KR20090063228A - 정신분열증 치료용 비페프루녹스를 위한 적정 계획 및 이에사용하기 위한 키트 - Google Patents
정신분열증 치료용 비페프루녹스를 위한 적정 계획 및 이에사용하기 위한 키트 Download PDFInfo
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- KR20090063228A KR20090063228A KR1020097006567A KR20097006567A KR20090063228A KR 20090063228 A KR20090063228 A KR 20090063228A KR 1020097006567 A KR1020097006567 A KR 1020097006567A KR 20097006567 A KR20097006567 A KR 20097006567A KR 20090063228 A KR20090063228 A KR 20090063228A
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- bifeprunox
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Classifications
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A—HUMAN NECESSITIES
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- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Addiction (AREA)
- Anesthesiology (AREA)
- Inorganic Chemistry (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US84124406P | 2006-08-31 | 2006-08-31 | |
| EP06119936.0 | 2006-08-31 | ||
| EP06119936 | 2006-08-31 | ||
| US60/841,244 | 2006-08-31 | ||
| US84149506P | 2006-09-01 | 2006-09-01 | |
| US60/841,495 | 2006-09-01 | ||
| EP06120016 | 2006-09-01 | ||
| EP06120016.8 | 2006-09-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20090063228A true KR20090063228A (ko) | 2009-06-17 |
Family
ID=38704953
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020097006567A KR20090063228A (ko) | 2006-08-31 | 2007-08-29 | 정신분열증 치료용 비페프루녹스를 위한 적정 계획 및 이에사용하기 위한 키트 |
Country Status (10)
| Country | Link |
|---|---|
| EP (2) | EP2059244A1 (pt) |
| JP (2) | JP2010501626A (pt) |
| KR (1) | KR20090063228A (pt) |
| AU (2) | AU2007291234A1 (pt) |
| BR (1) | BRPI0715445A2 (pt) |
| CA (2) | CA2661120A1 (pt) |
| EA (1) | EA200970239A1 (pt) |
| IL (1) | IL196867A0 (pt) |
| NO (1) | NO20091243L (pt) |
| WO (2) | WO2008025780A1 (pt) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010060742A1 (en) * | 2008-11-03 | 2010-06-03 | Solvay Pharmaceuticals B.V. | Combination of bifeprunox and an antipsychotic drug with d2/5-ht2a receptor antagonistic activity for treating cns disorders |
| WO2010070061A1 (en) * | 2008-12-19 | 2010-06-24 | Abbott Healthcare Products B.V. | Compositions, kits and methods of a titration schedule for bifeprunox compounds |
| LT2445502T (lt) | 2009-06-25 | 2017-09-25 | Alkermes Pharma Ireland Limited | Heterocikliniai junginiai, skirti neurologinių ir fiziologinių susirgimų gydymui |
| WO2011023796A1 (en) | 2009-08-31 | 2011-03-03 | Abbott Healthcare Products B.V. | Bifeprunox for treating addiction |
| JP6654042B2 (ja) | 2012-09-19 | 2020-02-26 | アルカームス ファーマ アイルランド リミテッド | 貯蔵安定性が改善された医薬組成物 |
| EP3119399A4 (en) | 2014-03-20 | 2017-09-27 | Alkermes Pharma Ireland Limited | Aripiprazole formulations having increased injection speeds |
| AU2019230014A1 (en) | 2018-03-05 | 2020-09-17 | Alkermes Pharma Ireland Limited | Aripiprazole dosing strategy |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TR199801942T2 (xx) | 1996-03-29 | 2000-08-21 | Duphar International Research B.V. | Piperazin ve piperidin bile�ikleri. |
| CA2310950C (en) * | 2000-04-03 | 2005-11-08 | Janssen Pharmaceutica N.V. | An efficacious dosage regiment of galantamine that reduces side effects |
| AR034206A1 (es) | 2001-02-16 | 2004-02-04 | Solvay Pharm Bv | Un procedimiento para la preparacion de mesilatos de derivados de piperazina y dichos mesilatos |
| AR045362A1 (es) * | 2003-08-18 | 2005-10-26 | Solvay Pharm Bv | Forma cristalina estable de mesilato de bifeprunox (monometansulfonato de 7-[4-([1,1- bifenil] -3- ilmetil) -1- piperazinil] - 2-(3h) -benzoxazolona |
| US7423040B2 (en) * | 2005-02-18 | 2008-09-09 | Irene Eijgendaal | Stable crystalline form of bifeprunox mesylate, dosage forms thereof and methods for using same |
| RU2394821C2 (ru) | 2005-08-22 | 2010-07-20 | Солвей Фармасьютикал Б.В. | N-оксиды как пролекарства производных пиперазина и пиперидина |
-
2007
- 2007-08-29 BR BRPI0715445-3A patent/BRPI0715445A2/pt not_active IP Right Cessation
- 2007-08-29 WO PCT/EP2007/058957 patent/WO2008025780A1/en active Application Filing
- 2007-08-29 AU AU2007291234A patent/AU2007291234A1/en not_active Abandoned
- 2007-08-29 EP EP07802974A patent/EP2059244A1/en not_active Withdrawn
- 2007-08-29 AU AU2007291235A patent/AU2007291235A1/en not_active Abandoned
- 2007-08-29 JP JP2009526089A patent/JP2010501626A/ja not_active Withdrawn
- 2007-08-29 EP EP07802975A patent/EP2059245A1/en not_active Withdrawn
- 2007-08-29 CA CA002661120A patent/CA2661120A1/en not_active Abandoned
- 2007-08-29 KR KR1020097006567A patent/KR20090063228A/ko not_active Application Discontinuation
- 2007-08-29 EA EA200970239A patent/EA200970239A1/ru unknown
- 2007-08-29 JP JP2009526088A patent/JP2010501625A/ja not_active Withdrawn
- 2007-08-29 CA CA002661800A patent/CA2661800A1/en not_active Abandoned
- 2007-08-29 WO PCT/EP2007/058958 patent/WO2008025781A1/en active Application Filing
-
2009
- 2009-02-03 IL IL196867A patent/IL196867A0/en unknown
- 2009-03-25 NO NO20091243A patent/NO20091243L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EA200970239A1 (ru) | 2009-08-28 |
| EP2059244A1 (en) | 2009-05-20 |
| WO2008025781A1 (en) | 2008-03-06 |
| AU2007291235A1 (en) | 2008-03-06 |
| JP2010501625A (ja) | 2010-01-21 |
| AU2007291234A1 (en) | 2008-03-06 |
| CA2661800A1 (en) | 2008-03-06 |
| NO20091243L (no) | 2009-03-25 |
| JP2010501626A (ja) | 2010-01-21 |
| BRPI0715445A2 (pt) | 2014-05-13 |
| CA2661120A1 (en) | 2008-03-06 |
| WO2008025780A1 (en) | 2008-03-06 |
| IL196867A0 (en) | 2009-11-18 |
| EP2059245A1 (en) | 2009-05-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| WITN | Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid |