IL112519A0 - 5-heteroarylindole derivatives - Google Patents

5-heteroarylindole derivatives

Info

Publication number: IL112519A0
Authority: IL; Israel
Prior art keywords: heteroarylindole; derivatives; heteroarylindole derivatives
Prior art date: 1994-02-10

Application number

IL11251995A

Other languages

English (en)

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-02-10

Filing date

1995-02-02

Publication date

1995-05-26

1995-02-02 Application filed by Pfizer filed Critical Pfizer

1995-05-26 Publication of IL112519A0 publication Critical patent/IL112519A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Neurosurgery (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Indole Compounds (AREA)

IL11251995A 1994-02-10 1995-02-02 5-heteroarylindole derivatives IL112519A0 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US19455394A	1994-02-10	1994-02-10

Publications (1)

Publication Number	Publication Date
IL112519A0 true IL112519A0 (en)	1995-05-26

Family

ID=22718035

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL11251995A IL112519A0 (en)	1994-02-10	1995-02-02	5-heteroarylindole derivatives

Country Status (12)

Country	Link
US (1)	US5688809A (no)
EP (1)	EP0743942A1 (no)
JP (1)	JP2829788B2 (no)
KR (1)	KR970701182A (no)
CN (1)	CN1067386C (no)
AU (1)	AU685881B2 (no)
CA (1)	CA2183084A1 (no)
FI (1)	FI950568A (no)
IL (1)	IL112519A0 (no)
NO (1)	NO963331L (no)
NZ (1)	NZ276172A (no)
WO (1)	WO1995021836A1 (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NZ502642A (en) *	1997-07-03	2002-06-28	Du Pont Pharm Co	Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders
US6365589B1 (en)	1998-07-02	2002-04-02	Bristol-Myers Squibb Pharma Company	Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists
UA82395C2 (en) *	2003-08-21	2008-04-10	Оси Фармасьютикалз, Инк.	N-substituted benzimidazolyl c-kit inhibitors
US7442709B2 (en) *	2003-08-21	2008-10-28	Osi Pharmaceuticals, Inc.	N3-substituted imidazopyridine c-Kit inhibitors
CN1839130A (zh)	2003-08-21	2006-09-27	Osi制药公司	N－取代的吡唑基－酰胺基－苯并咪唑基的c－kit抑制剂
JP2008521903A (ja) *	2004-12-01	2008-06-26	オーエスアイ・ファーマスーティカルズ・インコーポレーテッド	Ｎ置換されたベンズイミダゾリルＣ−ｋｉｔ阻害剤及びコンビナトリアルベンゾイミダゾールライブラリー
US8889730B2 (en)	2012-04-10	2014-11-18	Pfizer Inc.	Indole and indazole compounds that activate AMPK
US9394285B2 (en)	2013-03-15	2016-07-19	Pfizer Inc.	Indole and indazole compounds that activate AMPK
JP6800885B2 (ja)	2015-04-29	2020-12-16	ヤンセンファーマシューティカエヌ．ベー．	イミダゾピラジン及びピラゾロピリミジン、並びにａｍｐａ受容体調節物質としてのこれらの使用
US10611730B2 (en)	2015-04-29	2020-04-07	Janssen Pharmaceutica Nv	Benzimidazolone and benzothiazolone compounds and their use as AMPA receptor modulators
SG11201708190UA (en)	2015-04-29	2017-11-29	Janssen Pharmaceutica Nv	Azabenzimidazoles and their use as ampa receptor modulators
EP3288935B1 (en)	2015-04-29	2019-10-30	Janssen Pharmaceutica NV	Indolone compounds and their use as ampa receptor modulators
KR101831553B1 (ko)	2017-01-23	2018-02-22	계명대학교 산학협력단	전이성 유방암의 유용한 신규 화합물 및 이의 의학적 용도

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5066654A (en) *	1990-10-22	1991-11-19	A. H. Robins Company, Incorporated	2-aryl-3-heterocyclicmethyl-3H-imidazo[4,5-b]pyridines as anxiolytics and anticonvulsants
GB9210400D0 (en) *	1992-05-15	1992-07-01	Merck Sharp & Dohme	Therapeutic agents
TW251284B (no) *	1992-11-02	1995-07-11	Pfizer

1994
- 1994-12-08 NZ NZ276172A patent/NZ276172A/en unknown
- 1994-12-08 WO PCT/IB1994/000407 patent/WO1995021836A1/en not_active Application Discontinuation
- 1994-12-08 JP JP7508846A patent/JP2829788B2/ja not_active Expired - Fee Related
- 1994-12-08 CA CA002183084A patent/CA2183084A1/en not_active Abandoned
- 1994-12-08 AU AU10339/95A patent/AU685881B2/en not_active Ceased
- 1994-12-08 US US08/687,555 patent/US5688809A/en not_active Expired - Fee Related
- 1994-12-08 EP EP95900904A patent/EP0743942A1/en not_active Withdrawn
- 1994-12-08 CN CN94194978A patent/CN1067386C/zh not_active Expired - Fee Related
- 1994-12-08 KR KR1019960704346A patent/KR970701182A/ko not_active Application Discontinuation
1995
- 1995-02-02 IL IL11251995A patent/IL112519A0/xx unknown
- 1995-02-09 FI FI950568A patent/FI950568A/fi not_active Application Discontinuation
1996
- 1996-08-09 NO NO963331A patent/NO963331L/no unknown

Also Published As

Publication number	Publication date
FI950568A (fi)	1995-08-11
CA2183084A1 (en)	1995-08-17
WO1995021836A1 (en)	1995-08-17
AU685881B2 (en)	1998-01-29
KR970701182A (ko)	1997-03-17
NZ276172A (en)	1998-02-26
US5688809A (en)	1997-11-18
EP0743942A1 (en)	1996-11-27
NO963331D0 (no)	1996-08-09
JP2829788B2 (ja)	1998-12-02
CN1142823A (zh)	1997-02-12
AU1033995A (en)	1995-08-29
JPH09501949A (ja)	1997-02-25
FI950568A0 (fi)	1995-02-09
NO963331L (no)	1996-10-09
CN1067386C (zh)	2001-06-20

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