AU721257B2 - Process for preparing 4-aryl-piperidine derivatives - Google Patents

Process for preparing 4-aryl-piperidine derivatives Download PDF

Info

Publication number: AU721257B2
Authority: AU; Australia
Prior art keywords: compound; formula; treatment; viii; optically active
Prior art date: 1995-05-17
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Ceased

Application number

AU56845/96A

Other languages

English (en)

Other versions

AU5684596A (en

Inventor

Bjorn Bentzen

Mogens Engelstoft

John Bondo Hansen

Soren Lehmann

Svend Treppendahl

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Novo Nordisk AS

Original Assignee

Novo Nordisk AS

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-05-17

Filing date

1996-04-25

Publication date

2000-06-29

1996-04-25 Application filed by Novo Nordisk AS filed Critical Novo Nordisk AS

1996-11-29 Publication of AU5684596A publication Critical patent/AU5684596A/en

2000-06-29 Application granted granted Critical

2000-06-29 Publication of AU721257B2 publication Critical patent/AU721257B2/en

2016-04-25 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Hydrogenated Pyridines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AU56845/96A 1995-05-17 1996-04-25 Process for preparing 4-aryl-piperidine derivatives Ceased AU721257B2 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DK563/95		1995-05-17
DK56395		1995-05-17
PCT/DK1996/000185 WO1996036636A1 (en)	1995-05-17	1996-04-25	Process for preparing 4-aryl-piperidine derivatives

Publications (2)

Publication Number	Publication Date
AU5684596A AU5684596A (en)	1996-11-29
AU721257B2 true AU721257B2 (en)	2000-06-29

Family

ID=8094959

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU56845/96A Ceased AU721257B2 (en)	1995-05-17	1996-04-25	Process for preparing 4-aryl-piperidine derivatives

Country Status (11)

Country	Link
EP (1)	EP0828735A1 (pt)
JP (1)	JPH11505229A (pt)
CN (1)	CN1068597C (pt)
AU (1)	AU721257B2 (pt)
BR (1)	BR9608471A (pt)
CA (1)	CA2220963A1 (pt)
HU (1)	HUP9900318A3 (pt)
IL (1)	IL118294A0 (pt)
NZ (1)	NZ307479A (pt)
WO (1)	WO1996036636A1 (pt)
ZA (1)	ZA963951B (pt)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9526645D0 (en) *	1995-12-28	1996-02-28	Chiroscience Ltd	Stereoselective synthesis
ES2117557B1 (es) *	1996-02-29	1999-07-01	Ferrer Int	Nuevo procedimiento de obtencion de (-)-trans -n-p-fluorobenzoilmetil-4-(p-fluorofenil)-3- ((3,4-(metilendioxi)fenoxi ) metil)-piperidina.
EP1394160A1 (en)	1996-06-13	2004-03-03	SUMIKA FINE CHEMICALS Co., Ltd.	Process for preparing crystalline paroxetin hydrochloride
HU221921B1 (hu) *	1996-07-08	2003-02-28	Richter Gedeon Vegyészeti Gyár Rt.	N-benzil-piperidin- és tetrahidropiridinszármazékok és eljárás azok előállítására
GB9623359D0 (en) *	1996-11-09	1997-01-08	Smithkline Beecham Plc	Novel process
GB9700690D0 (en)	1997-01-15	1997-03-05	Smithkline Beecham Plc	Novel process
GB9710004D0 (en) *	1997-05-17	1997-07-09	Knoll Ag	Chemical process
CN1268889A (zh)	1997-05-29	2000-10-04	史密丝克莱恩比彻姆公司	新方法
JP2002503248A (ja)	1997-06-10	2002-01-29	シントン・ベスローテン・フェンノートシャップ	４−フェニルピペリジン化合物
CH689805A8 (fr) *	1998-07-02	2000-02-29	Smithkline Beecham Plc	Méthanesulfonate de paroxétine, procédé pour sa préparation et compositions pharmaceutiques le contenant.
GB9826175D0 (en) *	1998-11-28	1999-01-20	Smithkline Beecham Plc	Novel process
GB9828767D0 (en) *	1998-12-29	1999-02-17	Smithkline Beecham Plc	Novel process
IT1308629B1 (it) *	1999-02-23	2002-01-09	Recordati Chem Pharm	Processo per la produzione di paroxetina.
IT1313702B1 (it) *	1999-08-02	2002-09-09	Chemi Spa	Processo per la preparazione di derivati 3-sostituiti di 4-fenil-piperidine.
WO2001032178A1 (en) *	1999-10-29	2001-05-10	Novo Nordisk A/S	Use of 3,4-substituted piperidines
GB9930577D0 (en) *	1999-12-23	2000-02-16	Smithkline Beecham Plc	Novel process
WO2001085688A1 (en)	2000-05-12	2001-11-15	Synthon B.V.	TOSYLATE SALTS OF 4-(p-FLUOROPHENYL)-PIPERIDINE-3-CARBINOLS
WO2002006275A1 (en) *	2000-07-17	2002-01-24	Smithkline Beecham P.L.C.	Novel processes for the preparation of 4-phenylpiperidine derivatives
GB0021147D0 (en) *	2000-08-30	2000-10-11	Knoll Ag	Chemical process
GB0021145D0 (en) *	2000-08-30	2000-10-11	Knoll Ag	Chemical process
WO2002028834A1 (en) *	2000-10-06	2002-04-11	Smithkline Beecham P.L.C.	Process for the preparation of aryl-piperidine carbinols and intermediates thereof
ATE282594T1 (de)	2001-01-04	2004-12-15	Ferrer Int	Verfahren zur herstellung von (+)-trans-4-p- fluorophenyl-3-hydroxymethyl-1-methylpiperidin
WO2015071831A1 (en) *	2013-11-18	2015-05-21	Piramal Enterprises Limited	An improved process for minimising the formation of dehalogenated byproducts

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1422263A (en) *	1973-01-30	1976-01-21	Ferrosan As	4-phenyl-piperidine compounds
US4593036A (en) *	1984-02-07	1986-06-03	A/S Ferrosan	(-)-Trans-4-(4-fluorophenyl)-3-[(4-methoxyphenoxy)methyl]-1-methylpiperidine useful as 5-HT potentiator
IE66332B1 (en) *	1986-11-03	1995-12-27	Novo Nordisk As	Piperidine compounds and their preparation and use
DK715988D0 (da) *	1988-12-22	1988-12-22	Ferrosan As	Etherifikation og dealkylering af piperidin-derivater samt intermediater

1996
- 1996-04-25 HU HU9900318A patent/HUP9900318A3/hu unknown
- 1996-04-25 CA CA002220963A patent/CA2220963A1/en not_active Abandoned
- 1996-04-25 EP EP96914861A patent/EP0828735A1/en not_active Ceased
- 1996-04-25 NZ NZ307479A patent/NZ307479A/xx unknown
- 1996-04-25 WO PCT/DK1996/000185 patent/WO1996036636A1/en not_active Application Discontinuation
- 1996-04-25 JP JP8534464A patent/JPH11505229A/ja active Pending
- 1996-04-25 CN CN96193942A patent/CN1068597C/zh not_active Expired - Fee Related
- 1996-04-25 BR BR9608471A patent/BR9608471A/pt not_active Application Discontinuation
- 1996-04-25 AU AU56845/96A patent/AU721257B2/en not_active Ceased
- 1996-05-16 IL IL11829496A patent/IL118294A0/xx unknown
- 1996-05-17 ZA ZA963951A patent/ZA963951B/xx unknown

Also Published As

Publication number	Publication date
HUP9900318A2 (hu)	1999-09-28
CA2220963A1 (en)	1996-11-21
AU5684596A (en)	1996-11-29
BR9608471A (pt)	1998-12-29
CN1184476A (zh)	1998-06-10
EP0828735A1 (en)	1998-03-18
WO1996036636A1 (en)	1996-11-21
NZ307479A (en)	1999-08-30
IL118294A0 (en)	1996-09-12
JPH11505229A (ja)	1999-05-18
HUP9900318A3 (en)	2001-09-28
ZA963951B (en)	1997-01-21
CN1068597C (zh)	2001-07-18

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Legal Events

Date	Code	Title	Description
2000-10-26	FGA	Letters patent sealed or granted (standard patent)
2003-11-27	MK14	Patent ceased section 143(a) (annual fees not paid) or expired