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HN2008001532A - Derivados de dihidropirazolopirimidina - Google Patents

Derivados de dihidropirazolopirimidina

Info

Publication number
HN2008001532A
HN2008001532A HN2008001532A HN2008001532A HN2008001532A HN 2008001532 A HN2008001532 A HN 2008001532A HN 2008001532 A HN2008001532 A HN 2008001532A HN 2008001532 A HN2008001532 A HN 2008001532A HN 2008001532 A HN2008001532 A HN 2008001532A
Authority
HN
Honduras
Prior art keywords
derivatives
dihydropirazolopirimidine
quinine
inhibitor
useful
Prior art date
Application number
HN2008001532A
Other languages
English (en)
Inventor
Sakamoto Toshiiro
Sunami Satoshi
Yamamoto Fuyuki
Niyama Kenji
Bamba Makoto
Takashi Keiji
Furuyama Hidetomo
Sagara Takeshi
Otsuki Sachie
Nishibata Toshihide
Yoshizum Takashi
Hirai Hiroshi
Original Assignee
Banyu Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38655640&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HN2008001532(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Banyu Pharma Co Ltd filed Critical Banyu Pharma Co Ltd
Publication of HN2008001532A publication Critical patent/HN2008001532A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

LA PRESENTE INVENCION ES UTIL EN EL CAMPO DE LA MEDICINA. DE FORMA MAS PRECISA, LOS DERIVADOS DE DIHIDROPIRAZOLOPIRIMIDINA DE LA INVENCION SON UTILES EN EL CAMPO DEL TRATAMIENTO DE DIVERSOS CANCERES COMO INHIBIDOR DE QUINASA, ESPECIALMEMNTE COMO INHIBIDOR DE QUINASA WEEL
HN2008001532A 2006-04-27 2008-10-10 Derivados de dihidropirazolopirimidina HN2008001532A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2006124208 2006-04-27

Publications (1)

Publication Number Publication Date
HN2008001532A true HN2008001532A (es) 2009-06-10

Family

ID=38655640

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2008001532A HN2008001532A (es) 2006-04-27 2008-10-10 Derivados de dihidropirazolopirimidina

Country Status (39)

Country Link
US (4) US7935708B2 (es)
EP (2) EP2016080B1 (es)
JP (2) JP4513919B2 (es)
KR (1) KR101409161B1 (es)
CN (1) CN101432284B (es)
AR (1) AR060635A1 (es)
AT (1) ATE475662T1 (es)
AU (1) AU2007244185B2 (es)
BR (1) BRPI0710081A2 (es)
CA (1) CA2650119C (es)
CR (1) CR10359A (es)
CY (2) CY1111069T1 (es)
DE (1) DE602007008085D1 (es)
DK (2) DK2017278T3 (es)
DO (1) DOP2007000084A (es)
EC (1) ECSP088812A (es)
ES (2) ES2348751T3 (es)
GT (1) GT200800211A (es)
HK (1) HK1132498A1 (es)
HN (1) HN2008001532A (es)
HR (2) HRP20100563T1 (es)
HU (1) HUE032987T2 (es)
IL (1) IL194367A (es)
LT (1) LT2017278T (es)
MA (1) MA30428B1 (es)
MX (1) MX2008013063A (es)
MY (1) MY145408A (es)
NO (1) NO341617B1 (es)
NZ (1) NZ571196A (es)
PE (1) PE20080695A1 (es)
PL (2) PL2017278T3 (es)
PT (2) PT2016080E (es)
RU (1) RU2437885C2 (es)
SI (2) SI2016080T1 (es)
SV (1) SV2009003060A (es)
TW (1) TWI409262B (es)
UA (1) UA96152C2 (es)
WO (2) WO2007126122A1 (es)
ZA (1) ZA200807748B (es)

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CN113735863A (zh) * 2021-09-29 2021-12-03 武汉九州钰民医药科技有限公司 Wee1抑制剂adavosertib的制备工艺
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