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AR033168A1 - Solucion oral de aripiprazol - Google Patents

Solucion oral de aripiprazol

Info

Publication number
AR033168A1
AR033168A1 ARP020101366A ARP020101366A AR033168A1 AR 033168 A1 AR033168 A1 AR 033168A1 AR P020101366 A ARP020101366 A AR P020101366A AR P020101366 A ARP020101366 A AR P020101366A AR 033168 A1 AR033168 A1 AR 033168A1
Authority
AR
Argentina
Prior art keywords
solution
oral
aripiprazol
acid
aripiprazole
Prior art date
Application number
ARP020101366A
Other languages
English (en)
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23099862&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR033168(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of AR033168A1 publication Critical patent/AR033168A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Psychiatry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente se proporciona para una solucion farmacéutica adecuada para administracion oral que comprende aripiprazol, un sistema de solvente farmacéuticamente adecuado, uno o más agentes mejoradores/enmascarantes del sabor y uno o más agentes seleccionados del grupo que consiste de ácido láctico, ácido acético, ácido tartárico y ácido cítrico, en donde la solucion tiene un pH desde 2.5 hasta 4.5.
ARP020101366A 2001-04-25 2002-04-15 Solucion oral de aripiprazol AR033168A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US28671801P 2001-04-25 2001-04-25

Publications (1)

Publication Number Publication Date
AR033168A1 true AR033168A1 (es) 2003-12-03

Family

ID=23099862

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP020101366A AR033168A1 (es) 2001-04-25 2002-04-15 Solucion oral de aripiprazol

Country Status (37)

Country Link
US (1) US6977257B2 (es)
EP (2) EP2436384B2 (es)
JP (1) JP4401077B2 (es)
KR (1) KR100909329B1 (es)
CN (1) CN1512884B (es)
AR (1) AR033168A1 (es)
AT (1) ATE537831T1 (es)
AU (1) AU2002254722B2 (es)
BG (1) BG66177B1 (es)
BR (1) BR0208986A (es)
CA (1) CA2445276C (es)
CY (1) CY1112606T1 (es)
CZ (1) CZ306181B6 (es)
DK (1) DK1381367T3 (es)
EE (1) EE05581B1 (es)
ES (1) ES2377855T3 (es)
GE (1) GEP20053602B (es)
HK (2) HK1058316A1 (es)
HR (1) HRP20030870B1 (es)
HU (1) HU230456B1 (es)
IL (2) IL158202A0 (es)
IS (1) IS2863B (es)
MX (1) MXPA03009728A (es)
MY (1) MY129350A (es)
NO (1) NO324606B1 (es)
NZ (1) NZ528550A (es)
PE (1) PE20021086A1 (es)
PL (1) PL206882B1 (es)
PT (1) PT1381367E (es)
RS (1) RS52082B (es)
RU (1) RU2295960C2 (es)
SK (1) SK287948B6 (es)
TW (1) TWI337865B (es)
UA (1) UA76144C2 (es)
UY (1) UY27273A1 (es)
WO (1) WO2002085366A1 (es)
ZA (1) ZA200307797B (es)

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JP6034377B2 (ja) * 2011-06-27 2016-11-30 シャンハイ チョンシ ファーマシューティカル コーポレイション アリピプラゾール医薬製剤及びその調製方法
CN102846616B (zh) * 2011-06-27 2015-05-06 上海中西制药有限公司 一种阿立哌唑制剂及其制备方法
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ES2764383T3 (es) 2012-03-19 2020-06-03 Alkermes Pharma Ireland Ltd Composiciones farmacéuticas que comprenden ésteres de glicerol
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Also Published As

Publication number Publication date
DK1381367T3 (da) 2012-04-10
EP2436384B1 (en) 2015-06-10
SK12642003A3 (sk) 2004-07-07
EP2436384A3 (en) 2012-09-19
CZ20032821A3 (cs) 2004-09-15
IS6994A (is) 2003-10-14
HRP20030870B1 (en) 2011-10-31
GEP20053602B (en) 2005-08-10
RU2003132426A (ru) 2005-04-20
BG108216A (bg) 2004-12-30
NO20034705L (no) 2003-11-28
NO20034705D0 (no) 2003-10-21
EP1381367B1 (en) 2011-12-21
NZ528550A (en) 2005-03-24
HUP0303946A3 (en) 2005-06-28
EP1381367A1 (en) 2004-01-21
HK1168792A1 (en) 2013-01-11
CY1112606T1 (el) 2016-02-10
KR20030096332A (ko) 2003-12-24
SK287948B6 (sk) 2012-06-04
HK1058316A1 (en) 2004-05-14
CA2445276A1 (en) 2002-10-31
EE05581B1 (et) 2012-10-15
JP2004532225A (ja) 2004-10-21
HU230456B1 (hu) 2016-07-28
TWI337865B (en) 2011-03-01
EE200300523A (et) 2004-02-16
CN1512884B (zh) 2010-05-26
US20020193438A1 (en) 2002-12-19
MXPA03009728A (es) 2004-01-29
IS2863B (is) 2013-12-15
ATE537831T1 (de) 2012-01-15
IL158202A (en) 2008-04-13
MY129350A (en) 2007-03-30
JP4401077B2 (ja) 2010-01-20
UY27273A1 (es) 2002-11-29
UA76144C2 (uk) 2006-07-17
KR100909329B1 (ko) 2009-07-24
HUP0303946A2 (hu) 2004-04-28
CZ306181B6 (cs) 2016-09-14
BG66177B1 (bg) 2011-11-30
ZA200307797B (en) 2004-10-06
CN1512884A (zh) 2004-07-14
PE20021086A1 (es) 2002-12-14
PL364666A1 (en) 2004-12-13
PT1381367E (pt) 2012-03-01
PL206882B1 (pl) 2010-10-29
EP2436384B2 (en) 2018-05-23
US6977257B2 (en) 2005-12-20
RU2295960C2 (ru) 2007-03-27
WO2002085366A1 (en) 2002-10-31
EP1381367A4 (en) 2009-07-01
CA2445276C (en) 2009-10-13
EP2436384A2 (en) 2012-04-04
HRP20030870A2 (en) 2004-06-30
IL158202A0 (en) 2004-05-12
BR0208986A (pt) 2004-04-20
NO324606B1 (no) 2007-11-26
RS52082B (sr) 2012-06-30
YU84703A (sh) 2006-08-17
ES2377855T3 (es) 2012-04-02
AU2002254722B2 (en) 2006-11-09

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