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BRPI0611409A8 - Preparação oral compreendendo lurasidona - Google Patents

Preparação oral compreendendo lurasidona

Info

Publication number
BRPI0611409A8
BRPI0611409A8 BRPI0611409A BRPI0611409A BRPI0611409A8 BR PI0611409 A8 BRPI0611409 A8 BR PI0611409A8 BR PI0611409 A BRPI0611409 A BR PI0611409A BR PI0611409 A BRPI0611409 A BR PI0611409A BR PI0611409 A8 BRPI0611409 A8 BR PI0611409A8
Authority
BR
Brazil
Prior art keywords
preparation
oral preparation
lurasidone
water
preparation including
Prior art date
Application number
BRPI0611409A
Other languages
English (en)
Inventor
Fujihara Kazuyuki
Original Assignee
Dainippon Sumitomo Pharma Co
Sumitomo Dainippon Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37452103&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0611409(A8) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dainippon Sumitomo Pharma Co, Sumitomo Dainippon Pharma Co Ltd filed Critical Dainippon Sumitomo Pharma Co
Publication of BRPI0611409A2 publication Critical patent/BRPI0611409A2/pt
Publication of BRPI0611409A8 publication Critical patent/BRPI0611409A8/pt
Publication of BRPI0611409B1 publication Critical patent/BRPI0611409B1/pt
Publication of BRPI0611409B8 publication Critical patent/BRPI0611409B8/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nutrition Science (AREA)
  • Inorganic Chemistry (AREA)
  • Physiology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

PREPARAÇÃO ORAL E MÉTODO DE GRANULAÇÃO DE UMA MISTURA EM PÓ. A presente invenção refere-se a uma preparação para administração oral incluindo: um amido pré-gelatinizado contendo cloridrato de N-[4-[4-(1 ,2-benzisotiazol-3-il)-1-piperazinil]-(2R,3R)-2,3-tetrametieno-butil]-(1 'R,2'S,3'R,4'S)-2,3-biciclo[2,2,1]heptanodicarboxiimida (lurasidona) representado pela fórmula (1) como ingrediente ativo; um excipiente solúvel em água; e um ligante polimérico solúvel em água, a preparação apresentando um nível invariante de comportamento em eluição mesmo quando o teor de seu ingrediente ativo é variado.
BRPI0611409A 2005-05-26 2006-05-26 preparação oral compreendendo lurasidona BRPI0611409B8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2005153508 2005-05-26
JP2005-153508 2005-05-26
PCT/JP2006/310571 WO2006126681A1 (ja) 2005-05-26 2006-05-26 医薬品組成物

Publications (4)

Publication Number Publication Date
BRPI0611409A2 BRPI0611409A2 (pt) 2010-11-23
BRPI0611409A8 true BRPI0611409A8 (pt) 2015-12-15
BRPI0611409B1 BRPI0611409B1 (pt) 2020-12-29
BRPI0611409B8 BRPI0611409B8 (pt) 2021-05-25

Family

ID=37452103

Family Applications (2)

Application Number Title Priority Date Filing Date
BR122020005056-0A BR122020005056B1 (pt) 2005-05-26 2006-05-26 Método para preparar uma preparação oral que compreende cloridrato de n-[4-[4-(1,2- benziso-tiazol-3-il)-1-piperazinil]-(2r,3r)-2,3-tetrametileno-butil]-(1r,2s,3r,4s)-2,3-biciclo[2,2,1] heptanodicarboxiimida (lurasidona)
BRPI0611409A BRPI0611409B8 (pt) 2005-05-26 2006-05-26 preparação oral compreendendo lurasidona

Family Applications Before (1)

Application Number Title Priority Date Filing Date
BR122020005056-0A BR122020005056B1 (pt) 2005-05-26 2006-05-26 Método para preparar uma preparação oral que compreende cloridrato de n-[4-[4-(1,2- benziso-tiazol-3-il)-1-piperazinil]-(2r,3r)-2,3-tetrametileno-butil]-(1r,2s,3r,4s)-2,3-biciclo[2,2,1] heptanodicarboxiimida (lurasidona)

Country Status (22)

Country Link
US (5) US8729085B2 (pt)
EP (2) EP2422783B1 (pt)
JP (2) JP4733120B2 (pt)
KR (2) KR101552033B1 (pt)
CN (2) CN101184489B (pt)
AU (1) AU2006250340C1 (pt)
BR (2) BR122020005056B1 (pt)
CA (1) CA2606510C (pt)
CY (2) CY1114118T1 (pt)
DK (2) DK2422783T3 (pt)
ES (2) ES2408687T3 (pt)
FR (1) FR14C0069I2 (pt)
HK (1) HK1108379A1 (pt)
HU (1) HUS1400051I1 (pt)
LU (1) LU92550I2 (pt)
MX (1) MX2007014872A (pt)
NL (1) NL300690I2 (pt)
PL (1) PL1884242T3 (pt)
PT (1) PT1884242E (pt)
RU (1) RU2398586C3 (pt)
SI (1) SI1884242T1 (pt)
WO (1) WO2006126681A1 (pt)

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CN108567758A (zh) * 2017-03-08 2018-09-25 湖南洞庭药业股份有限公司 盐酸鲁拉西酮片剂及其制备方法
CN107875122A (zh) * 2017-12-17 2018-04-06 佛山市弘泰药物研发有限公司 一种盐酸鲁拉西酮自微乳制剂及其制备方法
CN107854445A (zh) * 2017-12-17 2018-03-30 佛山市弘泰药物研发有限公司 一种盐酸鲁拉西酮分散片及其制备方法
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Also Published As

Publication number Publication date
EP1884242B1 (en) 2013-04-17
DK2422783T3 (en) 2015-05-11
BR122020005056A2 (pt) 2010-11-23
EP1884242A1 (en) 2008-02-06
KR20080012306A (ko) 2008-02-11
EP2422783A1 (en) 2012-02-29
BRPI0611409B8 (pt) 2021-05-25
NL300690I2 (nl) 2017-11-02
JP4733120B2 (ja) 2011-07-27
AU2006250340B2 (en) 2012-02-09
US8883794B2 (en) 2014-11-11
CA2606510C (en) 2014-07-22
FR14C0069I2 (fr) 2015-11-20
RU2398586C2 (ru) 2010-09-10
US9555027B2 (en) 2017-01-31
SI1884242T1 (sl) 2013-07-31
KR101380088B1 (ko) 2014-04-10
CN101184489B (zh) 2011-01-19
WO2006126681A1 (ja) 2006-11-30
JP5285105B2 (ja) 2013-09-11
LU92550I2 (fr) 2015-11-02
PL1884242T3 (pl) 2013-09-30
CN102048734A (zh) 2011-05-11
ES2535478T3 (es) 2015-05-12
BRPI0611409B1 (pt) 2020-12-29
FR14C0069I1 (fr) 2014-10-24
JPWO2006126681A1 (ja) 2008-12-25
JP2011126915A (ja) 2011-06-30
CA2606510A1 (en) 2006-11-30
ES2408687T3 (es) 2013-06-21
US20140235651A1 (en) 2014-08-21
MX2007014872A (es) 2008-02-15
RU2007148997A (ru) 2009-07-10
US20090143404A1 (en) 2009-06-04
BR122020005056A8 (pt) 2022-11-22
CY2014039I1 (el) 2016-06-22
CY2014039I2 (el) 2016-06-22
US20180161322A1 (en) 2018-06-14
BRPI0611409A2 (pt) 2010-11-23
KR20130122019A (ko) 2013-11-06
EP2422783B1 (en) 2015-04-08
AU2006250340A1 (en) 2006-11-30
US9907794B2 (en) 2018-03-06
HK1108379A1 (en) 2008-05-09
US20150265611A1 (en) 2015-09-24
RU2398586C3 (ru) 2017-10-04
US20150056284A1 (en) 2015-02-26
CN102048734B (zh) 2013-11-20
US8729085B2 (en) 2014-05-20
HUS1400051I1 (hu) 2016-10-28
CN101184489A (zh) 2008-05-21
KR101552033B1 (ko) 2015-09-09
DK1884242T3 (da) 2013-05-06
PT1884242E (pt) 2013-05-21
AU2006250340C1 (en) 2014-06-12
BR122020005056B1 (pt) 2023-01-10
EP1884242A4 (en) 2009-07-01
CY1114118T1 (el) 2016-06-22

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