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FI111263B - Uudet erytromysiinijohdannaiset, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä sekä menetelmässä käytettävät välituoteamiinit - Google Patents

Uudet erytromysiinijohdannaiset, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä sekä menetelmässä käytettävät välituoteamiinit Download PDF

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Publication number
FI111263B
FI111263B FI964395A FI964395A FI111263B FI 111263 B FI111263 B FI 111263B FI 964395 A FI964395 A FI 964395A FI 964395 A FI964395 A FI 964395A FI 111263 B FI111263 B FI 111263B
Authority
FI
Finland
Prior art keywords
pharmaceuticals
preparation
amines used
erythromycin derivatives
intermediate amines
Prior art date
Application number
FI964395A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI964395A0 (fi
FI964395A (fi
Inventor
Constantin Agouridas
Jean-Francois Chantot
Alexis Denis
D Ambrieres Solange Gouin
Martret Odile Le
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of FI964395A0 publication Critical patent/FI964395A0/fi
Publication of FI964395A publication Critical patent/FI964395A/fi
Application granted granted Critical
Publication of FI111263B publication Critical patent/FI111263B/fi

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Indole Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
FI964395A 1994-05-03 1996-10-31 Uudet erytromysiinijohdannaiset, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä sekä menetelmässä käytettävät välituoteamiinit FI111263B (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9405368A FR2719587B1 (fr) 1994-05-03 1994-05-03 Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
PCT/FR1995/000565 WO1995029929A1 (fr) 1994-05-03 1995-05-02 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (3)

Publication Number Publication Date
FI964395A0 FI964395A0 (fi) 1996-10-31
FI964395A FI964395A (fi) 1996-10-31
FI111263B true FI111263B (fi) 2003-06-30

Family

ID=9462785

Family Applications (1)

Application Number Title Priority Date Filing Date
FI964395A FI111263B (fi) 1994-05-03 1996-10-31 Uudet erytromysiinijohdannaiset, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä sekä menetelmässä käytettävät välituoteamiinit

Country Status (43)

Country Link
US (2) US5635485A (xx)
EP (1) EP0680967B1 (xx)
JP (4) JP2992540B2 (xx)
KR (1) KR100312267B1 (xx)
CN (2) CN1052984C (xx)
AP (1) AP558A (xx)
AT (1) ATE172203T1 (xx)
AU (1) AU684027B2 (xx)
BG (1) BG63087B1 (xx)
BR (1) BR9507700A (xx)
CA (1) CA2189271C (xx)
CZ (1) CZ293455B6 (xx)
DE (2) DE10299001I1 (xx)
DK (1) DK0680967T3 (xx)
DZ (1) DZ1878A1 (xx)
EE (1) EE03263B1 (xx)
ES (1) ES2122472T3 (xx)
FI (1) FI111263B (xx)
FR (1) FR2719587B1 (xx)
GE (1) GEP19991538B (xx)
HK (1) HK1010732A1 (xx)
HU (2) HU219599B (xx)
IL (1) IL113245A (xx)
LU (1) LU90872I2 (xx)
LV (1) LV11739B (xx)
MA (1) MA23534A1 (xx)
MD (1) MD1233C2 (xx)
NL (1) NL300077I1 (xx)
NO (2) NO308853B1 (xx)
NZ (1) NZ285416A (xx)
OA (1) OA10319A (xx)
PL (1) PL182034B1 (xx)
RO (1) RO113350B1 (xx)
RU (1) RU2144036C1 (xx)
SI (1) SI0680967T1 (xx)
SK (1) SK281707B6 (xx)
TJ (1) TJ313B (xx)
TN (1) TNSN95049A1 (xx)
TW (1) TW341573B (xx)
UA (1) UA51618C2 (xx)
WO (1) WO1995029929A1 (xx)
YU (1) YU49235B (xx)
ZA (1) ZA953501B (xx)

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Also Published As

Publication number Publication date
WO1995029929A1 (fr) 1995-11-09
TNSN95049A1 (fr) 1996-02-06
CN1052984C (zh) 2000-05-31
KR100312267B1 (ko) 2002-06-22
NO964654D0 (no) 1996-11-04
LU90872I2 (fr) 2002-03-12
AP9500744A0 (en) 1995-07-31
ATE172203T1 (de) 1998-10-15
SK140296A3 (en) 1998-04-08
JP4658902B2 (ja) 2011-03-23
DE10299001I2 (de) 2012-07-05
YU27095A (sh) 1998-05-15
MD1233C2 (ro) 2000-10-31
BG63087B1 (bg) 2001-03-30
TJ313B (en) 2001-08-06
FI964395A0 (fi) 1996-10-31
US6100404A (en) 2000-08-08
UA51618C2 (uk) 2002-12-16
LV11739A (lv) 1997-04-20
HK1010732A1 (en) 1999-06-25
JP4750755B2 (ja) 2011-08-17
CZ293455B6 (cs) 2004-05-12
NO2001027I1 (no) 2002-01-28
RO113350B1 (ro) 1998-06-30
CA2189271C (fr) 2005-12-27
DK0680967T3 (da) 1999-06-23
RU2144036C1 (ru) 2000-01-10
CN1151746A (zh) 1997-06-11
DE69505296T2 (de) 1999-04-22
IL113245A0 (en) 1995-07-31
BG100951A (en) 1997-08-29
CN1088709C (zh) 2002-08-07
MD1233B1 (en) 1999-05-31
CN1229082A (zh) 1999-09-22
OA10319A (fr) 1997-10-07
NZ285416A (en) 1997-07-27
FR2719587B1 (fr) 1996-07-12
MA23534A1 (fr) 1995-12-31
JP3998828B2 (ja) 2007-10-31
SI0680967T1 (en) 1999-02-28
JPH11152296A (ja) 1999-06-08
JPH0853489A (ja) 1996-02-27
HU227493B1 (en) 2011-07-28
HU9603038D0 (en) 1997-01-28
NL300077I1 (nl) 2002-03-01
EE03263B1 (et) 2000-04-17
JP2992540B2 (ja) 1999-12-20
DE69505296D1 (de) 1998-11-19
NO964654L (no) 1996-11-04
CZ321496A3 (en) 1997-08-13
FI964395A (fi) 1996-10-31
HU219599B (hu) 2001-05-28
EP0680967B1 (fr) 1998-10-14
BR9507700A (pt) 1997-08-19
AP558A (en) 1996-11-07
MX9605208A (es) 1997-09-30
GEP19991538B (en) 1999-03-05
TW341573B (en) 1998-10-01
SK281707B6 (sk) 2001-07-10
EP0680967A1 (fr) 1995-11-08
US5635485A (en) 1997-06-03
LV11739B (en) 1997-08-20
AU2449995A (en) 1995-11-29
FR2719587A1 (fr) 1995-11-10
PL182034B1 (pl) 2001-10-31
HUT75698A (en) 1997-05-28
JP2007269810A (ja) 2007-10-18
PL317071A1 (en) 1997-03-03
CA2189271A1 (fr) 1995-11-09
ZA953501B (en) 1996-05-02
DE10299001I1 (de) 2012-07-05
HU9904687D0 (en) 2000-03-28
YU49235B (sh) 2004-12-31
NO308853B1 (no) 2000-11-06
DZ1878A1 (fr) 2002-02-17
IL113245A (en) 1999-11-30
ES2122472T3 (es) 1998-12-16
JP2007045847A (ja) 2007-02-22
AU684027B2 (en) 1997-11-27

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