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PT88204A - New 2-piperidinyl:methyl-1,2,3,4-tetra:hydro-isoquinoline derivs. - with selective action on HT one A serotoninergic receptors, e.g. for treating depression and cardiovascular disease - Google Patents

New 2-piperidinyl:methyl-1,2,3,4-tetra:hydro-isoquinoline derivs. - with selective action on HT one A serotoninergic receptors, e.g. for treating depression and cardiovascular disease

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Publication number
PT88204A
PT88204A PT8820488A PT8820488A PT88204A PT 88204 A PT88204 A PT 88204A PT 8820488 A PT8820488 A PT 8820488A PT 8820488 A PT8820488 A PT 8820488A PT 88204 A PT88204 A PT 88204A
Authority
PT
Portugal
Prior art keywords
new
piperidinyl
hydro
tetra
methyl
Prior art date
Application number
PT8820488A
Other languages
Portuguese (pt)
Inventor
Pascal George
Mireille Sevrin
Christian Maloizel
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8711288A external-priority patent/FR2619110B1/en
Priority claimed from FR8718342A external-priority patent/FR2625504B2/en
Priority claimed from FR8805130A external-priority patent/FR2630114B2/en
Application filed by Synthelabo filed Critical Synthelabo
Publication of PT88204A publication Critical patent/PT88204A/en

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  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Ni(piperidinylmethyl) -tetrahydroisoquinoline derivs. of formula (I) and their pharmaceutically acceptable acid addn. salts are new: R = (a) H; (b) 1-6C alkyl, allyl, 3-6C cycloalkylmethyl, benzyl (opt. substd. by 1-3 of halo, CF3, NO2, NH2, NMe2, CN, CONH2, or 1-3C alkyl, alkoxy or alkylthio), 2-phenylethyl, 3-phenylpropyl, 3-phenylpropen-2-yl, phenylcarbonylmethyl, naphthylmethyl, pyridylmethyl, furanylmethyl, or thienylmethyl; (c) 2-6C alkanoyl, 3-6C cycloalkylcarbonyl, CF3CO, phenylcarbonyl (opt. substd. by halo, CF3, NO2 or 1-3C alkyl, alkoxy or alkylthio), 1-oxo-3-phenylpropen-2-yl, naphthylcarbonyl, pyridinylcarbonyl, furancarbonyl, thienylcarbonyl or 2- or 5-indolylcarbonyl.
PT8820488A 1987-08-07 1988-08-05 New 2-piperidinyl:methyl-1,2,3,4-tetra:hydro-isoquinoline derivs. - with selective action on HT one A serotoninergic receptors, e.g. for treating depression and cardiovascular disease PT88204A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR8711288A FR2619110B1 (en) 1987-08-07 1987-08-07 ((PIPERIDINYL-4) METHYL) -2 TETRAHYDRO-1,2,3,4 ISOQUINOLEINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR8718342A FR2625504B2 (en) 1987-08-07 1987-12-30 ((BENZOYL-1 PIPERIDINYL-4) METHYL) -2 TETRAHYDRO-1,2,3,4 ISOQUINOLEINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR8805130A FR2630114B2 (en) 1987-08-07 1988-04-19 (PIPERIDINYL-4) METHYL) -2 TETRAHYDRO-1,2,3,4 ISOQUINOLEINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Publications (1)

Publication Number Publication Date
PT88204A true PT88204A (en) 1989-06-30

Family

ID=27251492

Family Applications (1)

Application Number Title Priority Date Filing Date
PT8820488A PT88204A (en) 1987-08-07 1988-08-05 New 2-piperidinyl:methyl-1,2,3,4-tetra:hydro-isoquinoline derivs. - with selective action on HT one A serotoninergic receptors, e.g. for treating depression and cardiovascular disease

Country Status (1)

Country Link
PT (1) PT88204A (en)

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Effective date: 19941115