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SK4602003A3 - EP4 receptor inhibitors to treat rheumatoid arthritis - Google Patents

EP4 receptor inhibitors to treat rheumatoid arthritis Download PDF

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Publication number
SK4602003A3
SK4602003A3 SK460-2003A SK4602003A SK4602003A3 SK 4602003 A3 SK4602003 A3 SK 4602003A3 SK 4602003 A SK4602003 A SK 4602003A SK 4602003 A3 SK4602003 A3 SK 4602003A3
Authority
SK
Slovakia
Prior art keywords
ethyl
phenyl
amino
imidazo
dimethyl
Prior art date
Application number
SK460-2003A
Other languages
English (en)
Slovak (sk)
Inventor
Laurent Audoly
Takako Okumura
Masato Shimojo
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of SK4602003A3 publication Critical patent/SK4602003A3/sk

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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