NO20020343L - Kaspase-inhibitorer og anvendelse derav - Google Patents
Kaspase-inhibitorer og anvendelse deravInfo
- Publication number
- NO20020343L NO20020343L NO20020343A NO20020343A NO20020343L NO 20020343 L NO20020343 L NO 20020343L NO 20020343 A NO20020343 A NO 20020343A NO 20020343 A NO20020343 A NO 20020343A NO 20020343 L NO20020343 L NO 20020343L
- Authority
- NO
- Norway
- Prior art keywords
- caspase inhibitors
- caspase
- inhibitors
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/30—Oxygen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
- C07D333/16—Radicals substituted by singly bound hetero atoms other than halogen by oxygen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Physical Education & Sports Medicine (AREA)
- Oncology (AREA)
- Diabetes (AREA)
- Biomedical Technology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurosurgery (AREA)
- Communicable Diseases (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Hematology (AREA)
- Virology (AREA)
- Pulmonology (AREA)
- Cardiology (AREA)
- Immunology (AREA)
- Heart & Thoracic Surgery (AREA)
- Molecular Biology (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US20636200P | 2000-05-23 | 2000-05-23 | |
US21700600P | 2000-07-10 | 2000-07-10 | |
PCT/US2001/017075 WO2001090070A2 (en) | 2000-05-23 | 2001-05-23 | Caspase inhibitors and uses thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20020343D0 NO20020343D0 (no) | 2002-01-22 |
NO20020343L true NO20020343L (no) | 2002-03-21 |
Family
ID=26901274
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20020343A NO20020343L (no) | 2000-05-23 | 2002-01-22 | Kaspase-inhibitorer og anvendelse derav |
Country Status (16)
Country | Link |
---|---|
US (1) | US7053057B2 (no) |
EP (1) | EP1283827A2 (no) |
JP (1) | JP2003534325A (no) |
KR (1) | KR20020025959A (no) |
AP (1) | AP2002002407A0 (no) |
AR (1) | AR028619A1 (no) |
AU (1) | AU2001265008A1 (no) |
CA (1) | CA2380935A1 (no) |
MX (1) | MXPA02000823A (no) |
NO (1) | NO20020343L (no) |
NZ (1) | NZ516918A (no) |
PE (1) | PE20020058A1 (no) |
PL (1) | PL357713A1 (no) |
SK (1) | SK1192002A3 (no) |
TR (1) | TR200200767T1 (no) |
WO (1) | WO2001090070A2 (no) |
Families Citing this family (46)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2002541237A (ja) | 1999-04-09 | 2002-12-03 | サイトビア インコーポレイテッド | カスパーゼインヒビターおよびその使用 |
EP1163208B1 (en) * | 1999-08-06 | 2004-05-12 | Vertex Pharmaceuticals Incorporated | Caspase inhibitors and uses thereof |
ATE409688T1 (de) | 1999-08-27 | 2008-10-15 | Cytovia Inc | Substituierte alpha-hydroxy-säuren als caspase- hemmer und ihre verwendung |
PE20011350A1 (es) | 2000-05-19 | 2002-01-15 | Vertex Pharma | PROFARMACO DE UN INHIBIDOR DE ENZIMA CONVERTIDORA DE INTERLEUCINA-1ß (ICE) |
US6878743B2 (en) | 2001-09-18 | 2005-04-12 | Sunesis Pharmaceuticals, Inc. | Small molecule inhibitors of caspases |
US7410956B2 (en) | 2002-02-11 | 2008-08-12 | Vertex Pharmaceuticals Incorporated | Caspase inhibitor prodrugs |
EP1499898A2 (en) * | 2002-04-19 | 2005-01-26 | Vertex Pharmaceuticals Incorporated | Regulation of tnf-alpha |
CA2501196A1 (en) * | 2002-10-10 | 2004-04-22 | Becton, Dickinson And Company | Sample collection system with caspase inhibitor |
CA2526493A1 (en) * | 2003-05-22 | 2004-12-02 | Theraptosis S.A. | Means for preventing and treating cellular death and their biological applications |
AU2003902704A0 (en) * | 2003-05-29 | 2003-06-19 | Crc For Waste Management And Pollution Control Limited Of Unsw | Process for producing a nanoscale zero-valent metal |
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2001
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- 2001-05-23 MX MXPA02000823A patent/MXPA02000823A/es not_active Application Discontinuation
- 2001-05-23 SK SK119-2002A patent/SK1192002A3/sk unknown
- 2001-05-23 PL PL01357713A patent/PL357713A1/xx not_active Application Discontinuation
- 2001-05-23 WO PCT/US2001/017075 patent/WO2001090070A2/en active IP Right Grant
- 2001-05-23 CA CA002380935A patent/CA2380935A1/en not_active Abandoned
- 2001-05-23 AU AU2001265008A patent/AU2001265008A1/en not_active Abandoned
- 2001-05-23 TR TR2002/00767T patent/TR200200767T1/xx unknown
- 2001-05-23 AP APAP/P/2002/002407A patent/AP2002002407A0/en unknown
- 2001-05-23 NZ NZ516918A patent/NZ516918A/en unknown
- 2001-05-23 US US09/863,649 patent/US7053057B2/en not_active Expired - Fee Related
- 2001-05-23 EP EP01939497A patent/EP1283827A2/en not_active Withdrawn
- 2001-05-23 JP JP2001586259A patent/JP2003534325A/ja active Pending
- 2001-05-23 AR ARP010102477A patent/AR028619A1/es unknown
- 2001-05-23 PE PE2001000468A patent/PE20020058A1/es not_active Application Discontinuation
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2002
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KR20020025959A (ko) | 2002-04-04 |
MXPA02000823A (es) | 2002-07-30 |
CA2380935A1 (en) | 2001-11-29 |
WO2001090070A2 (en) | 2001-11-29 |
US7053057B2 (en) | 2006-05-30 |
EP1283827A2 (en) | 2003-02-19 |
NZ516918A (en) | 2004-06-25 |
AR028619A1 (es) | 2003-05-14 |
WO2001090070A3 (en) | 2002-04-11 |
PE20020058A1 (es) | 2002-01-31 |
US20020061853A1 (en) | 2002-05-23 |
PL357713A1 (en) | 2004-07-26 |
JP2003534325A (ja) | 2003-11-18 |
AP2002002407A0 (en) | 2002-03-31 |
SK1192002A3 (en) | 2002-09-10 |
TR200200767T1 (tr) | 2002-09-23 |
AU2001265008A1 (en) | 2001-12-03 |
NO20020343D0 (no) | 2002-01-22 |
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