FI111263B - Uudet erytromysiinijohdannaiset, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä sekä menetelmässä käytettävät välituoteamiinit - Google Patents
Uudet erytromysiinijohdannaiset, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä sekä menetelmässä käytettävät välituoteamiinit Download PDFInfo
- Publication number
- FI111263B FI111263B FI964395A FI964395A FI111263B FI 111263 B FI111263 B FI 111263B FI 964395 A FI964395 A FI 964395A FI 964395 A FI964395 A FI 964395A FI 111263 B FI111263 B FI 111263B
- Authority
- FI
- Finland
- Prior art keywords
- pharmaceuticals
- preparation
- amines used
- erythromycin derivatives
- intermediate amines
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Virology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Indole Compounds (AREA)
- Quinoline Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pyrrole Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9405368A FR2719587B1 (fr) | 1994-05-03 | 1994-05-03 | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
PCT/FR1995/000565 WO1995029929A1 (fr) | 1994-05-03 | 1995-05-02 | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
Publications (3)
Publication Number | Publication Date |
---|---|
FI964395A0 FI964395A0 (fi) | 1996-10-31 |
FI964395A FI964395A (fi) | 1996-10-31 |
FI111263B true FI111263B (fi) | 2003-06-30 |
Family
ID=9462785
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI964395A FI111263B (fi) | 1994-05-03 | 1996-10-31 | Uudet erytromysiinijohdannaiset, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä sekä menetelmässä käytettävät välituoteamiinit |
Country Status (43)
Country | Link |
---|---|
US (2) | US5635485A (xx) |
EP (1) | EP0680967B1 (xx) |
JP (4) | JP2992540B2 (xx) |
KR (1) | KR100312267B1 (xx) |
CN (2) | CN1052984C (xx) |
AP (1) | AP558A (xx) |
AT (1) | ATE172203T1 (xx) |
AU (1) | AU684027B2 (xx) |
BG (1) | BG63087B1 (xx) |
BR (1) | BR9507700A (xx) |
CA (1) | CA2189271C (xx) |
CZ (1) | CZ293455B6 (xx) |
DE (2) | DE10299001I1 (xx) |
DK (1) | DK0680967T3 (xx) |
DZ (1) | DZ1878A1 (xx) |
EE (1) | EE03263B1 (xx) |
ES (1) | ES2122472T3 (xx) |
FI (1) | FI111263B (xx) |
FR (1) | FR2719587B1 (xx) |
GE (1) | GEP19991538B (xx) |
HK (1) | HK1010732A1 (xx) |
HU (2) | HU219599B (xx) |
IL (1) | IL113245A (xx) |
LU (1) | LU90872I2 (xx) |
LV (1) | LV11739B (xx) |
MA (1) | MA23534A1 (xx) |
MD (1) | MD1233C2 (xx) |
NL (1) | NL300077I1 (xx) |
NO (2) | NO308853B1 (xx) |
NZ (1) | NZ285416A (xx) |
OA (1) | OA10319A (xx) |
PL (1) | PL182034B1 (xx) |
RO (1) | RO113350B1 (xx) |
RU (1) | RU2144036C1 (xx) |
SI (1) | SI0680967T1 (xx) |
SK (1) | SK281707B6 (xx) |
TJ (1) | TJ313B (xx) |
TN (1) | TNSN95049A1 (xx) |
TW (1) | TW341573B (xx) |
UA (1) | UA51618C2 (xx) |
WO (1) | WO1995029929A1 (xx) |
YU (1) | YU49235B (xx) |
ZA (1) | ZA953501B (xx) |
Families Citing this family (85)
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WO1997001539A1 (en) * | 1995-06-27 | 1997-01-16 | Takeda Chemical Industries, Ltd. | 4-acylamino(halogeno) alkyl-quinoline derivatives, their preparation and their use as melatonin agonists |
FR2742757B1 (fr) * | 1995-12-22 | 1998-01-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
UA51730C2 (uk) * | 1996-09-04 | 2002-12-16 | Ебботт Лабораторіз | 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців |
KR100568455B1 (ko) * | 1996-09-04 | 2006-04-07 | 아보트 러보러터리즈 | 항균 활성을 지닌 6-o-치환된 케톨라이드 |
FR2757168B1 (fr) * | 1996-12-12 | 1999-06-11 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
FR2760017B1 (fr) * | 1997-02-27 | 1999-04-30 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments |
US5780605A (en) * | 1997-09-08 | 1998-07-14 | Abbott Laboratories | 6,9-bridged erythromycin derivatives |
FR2771008B1 (fr) * | 1997-11-17 | 2000-04-28 | Hoechst Marion Roussel Inc | Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose |
JP4573925B2 (ja) * | 1998-07-09 | 2010-11-04 | アベンティス・ファーマ・ソシエテ・アノニム | 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用 |
FR2781484B1 (fr) * | 1998-07-21 | 2001-08-10 | Hoechst Marion Roussel Inc | Nouveaux derives de la 6-deoxy erythromycine, leur procede de preparation et leur application comme medicaments |
EP1115732B1 (en) * | 1998-09-22 | 2005-06-29 | Pfizer Products Inc. | Carbamate and carbazate ketolide antibiotics |
FR2785612A1 (fr) * | 1998-11-10 | 2000-05-12 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
FR2786188B1 (fr) * | 1998-11-24 | 2002-10-31 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur applicaion comme medicaments |
TW526202B (en) * | 1998-11-27 | 2003-04-01 | Shionogi & Amp Co | Broad spectrum cephem having benzo[4,5-b]pyridium methyl group of antibiotic activity |
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CA2370743A1 (en) | 1999-04-16 | 2000-10-26 | Dennis Hlasta | Ketolide antibacterials |
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CN105524132B (zh) * | 2014-09-30 | 2019-07-02 | 中国医学科学院药物研究所 | 含有喹啉取代基的红霉素a酮内酯类抗生素衍生物、其制备方法及应用 |
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FR2697524B1 (fr) * | 1992-11-05 | 1994-12-23 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
TW444018B (en) * | 1992-12-17 | 2001-07-01 | Pfizer | Pyrazolopyrimidines |
HRP930014A2 (en) * | 1993-01-08 | 1994-08-31 | Pliva Pharm & Chem Works | 9-deoxo-9a-aza-11-deoxy-9a-homoeritromycin a 9a, 11-cyclic carbamates |
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1994
- 1994-05-03 FR FR9405368A patent/FR2719587B1/fr not_active Expired - Lifetime
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1995
- 1995-02-05 UA UA96104110A patent/UA51618C2/uk unknown
- 1995-04-04 IL IL11324595A patent/IL113245A/xx not_active IP Right Cessation
- 1995-04-21 US US08/426,067 patent/US5635485A/en not_active Expired - Lifetime
- 1995-04-27 MA MA23866A patent/MA23534A1/fr unknown
- 1995-04-28 YU YU27095A patent/YU49235B/sh unknown
- 1995-05-01 JP JP7128791A patent/JP2992540B2/ja not_active Expired - Lifetime
- 1995-05-02 AT AT95400987T patent/ATE172203T1/de active
- 1995-05-02 BR BR9507700A patent/BR9507700A/pt not_active IP Right Cessation
- 1995-05-02 HU HU9904687A patent/HU219599B/hu unknown
- 1995-05-02 WO PCT/FR1995/000565 patent/WO1995029929A1/fr active IP Right Grant
- 1995-05-02 SK SK1402-96A patent/SK281707B6/sk not_active IP Right Cessation
- 1995-05-02 HU HU9603038A patent/HU227493B1/hu unknown
- 1995-05-02 DE DE2002199001 patent/DE10299001I1/de active Granted
- 1995-05-02 KR KR1019960706191A patent/KR100312267B1/ko not_active IP Right Cessation
- 1995-05-02 DZ DZ950049A patent/DZ1878A1/fr active
- 1995-05-02 CN CN95193911A patent/CN1052984C/zh not_active Expired - Lifetime
- 1995-05-02 ES ES95400987T patent/ES2122472T3/es not_active Expired - Lifetime
- 1995-05-02 AU AU24499/95A patent/AU684027B2/en not_active Expired
- 1995-05-02 RO RO96-02081A patent/RO113350B1/ro unknown
- 1995-05-02 RU RU96123129A patent/RU2144036C1/ru active
- 1995-05-02 GE GEAP19953425A patent/GEP19991538B/en unknown
- 1995-05-02 NZ NZ285416A patent/NZ285416A/en not_active IP Right Cessation
- 1995-05-02 CZ CZ19963214A patent/CZ293455B6/cs not_active IP Right Cessation
- 1995-05-02 CA CA002189271A patent/CA2189271C/fr not_active Expired - Lifetime
- 1995-05-02 EE EE9600151A patent/EE03263B1/xx active Protection Beyond IP Right Term
- 1995-05-02 PL PL95317071A patent/PL182034B1/pl unknown
- 1995-05-02 ZA ZA953501A patent/ZA953501B/xx unknown
- 1995-05-02 DK DK95400987T patent/DK0680967T3/da active
- 1995-05-02 EP EP95400987A patent/EP0680967B1/fr not_active Expired - Lifetime
- 1995-05-02 MD MD97-0010A patent/MD1233C2/ro unknown
- 1995-05-02 DE DE69505296T patent/DE69505296T2/de not_active Expired - Lifetime
- 1995-05-02 TN TNTNSN95049A patent/TNSN95049A1/fr unknown
- 1995-05-02 AP APAP/P/1995/000744A patent/AP558A/en active
- 1995-05-02 SI SI9530184T patent/SI0680967T1/xx unknown
- 1995-06-29 TW TW084106692A patent/TW341573B/zh not_active IP Right Cessation
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1996
- 1996-10-31 FI FI964395A patent/FI111263B/fi not_active IP Right Cessation
- 1996-11-01 OA OA60917A patent/OA10319A/fr unknown
- 1996-11-01 LV LVP-96-421A patent/LV11739B/lv unknown
- 1996-11-01 TJ TJ96000417A patent/TJ313B/xx unknown
- 1996-11-01 BG BG100951A patent/BG63087B1/bg unknown
- 1996-11-04 NO NO964654A patent/NO308853B1/no not_active IP Right Cessation
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1997
- 1997-01-09 US US08/780,861 patent/US6100404A/en not_active Expired - Lifetime
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1998
- 1998-08-24 JP JP25181798A patent/JP3998828B2/ja not_active Expired - Lifetime
- 1998-11-05 HK HK98111758A patent/HK1010732A1/xx not_active IP Right Cessation
- 1998-12-07 CN CN98123072A patent/CN1088709C/zh not_active Expired - Lifetime
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2001
- 2001-12-28 NL NL300077C patent/NL300077I1/nl unknown
- 2001-12-28 NO NO2001027C patent/NO2001027I1/no unknown
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2002
- 2002-01-08 LU LU90872C patent/LU90872I2/xx unknown
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2006
- 2006-11-21 JP JP2006314281A patent/JP4658902B2/ja not_active Expired - Lifetime
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2007
- 2007-06-06 JP JP2007150991A patent/JP4750755B2/ja not_active Expired - Lifetime
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
GB | Transfer or assigment of application |
Owner name: HOECHST MARION ROUSSEL |
|
SPCF | Supplementary protection certificate application filed |
Spc suppl protection certif: L20030009 |
|
SPCG | Supplementary protection certificate granted |
Spc suppl protection certif: NUMBER:214 |
|
MA | Patent expired |