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BRPI0417052A - processo para a preparação de compostos - Google Patents

processo para a preparação de compostos

Info

Publication number
BRPI0417052A
BRPI0417052A BRPI0417052-0A BRPI0417052A BRPI0417052A BR PI0417052 A BRPI0417052 A BR PI0417052A BR PI0417052 A BRPI0417052 A BR PI0417052A BR PI0417052 A BRPI0417052 A BR PI0417052A
Authority
BR
Brazil
Prior art keywords
formula
thio
phenyl
compounds
preparation
Prior art date
Application number
BRPI0417052-0A
Other languages
English (en)
Inventor
Gerhard Hamprecht
Michael Punl
Bernd Wolf
Michael Keil
Robert Reinhard
Werner Seitz
Guido Mayer
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of BRPI0417052A publication Critical patent/BRPI0417052A/pt
Publication of BRPI0417052B1 publication Critical patent/BRPI0417052B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/56—One oxygen atom and one sulfur atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

"PROCESSO PARA A PREPARAçãO DE COMPOSTOS". A invenção diz respeito a um método para a produção de 3-fenil(tio)uracilas ou 3-fenilditiouracilas de fórmula (I), mediante a reação de um feniliso(tio)cianato de fórmula (II) com uma enamina de fórmula (III) e opcionalmente a reação em uma etapa adicional da 3-fenil(tio)uracila ou 3fenilditiouracila de fórmula (I) com R¬ 1¬ = R¬ 1a¬, se R¬ 1¬ for hidrogênio, com um agente de aminação de fórmula (IV) para dar 3-fenil(tio)uracilas ou 3-fenilditiouracilas de fórmula (I) com R¬ 1¬ = amina, em que as variáveis R¬ 1¬, R¬ 1a¬, R¬ 2¬, R¬ 3¬, R¬ 4¬, X¬ 1¬, X¬ 2¬, X¬ 3¬, Ar e A L1 são definidas de acordo com a reivindicação 1.
BRPI0417052-0A 2003-12-03 2004-12-01 Processos para a preparação de 3-fenil(tio)uracilas e 3-fenilditiouracilas BRPI0417052B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10356474 2003-12-03
DE10356474.8 2003-12-03
PCT/EP2004/013615 WO2005054208A1 (de) 2003-12-03 2004-12-01 Verfahren zur herstellung von 3-phenyl(thio)uracilen und 3-phenyldithiouracilen

Publications (2)

Publication Number Publication Date
BRPI0417052A true BRPI0417052A (pt) 2007-02-06
BRPI0417052B1 BRPI0417052B1 (pt) 2014-02-25

Family

ID=34638289

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0417052-0A BRPI0417052B1 (pt) 2003-12-03 2004-12-01 Processos para a preparação de 3-fenil(tio)uracilas e 3-fenilditiouracilas

Country Status (12)

Country Link
US (1) US7737275B2 (pt)
EP (1) EP1692115B1 (pt)
JP (1) JP4528306B2 (pt)
KR (1) KR101135263B1 (pt)
CN (1) CN100558714C (pt)
AT (1) ATE381547T1 (pt)
BR (1) BRPI0417052B1 (pt)
DE (1) DE502004005772D1 (pt)
DK (1) DK1692115T3 (pt)
ES (1) ES2295957T3 (pt)
IL (1) IL175713A (pt)
WO (1) WO2005054208A1 (pt)

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US7699852B2 (en) 2003-11-19 2010-04-20 Zimmer Spine, Inc. Fenestrated bone tap and method
SI1893586T1 (sl) * 2005-05-24 2008-12-31 Basf Se Postopek za pripravo 1-alkil-3-feniluracilov
NZ575891A (en) * 2006-10-13 2011-07-29 Basf Se Hydrates of a phenyluracil
WO2008043835A2 (de) 2006-10-13 2008-04-17 Basf Se Kristalline form von 2-chlor-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluormethyl)-1-(2h)-pyrimidinyl]-4-fluor-n-[[methyl-(1-methylethyl)amino]sulfonyl]benzamid
EP2470018A2 (en) 2009-08-27 2012-07-04 Basf Se Aqueous suspension concentrate formulations containing saflufenacil
AU2010288527B2 (en) 2009-08-27 2015-05-14 Basf Se Aqueous concentrate formulations containing saflufenacil and glyphosate
EP2499136B1 (en) 2009-11-13 2013-12-04 Basf Se 3-(3,4-dihydro-2h-benzo[1,4]oxazin-6-yl)-1h-pyrimidin-2,4-dione compounds as herbicides
US8703650B2 (en) 2009-12-09 2014-04-22 Basf Se Liquid suspension concentrate formulations containing saflufenacil
BR112012012586B1 (pt) 2009-12-09 2017-07-25 Basf Se "concentrated formulation of suspension, use of the concentrated formulation of liquid suspension and method to control the understooded vegetation
WO2011104213A2 (de) 2010-02-26 2011-09-01 Bayer Cropscience Ag Herbizide zusammensetzung enthaltend die hydrate von saflufenacil und glyphosate oder glufosinate
CN103130727B (zh) * 2013-02-27 2015-07-08 江苏省农用激素工程技术研究中心有限公司 苯嘧磺草胺中间体的制备方法
WO2015091642A1 (en) 2013-12-19 2015-06-25 BASF Agro B.V. Dilute aqueous compositions of saflufenacil
EP3598983A1 (en) * 2014-10-03 2020-01-29 Synaffix B.V. Sulfamide linker, conjugates thereof, and methods of preparation
UA122680C2 (uk) 2015-01-15 2020-12-28 Басф Се Гербіцидна комбінація, яка включає сафлуфенацил та глюфосинат
BR112017015652B1 (pt) 2015-01-22 2022-06-07 BASF Agro B.V. Combinação herbicida, método de controle de vegetação indesejável e método de tratamento por extermínio de vegetação
LT3319434T (lt) 2015-07-10 2019-07-10 BASF Agro B.V. Herbicidinė kompozicija, apimanti cinmetiliną ir petoksamidą
US10813356B2 (en) 2015-07-10 2020-10-27 BASF Agro B.V. Herbicidal composition comprising cinmethylin and dimethenamid
US20180184658A1 (en) 2015-07-10 2018-07-05 BASF Agro B.V. Herbicidal composition comprising cinmethylin and saflufenacil
WO2017009142A1 (en) 2015-07-10 2017-01-19 BASF Agro B.V. Herbicidal composition comprising cinmethylin and specific pigment synthesis inhibitors
US11219212B2 (en) 2015-07-10 2022-01-11 BASF Agro B.V. Herbicidal composition comprising cinmethylin and imazamox
EA201890270A1 (ru) 2015-07-10 2018-08-31 Басф Агро Б.В. Гербицидная композиция, которая содержит цинметилин и специфические хинолинкарбоновые кислоты
US11219215B2 (en) 2015-07-10 2022-01-11 BASF Agro B.V. Herbicidal composition comprising cinmethylin and specific inhibitors of protoporphyrinogen oxidase
AU2016294380B2 (en) 2015-07-10 2020-12-24 BASF Agro B.V. Herbicidal composition comprising cinmethylin and pyroxasulfone
US20180192647A1 (en) 2015-07-10 2018-07-12 BASF Agro B.V. Herbicidal composition comprising cinmethylin and acetochlor or pretilachlor
AU2016299729B2 (en) 2015-07-24 2020-07-23 Basf Se Pyridine compounds useful for combating phytopathogenic fungi
ES2767693T3 (es) 2015-09-03 2020-06-18 Basf Agro Bv Composiciones de micropartículas que comprenden saflufenacilo
CN114249710B (zh) 2016-05-24 2024-07-23 巴斯夫欧洲公司 除草的尿嘧啶吡啶类
WO2018019845A1 (en) 2016-07-29 2018-02-01 Basf Se Method for controlling ppo resistant weeds
KR20180081275A (ko) * 2017-01-06 2018-07-16 주식회사 팜한농 3-아릴우라실 화합물의 제조 방법
PE20220843A1 (es) 2019-08-26 2022-05-24 Adama Agan Ltd Novedosas composiciones liquidas solubles de saflufenacil, metodo de preparacion y uso de estas
EP4114828A1 (en) 2020-03-06 2023-01-11 Basf Se Herbicidal phenyluracils
AR124927A1 (es) 2021-02-24 2023-05-17 Adama Agan Ltd Composiciones herbicidas que comprenden inhibidores de acetolactato sintasa a base de imidazolinona y usos de los mismos
US20240174620A1 (en) 2021-03-04 2024-05-30 Adama Agan Ltd. Solid forms of saflufenacil-sodium and saflufenacil-potassium, process of preparation and use thereof
WO2022201155A1 (en) 2021-03-26 2022-09-29 Adama Agan Ltd. Preparation of 2-chloro-4-fluoro-5-nitrobenzoic acid
AR126744A1 (es) 2021-08-09 2023-11-08 Adama Agan Ltd Nuevo proceso de producción de saflufenacil utilizando productos intermedios novedosos
CA3227501A1 (en) 2021-08-30 2023-03-09 Rahul Kaduskar Crystalline forms of methyl 2-[2-[2-bromo-4-fluoro-5-[3-methyl-2,6-dioxo-4-(trifluoromethyl)pyrimidin-1-yl]phenoxy]phenoxy]-2-methoxy-acetate
WO2023030934A1 (en) 2021-08-31 2023-03-09 Basf Se Herbicidal composition comprising phenyluracils
WO2023030935A1 (en) 2021-08-31 2023-03-09 Basf Se Method for controlling ppo-i resistant weeds
WO2023232507A1 (en) 2022-05-30 2023-12-07 BASF Agro B.V. Process for recovering saflufenacil from process streams
WO2024012913A1 (en) 2022-07-13 2024-01-18 BASF Agro B.V. Herbicidal eode formulation comprising several active ingredients
WO2024042134A1 (en) 2022-08-26 2024-02-29 BASF Agro B.V. Aqueous herbicide formulations
WO2024047648A1 (en) 2022-08-31 2024-03-07 Adama Agan Ltd. Preparation of 2-chloro-4-fluoro-5-nitrobenzoic acid
WO2024133722A1 (en) 2022-12-22 2024-06-27 Basf Agro B. V. Methods of controlling undesirable plants with ppo herbicides and combinations in herbicide tolerant crop plants
WO2024200525A1 (en) 2023-03-29 2024-10-03 Basf Agro B. V. Method for controlling parasitic weeds (orobanche) in protoporphyrinogen oxidase (ppo)-inhibitor tolerant sunflower crop
WO2024201460A1 (en) 2023-03-30 2024-10-03 Adama Agan Ltd. Process for the preparation of sulfamide derivatives

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US4309209A (en) * 1977-08-15 1982-01-05 Chevron Research Herbicidal method and composition
US6207830B1 (en) * 1987-09-23 2001-03-27 Syngenta Crop Protection, Inc. Process for the production of 3-aryl-uracils
US4943309A (en) * 1988-09-06 1990-07-24 Uniroyal Chemical Company, Inc. Method of defoleating cotton plants employing 3-carbonylphenyl uracil derivatives
US5169430A (en) * 1991-08-09 1992-12-08 Uniroyal Chemical Company, Inc. Benzenesulfonamide derivatives and methods for their production
DE4139952A1 (de) 1991-12-04 1993-06-09 Bayer Ag, 5090 Leverkusen, De N-aryl-stickstoffheterocyclen
EP0831091A3 (en) * 1996-09-23 1998-04-15 Novartis AG Process for the production of 3-aryl-uracils
DE19741411A1 (de) * 1996-09-23 1998-03-26 Ciba Geigy Ag Verfahren zur Herstellung von 3-Aryluracilen
DE19652431A1 (de) * 1996-12-17 1998-06-18 Bayer Ag Heterocyclyluracile
WO2001083459A2 (en) * 2000-05-04 2001-11-08 Basf Aktiengesellschaft Uracil substituted phenyl sulfamoyl carboxamides
PL209105B1 (pl) * 2001-09-14 2011-07-29 Basf Ag Kompozycja o działaniu chwastobójczym, sposób zwalczania niepożądanej roślinności i zastosowanie tej kompozycji
CA2485360A1 (en) 2002-05-16 2003-11-27 Basf Aktiengesellschaft Method for the production of sulphamic acid halogenides

Also Published As

Publication number Publication date
KR101135263B1 (ko) 2012-04-12
WO2005054208A1 (de) 2005-06-16
DE502004005772D1 (de) 2008-01-31
CN100558714C (zh) 2009-11-11
CN1890222A (zh) 2007-01-03
ES2295957T3 (es) 2008-04-16
ATE381547T1 (de) 2008-01-15
BRPI0417052B1 (pt) 2014-02-25
US20060293520A1 (en) 2006-12-28
JP4528306B2 (ja) 2010-08-18
EP1692115B1 (de) 2007-12-19
EP1692115A1 (de) 2006-08-23
DK1692115T3 (da) 2008-03-25
KR20060120187A (ko) 2006-11-24
JP2007513110A (ja) 2007-05-24
IL175713A0 (en) 2006-09-05
IL175713A (en) 2010-12-30
US7737275B2 (en) 2010-06-15

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B25D Requested change of name of applicant approved

Owner name: BASF SE (DE)

B15K Others concerning applications: alteration of classification

Free format text: "ALTERADA A CLASSIFICACAO DE: C07D 239/56

Ipc: C07D 239/56 (2006.01), C07D 239/54 (2006.01)

Free format text: ALTERADA A CLASSIFICACAO DE: C07D 239/56; C07D 239/54 PARA: C07D 239/56; C07D 239/54; A01N43/48

Ipc: C07D 239/56 (2006.01), C07D 239/54 (2006.01)

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 01/12/2004, OBSERVADAS AS CONDICOES LEGAIS.

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 20A ANUIDADE.