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EA200900658A1 - Производные индазолилэфиров или -амидов для лечения расстройств, опосредованных глюкокортиодными рецепторами - Google Patents

Производные индазолилэфиров или -амидов для лечения расстройств, опосредованных глюкокортиодными рецепторами

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Publication number
EA200900658A1
EA200900658A1 EA200900658A EA200900658A EA200900658A1 EA 200900658 A1 EA200900658 A1 EA 200900658A1 EA 200900658 A EA200900658 A EA 200900658A EA 200900658 A EA200900658 A EA 200900658A EA 200900658 A1 EA200900658 A1 EA 200900658A1
Authority
EA
Eurasian Patent Office
Prior art keywords
derivatives
amides
ethers
indasolyl
glucocortia
Prior art date
Application number
EA200900658A
Other languages
English (en)
Other versions
EA016895B1 (ru
Inventor
Маркус Бергер
Ян Дамен
Андерс Эрикссон
Балинт Габос
Томас Ханссон
Мартин Хеммерлинг
Кристер Хенрикссон
Светлана Иванова
Матти Лепистё
Даррен Маккерречер
Магнус Мунк Ав Розеншёльд
Стинабритт Нильссон
Хартмут Ревинкель
Камилла Тафлин
Карл Эдман
Original Assignee
Астразенека Аб
Байер Шеринг Фарма Актиенгезелльшафт
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Астразенека Аб, Байер Шеринг Фарма Актиенгезелльшафт filed Critical Астразенека Аб
Publication of EA200900658A1 publication Critical patent/EA200900658A1/ru
Publication of EA016895B1 publication Critical patent/EA016895B1/ru

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    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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Abstract

Настоящее изобретение относится к новым производным индазолилэфиров или -амидов, к фармацевтическим композициям, содержащим такие производные, к способам получения таких новых производных и к применению таких производных в качестве лекарственных средств. Соединение формулы (I)
EA200900658A 2006-12-21 2007-12-20 Производные индазолил-эфиров или -амидов для лечения расстройств, опосредованных глюкокортикоидными рецепторами EA016895B1 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US87118406P 2006-12-21 2006-12-21
US94174507P 2007-06-04 2007-06-04
US97852607P 2007-10-09 2007-10-09
PCT/SE2007/001136 WO2008076048A1 (en) 2006-12-21 2007-12-20 Indazolyl ester and amide derivatives for the treatment of glucocorticoid receptor mediated disorders

Publications (2)

Publication Number Publication Date
EA200900658A1 true EA200900658A1 (ru) 2009-12-30
EA016895B1 EA016895B1 (ru) 2012-08-30

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CL2007003804A1 (es) 2008-08-22
US20120252770A1 (en) 2012-10-04
HK1133651A1 (en) 2010-04-01
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ECSP099452A (es) 2009-07-31
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US20080214641A1 (en) 2008-09-04
AU2007334659B2 (en) 2011-01-27
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CR10875A (es) 2009-07-20
IL198880A (en) 2013-10-31
GT200900175A (es) 2014-03-18
US8143290B2 (en) 2012-03-27
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EA016895B1 (ru) 2012-08-30
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CA2673277A1 (en) 2008-06-26
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