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ES8607258A1 - Un procedimiento para la preparacion de derivados de triazol - Google Patents

Un procedimiento para la preparacion de derivados de triazol

Info

Publication number
ES8607258A1
ES8607258A1 ES549298A ES549298A ES8607258A1 ES 8607258 A1 ES8607258 A1 ES 8607258A1 ES 549298 A ES549298 A ES 549298A ES 549298 A ES549298 A ES 549298A ES 8607258 A1 ES8607258 A1 ES 8607258A1
Authority
ES
Spain
Prior art keywords
antifungal agents
triazole antifungal
triazole
fluoro
chloro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES549298A
Other languages
English (en)
Other versions
ES549298A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Pfizer Corp
Original Assignee
Pfizer Corp Belgium
Pfizer Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp filed Critical Pfizer Corp Belgium
Publication of ES8607258A1 publication Critical patent/ES8607258A1/es
Publication of ES549298A0 publication Critical patent/ES549298A0/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Environmental Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)

Abstract

METODO DE OBTENCION DE DERIVADOS DE TRIAZOL DE FORMULA (I), DONDE R Y R1 SON CADA UNO UN GRUPO FENILO CON 1 A 3 SUSTITUYENTES, SELECCIONADOS DE FORMA INDEPENDIENTE ENTRE: F, CL, BR, I, CF3, ALQUILO DE 1 A 4 ATOMOS DE C; O BIEN R ES UN GRUPO 5-CLOROPIRID-2-ILO; X REPRESENTA: -OH,-F,-CL O -BR. CONSISTENTE EN HACER REACCIONAR UNA CETONA CON UN DERIVADO DE GRIGNARD O DE LITIO. LA REACCION SE LLEVA A CABO EN AGITACION Y A TEMPERATURA AMBIENTE, DURANTE ALGUNAS HORAS, Y EN UN DISOLVENTE ORGANICO (ETER DIETILICO O TETRAHIDROFURANO); OBTENIENDOSE EL PRODUCTO DE FORMULA (I) QUE ES AISLADO Y PURIFICADO POR METODOS CONVENCIONALES. DE APLICACION AGRICOLA Y FARMACEUTICA POR SU ACTIVIDAD ANTIFUNGICA.
ES549298A 1984-11-27 1985-11-26 Un procedimiento para la preparacion de derivados de triazol Expired ES8607258A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB848429932A GB8429932D0 (en) 1984-11-27 1984-11-27 Triazole antifungal agents

Publications (2)

Publication Number Publication Date
ES8607258A1 true ES8607258A1 (es) 1986-05-16
ES549298A0 ES549298A0 (es) 1986-05-16

Family

ID=10570335

Family Applications (1)

Application Number Title Priority Date Filing Date
ES549298A Expired ES8607258A1 (es) 1984-11-27 1985-11-26 Un procedimiento para la preparacion de derivados de triazol

Country Status (19)

Country Link
US (1) US4767777A (es)
EP (1) EP0183494B1 (es)
JP (1) JPS61137868A (es)
KR (1) KR870001381B1 (es)
AT (1) ATE39923T1 (es)
AU (1) AU556517B2 (es)
CA (1) CA1276935C (es)
DE (1) DE3567455D1 (es)
DK (1) DK162990C (es)
ES (1) ES8607258A1 (es)
FI (1) FI854660A (es)
GB (1) GB8429932D0 (es)
GR (1) GR852833B (es)
HU (1) HUT41394A (es)
IE (1) IE58146B1 (es)
IL (1) IL77151A0 (es)
PH (1) PH21332A (es)
PL (1) PL145094B1 (es)
PT (1) PT81556B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8414519D0 (en) * 1984-06-07 1984-07-11 Pfizer Ltd Triazole antifungal agents
GB8511344D0 (en) * 1985-05-03 1985-06-12 Ici Plc Heterocyclic compounds
DE3608727A1 (de) * 1986-03-15 1987-09-17 Hoechst Ag 1,1-disubstituierte cyclopropanderivate, verfahren zu ihrer herstellung sowie ihre verwendung als antimykotika oder als zwischenprodukte
US5247094A (en) * 1990-01-24 1993-09-21 Bayer Aktiengesellschaft 1-(3- or 5-halo-1,2,4-triazol-1-yl)ethyl phenyl ketone intermediates
US5223178A (en) * 1990-12-10 1993-06-29 Rohm And Haas Company Use of certain triazoles to protect materials from fungal attack, articles and compositions
EP0597049A1 (en) * 1992-03-04 1994-05-18 Jemlan, Inc. Antifungal agents
TWI290549B (en) * 2000-06-02 2007-12-01 Astrazeneca Ab Process for the preparation of cyclopropyl carboxylic acid ester and derivatives
AR075257A1 (es) 2008-02-01 2011-03-23 Hexima Ltd Sistema de proteccion de plantas contra la infeccion por agentes patogenos
US9889184B2 (en) 2008-08-05 2018-02-13 Hexima Limited Anti-pathogen systems
BR112013020131A8 (pt) 2011-02-07 2018-01-09 Hexima Ltd defensinas de plantas modificadas úteis como agentes antipatogênicas

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH658654A5 (de) * 1983-03-04 1986-11-28 Sandoz Ag Azolderivate, verfahren zu ihrer herstellung und mittel die diese verbindungen enthalten.
NL8402755A (nl) * 1983-09-22 1985-04-16 Sandoz Ag Azool-derivaten, werkwijze voor het bereiden daarvan, preparaten die ze bevatten, en toepassing daarvan.
GB8414519D0 (en) * 1984-06-07 1984-07-11 Pfizer Ltd Triazole antifungal agents
DE3440114A1 (de) * 1984-11-02 1986-05-07 Bayer Ag, 5090 Leverkusen Antimykotische mittel
CN1008735B (zh) * 1984-11-02 1990-07-11 拜尔公司 以取代的氮杂茂基甲基-环丙基-甲醇衍生物为活性成分的组合物

Also Published As

Publication number Publication date
AU556517B2 (en) 1986-11-06
PH21332A (en) 1987-10-13
KR870001381B1 (ko) 1987-07-24
PT81556A (en) 1985-12-01
JPS61137868A (ja) 1986-06-25
GR852833B (es) 1986-03-27
US4767777A (en) 1988-08-30
DK162990B (da) 1992-01-06
ATE39923T1 (de) 1989-01-15
HUT41394A (en) 1987-04-28
KR860004036A (ko) 1986-06-16
FI854660A0 (fi) 1985-11-26
GB8429932D0 (en) 1985-01-03
DK545385D0 (da) 1985-11-26
EP0183494A3 (en) 1986-12-30
PT81556B (pt) 1988-03-03
EP0183494B1 (en) 1989-01-11
PL256439A1 (en) 1987-02-23
DK162990C (da) 1992-05-25
DK545385A (da) 1986-05-28
CA1276935C (en) 1990-11-27
FI854660A (fi) 1986-05-28
IE58146B1 (en) 1993-07-14
AU5035985A (en) 1986-06-05
PL145094B1 (en) 1988-08-31
EP0183494A2 (en) 1986-06-04
IE852970L (en) 1986-05-27
ES549298A0 (es) 1986-05-16
JPH0533702B2 (es) 1993-05-20
DE3567455D1 (en) 1989-02-16
IL77151A0 (en) 1986-04-29

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