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NO20044113L - Inhibitorer av histon-deacetylase - Google Patents

Inhibitorer av histon-deacetylase

Info

Publication number
NO20044113L
NO20044113L NO20044113A NO20044113A NO20044113L NO 20044113 L NO20044113 L NO 20044113L NO 20044113 A NO20044113 A NO 20044113A NO 20044113 A NO20044113 A NO 20044113A NO 20044113 L NO20044113 L NO 20044113L
Authority
NO
Norway
Prior art keywords
inhibitors
histone deacetylase
deacetylase
histone
Prior art date
Application number
NO20044113A
Other languages
English (en)
Inventor
Marc Gustaaf Celine Verdonck
Kristof Van Emelen
Patrick Rene Angibaud
Lieven Meerpoel
Sven Franciscus Anna Va Brandt
Alexey Borisovich Dyatkin
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of NO20044113L publication Critical patent/NO20044113L/no

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/402—1-aryl substituted, e.g. piretanide
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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OA12791A (en) 2006-07-10
HK1078473A1 (en) 2006-03-17
UA78033C2 (en) 2007-02-15
AU2003212335B8 (en) 2009-04-23
AU2003212337B2 (en) 2009-06-11
US8916554B2 (en) 2014-12-23
ZA200407237B (en) 2005-09-28
AU2003218736B2 (en) 2009-01-08
EP1485099B1 (en) 2010-07-07
US9150560B2 (en) 2015-10-06
CA2476065A1 (en) 2003-09-18
DE60326549D1 (en) 2009-04-23
IL164006A (en) 2010-11-30
ES2347544T3 (es) 2010-11-02
ZA200407235B (en) 2005-10-04
US20130245034A1 (en) 2013-09-19

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