) 1996-11-13
KR100430207B1 (ko) 2004-07-19
DE69516141D1 (de) 2000-05-11
JP2000026402A (ja) 2000-01-25
BR9507995A (pt) 1997-08-05
US5889056A (en) 1999-03-30
MX9606136A (es) 1998-06-30
HUT77407A (hu) 1998-04-28
GR3033746T3 (en) 2000-10-31
JP3614711B2 (ja) 2005-01-26
DK0957087T3 (da) 2003-03-24
PT957087E (pt) 2003-04-30
PT765308E (pt) 2000-09-29
CY2238B1 (en) 2003-07-04
WO1995034534A1 (en) 1995-12-21
IL114142A0 (en) 1995-10-31
CY2455B1 (en) 2005-06-03
RU2162841C2 (ru) 2001-02-10

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