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NO20020343L - Kaspase-inhibitorer og anvendelse derav - Google Patents

Kaspase-inhibitorer og anvendelse derav

Info

Publication number
NO20020343L
NO20020343L NO20020343A NO20020343A NO20020343L NO 20020343 L NO20020343 L NO 20020343L NO 20020343 A NO20020343 A NO 20020343A NO 20020343 A NO20020343 A NO 20020343A NO 20020343 L NO20020343 L NO 20020343L
Authority
NO
Norway
Prior art keywords
caspase inhibitors
caspase
inhibitors
Prior art date
Application number
NO20020343A
Other languages
English (en)
Other versions
NO20020343D0 (no
Inventor
Julian Golec
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of NO20020343D0 publication Critical patent/NO20020343D0/no
Publication of NO20020343L publication Critical patent/NO20020343L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
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    • C—CHEMISTRY; METALLURGY
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    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
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    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
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  • Addiction (AREA)
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NO20020343A 2000-05-23 2002-01-22 Kaspase-inhibitorer og anvendelse derav NO20020343L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US20636200P 2000-05-23 2000-05-23
US21700600P 2000-07-10 2000-07-10
PCT/US2001/017075 WO2001090070A2 (en) 2000-05-23 2001-05-23 Caspase inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
NO20020343D0 NO20020343D0 (no) 2002-01-22
NO20020343L true NO20020343L (no) 2002-03-21

Family

ID=26901274

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20020343A NO20020343L (no) 2000-05-23 2002-01-22 Kaspase-inhibitorer og anvendelse derav

Country Status (16)

Country Link
US (1) US7053057B2 (no)
EP (1) EP1283827A2 (no)
JP (1) JP2003534325A (no)
KR (1) KR20020025959A (no)
AP (1) AP2002002407A0 (no)
AR (1) AR028619A1 (no)
AU (1) AU2001265008A1 (no)
CA (1) CA2380935A1 (no)
MX (1) MXPA02000823A (no)
NO (1) NO20020343L (no)
NZ (1) NZ516918A (no)
PE (1) PE20020058A1 (no)
PL (1) PL357713A1 (no)
SK (1) SK1192002A3 (no)
TR (1) TR200200767T1 (no)
WO (1) WO2001090070A2 (no)

Families Citing this family (46)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002541237A (ja) 1999-04-09 2002-12-03 サイトビア インコーポレイテッド カスパーゼインヒビターおよびその使用
EP1163208B1 (en) * 1999-08-06 2004-05-12 Vertex Pharmaceuticals Incorporated Caspase inhibitors and uses thereof
ATE409688T1 (de) 1999-08-27 2008-10-15 Cytovia Inc Substituierte alpha-hydroxy-säuren als caspase- hemmer und ihre verwendung
PE20011350A1 (es) 2000-05-19 2002-01-15 Vertex Pharma PROFARMACO DE UN INHIBIDOR DE ENZIMA CONVERTIDORA DE INTERLEUCINA-1ß (ICE)
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AR028619A1 (es) 2003-05-14
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AP2002002407A0 (en) 2002-03-31
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