DK174280B1 - Fremgangsmåde til fremstilling af allyl-2-thioxopenam-3-carboxylat-forbindelser og mellemprodukter ved fremgangsmåden - Google Patents

Fremgangsmåde til fremstilling af allyl-2-thioxopenam-3-carboxylat-forbindelser og mellemprodukter ved fremgangsmåden Download PDF

Info

Publication number: DK174280B1
Authority: DK; Denmark
Prior art keywords: product; mmol; preparation; compound; formula
Prior art date: 1986-06-02

Application number

DK198702798A

Other languages

Danish (da)

English (en)

Other versions

DK279887A (da

DK279887D0 (da

Inventor

Katherine Elizabeth Brighty

David Louis Lindner

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-06-02

Filing date

1987-06-01

Publication date

2002-11-04

1987-06-01 Application filed by Pfizer filed Critical Pfizer

1987-06-01 Publication of DK279887D0 publication Critical patent/DK279887D0/da

1987-12-03 Publication of DK279887A publication Critical patent/DK279887A/da

2002-11-04 Application granted granted Critical

2002-11-04 Publication of DK174280B1 publication Critical patent/DK174280B1/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Electroluminescent Light Sources (AREA)
Diaphragms For Electromechanical Transducers (AREA)
Steroid Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

DK198702798A 1986-06-02 1987-06-01 Fremgangsmåde til fremstilling af allyl-2-thioxopenam-3-carboxylat-forbindelser og mellemprodukter ved fremgangsmåden DK174280B1 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US86976086		1986-06-02
US06/869,760 US4782145A (en)	1986-06-02	1986-06-02	Process for penem derivatives

Publications (3)

Publication Number	Publication Date
DK279887D0 DK279887D0 (da)	1987-06-01
DK279887A DK279887A (da)	1987-12-03
DK174280B1 true DK174280B1 (da)	2002-11-04

Family

ID=25354215

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK198702798A DK174280B1 (da)	1986-06-02	1987-06-01	Fremgangsmåde til fremstilling af allyl-2-thioxopenam-3-carboxylat-forbindelser og mellemprodukter ved fremgangsmåden

Country Status (19)

Country	Link
US (1)	US4782145A (ja)
EP (1)	EP0249358B1 (ja)
JP (1)	JPS62294685A (ja)
KR (1)	KR890004560B1 (ja)
AT (1)	ATE56452T1 (ja)
AU (1)	AU574610B2 (ja)
CA (1)	CA1279312C (ja)
DE (1)	DE3764875D1 (ja)
DK (1)	DK174280B1 (ja)
ES (1)	ES2018022B3 (ja)
FI (1)	FI87649C (ja)
GR (1)	GR3000862T3 (ja)
HU (1)	HU196601B (ja)
IE (1)	IE59871B1 (ja)
IL (1)	IL82695A0 (ja)
NZ (1)	NZ220498A (ja)
PT (1)	PT84983B (ja)
YU (1)	YU46208B (ja)
ZA (1)	ZA873876B (ja)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4895940A (en) *	1988-10-19	1990-01-23	Pfizer Inc.	Process for the preparation of penems
US4992543A (en) *	1988-10-19	1991-02-12	Pfizer Inc.	Penem derivatives
US5191075A (en) *	1988-10-19	1993-03-02	Pfizer Inc	Process for the preparation of penems
JP2569455B2 (ja) *	1992-03-06	1997-01-08	田辺製薬株式会社	β−ラクタム誘導体の製法
US5399679A (en) *	1992-06-16	1995-03-21	Farmitalia Carlo Erba S.R.L.	(1'R,3S,4R)4-acylthio azetidinones
US5698547A (en) *	1994-04-01	1997-12-16	Microcide Pharmaceuticals, Inc.	Cephalosporin antibiotics
US5688786A (en) *	1994-04-01	1997-11-18	Microcide Pharmaceuticals, Inc.	β-lactam antibiotics
BR9507267A (pt) *	1994-04-01	1997-09-23	Microcide Pharmaceuticals Inc	Antibióticos de cefalosporina

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3175042D1 (en) *	1980-11-06	1986-09-04	Hoechst Uk Ltd	7-oxo-4-thia-1-aza(3,2,0)heptane and 7-oxo-4-thia-1-aza(3,2,0)hept-2-ene derivatives
DE3372773D1 (de) *	1982-03-26	1987-09-03	Hoechst Uk Ltd	7-oxo-4-thia-1-azabicyclo(3,2,0)heptane derivatives
EP0110280B1 (en) *	1982-11-29	1994-10-12	Schering Corporation	Process for the production of penem compounds
US4530793A (en) *	1982-11-29	1985-07-23	Schering Corporation	Processes for the production of penems
FI77459C (fi) *	1982-12-08	1989-03-10	Erba Farmitalia	Foerfarande foer framstaellning av (5r)-penemderivat.
US4695626A (en) *	1986-07-29	1987-09-22	Pfizer Inc.	1-aza-4,5-dithiabicyclo [4.2.0] oct-2-en-8-one-2 carboxylate esters

1986
- 1986-06-02 US US06/869,760 patent/US4782145A/en not_active Expired - Lifetime
1987
- 1987-05-19 FI FI872195A patent/FI87649C/fi not_active IP Right Cessation
- 1987-05-27 ES ES87304669T patent/ES2018022B3/es not_active Expired - Lifetime
- 1987-05-27 EP EP87304669A patent/EP0249358B1/en not_active Expired - Lifetime
- 1987-05-27 AT AT87304669T patent/ATE56452T1/de not_active IP Right Cessation
- 1987-05-27 DE DE8787304669T patent/DE3764875D1/de not_active Expired - Fee Related
- 1987-05-29 ZA ZA873876A patent/ZA873876B/xx unknown
- 1987-05-29 IE IE143087A patent/IE59871B1/en not_active IP Right Cessation
- 1987-05-29 IL IL82695A patent/IL82695A0/xx not_active IP Right Cessation
- 1987-05-29 NZ NZ220498A patent/NZ220498A/xx unknown
- 1987-05-29 CA CA000538429A patent/CA1279312C/en not_active Expired - Fee Related
- 1987-06-01 KR KR1019870005506A patent/KR890004560B1/ko not_active IP Right Cessation
- 1987-06-01 DK DK198702798A patent/DK174280B1/da not_active IP Right Cessation
- 1987-06-01 JP JP62135002A patent/JPS62294685A/ja active Granted
- 1987-06-01 YU YU100087A patent/YU46208B/sh unknown
- 1987-06-01 PT PT84983A patent/PT84983B/pt not_active IP Right Cessation
- 1987-06-01 AU AU73695/87A patent/AU574610B2/en not_active Ceased
- 1987-06-01 HU HU872511A patent/HU196601B/hu not_active IP Right Cessation
1990
- 1990-09-24 GR GR90400693T patent/GR3000862T3/el unknown

Also Published As

Publication number	Publication date
EP0249358B1 (en)	1990-09-12
IL82695A0 (en)	1987-11-30
HU196601B (en)	1988-12-28
HUT45066A (en)	1988-05-30
DK279887A (da)	1987-12-03
ZA873876B (en)	1987-11-30
GR3000862T3 (en)	1991-11-15
KR890004560B1 (ko)	1989-11-15
CA1279312C (en)	1991-01-22
IE59871B1 (en)	1994-04-20
FI87649B (fi)	1992-10-30
AU574610B2 (en)	1988-07-07
JPH0544950B2 (ja)	1993-07-07
FI87649C (fi)	1993-02-10
PT84983A (en)	1987-07-01
FI872195A (fi)	1987-12-03
FI872195A0 (fi)	1987-05-19
JPS62294685A (ja)	1987-12-22
YU100087A (en)	1988-12-31
AU7369587A (en)	1987-12-10
PT84983B (pt)	1990-02-08
ES2018022B3 (es)	1991-03-16
EP0249358A1 (en)	1987-12-16
ATE56452T1 (de)	1990-09-15
IE871430L (en)	1987-12-02
US4782145A (en)	1988-11-01
DK279887D0 (da)	1987-06-01
KR880000442A (ko)	1988-03-25
NZ220498A (en)	1989-08-29
DE3764875D1 (de)	1990-10-18
YU46208B (sh)	1993-05-28

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Date	Code	Title	Description
2005-01-31	PBP	Patent lapsed	Country of ref document: DK