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BRPI0212137A2 - diidropteridinonas, processos para prepará-las e seu uso como composições farmacêuticas - Google Patents

diidropteridinonas, processos para prepará-las e seu uso como composições farmacêuticas

Info

Publication number
BRPI0212137A2
BRPI0212137A2 BRPI0212137A BR0212137A BRPI0212137A2 BR PI0212137 A2 BRPI0212137 A2 BR PI0212137A2 BR PI0212137 A BRPI0212137 A BR PI0212137A BR 0212137 A BR0212137 A BR 0212137A BR PI0212137 A2 BRPI0212137 A2 BR PI0212137A2
Authority
BR
Brazil
Prior art keywords
dihydropteridinones
preparing
processes
pharmaceutical compositions
pharmaceutical
Prior art date
Application number
BRPI0212137A
Other languages
English (en)
Inventor
Christian Eickmeier
Eckhart Bauer
Gerald Pohl
Gisela Schnapp
Jens Jürgen Quant
Martin Steegmaier
Matthias Grauert
Matthias Hoffmann
Norbert Redemann
Steffen Breitfelder
Thorsten Lehmann-Lintz
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of BRPI0212137A2 publication Critical patent/BRPI0212137A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
BRPI0212137A 2001-09-04 2002-08-30 diidropteridinonas, processos para prepará-las e seu uso como composições farmacêuticas BRPI0212137A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10143272 2001-09-04
PCT/EP2002/009728 WO2003020722A1 (de) 2001-09-04 2002-08-30 Neue dihydropteridinone, verfahren zu deren herstellung und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
BRPI0212137A2 true BRPI0212137A2 (pt) 2016-06-28

Family

ID=7697637

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0212137A BRPI0212137A2 (pt) 2001-09-04 2002-08-30 diidropteridinonas, processos para prepará-las e seu uso como composições farmacêuticas

Country Status (30)

Country Link
EP (1) EP1427730B1 (pt)
JP (1) JP3876254B2 (pt)
KR (1) KR100955589B1 (pt)
CN (1) CN1551881A (pt)
AR (1) AR036586A1 (pt)
AT (1) ATE332898T1 (pt)
AU (1) AU2002337047B2 (pt)
BR (1) BRPI0212137A2 (pt)
CA (1) CA2458699C (pt)
CO (1) CO5560575A2 (pt)
CY (1) CY1105337T1 (pt)
DE (1) DE50207522D1 (pt)
DK (1) DK1427730T3 (pt)
EA (1) EA007062B1 (pt)
EC (1) ECSP045003A (pt)
ES (1) ES2268093T3 (pt)
HR (1) HRP20040213A2 (pt)
HU (1) HUP0401293A3 (pt)
IL (2) IL160440A0 (pt)
MX (1) MXPA04002067A (pt)
MY (1) MY129751A (pt)
NO (1) NO328804B1 (pt)
NZ (1) NZ531928A (pt)
PL (1) PL369740A1 (pt)
PT (1) PT1427730E (pt)
RS (1) RS51012B (pt)
UA (1) UA76512C2 (pt)
UY (1) UY27427A1 (pt)
WO (1) WO2003020722A1 (pt)
ZA (1) ZA200401365B (pt)

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