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ZA963951B - Process for preparing 4-aryl-piperidine derivatives with a high yield of the desired enantiomer - Google Patents

Process for preparing 4-aryl-piperidine derivatives with a high yield of the desired enantiomer

Info

Publication number
ZA963951B
ZA963951B ZA963951A ZA963951A ZA963951B ZA 963951 B ZA963951 B ZA 963951B ZA 963951 A ZA963951 A ZA 963951A ZA 963951 A ZA963951 A ZA 963951A ZA 963951 B ZA963951 B ZA 963951B
Authority
ZA
South Africa
Prior art keywords
aryl
preparing
high yield
piperidine derivatives
desired enantiomer
Prior art date
Application number
ZA963951A
Other languages
English (en)
Inventor
John Bondo Hansen
Svend Treppendahl
Mogens Engelstoft
Bjorn Bentzen
Soren Lehmann
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of ZA963951B publication Critical patent/ZA963951B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA963951A 1995-05-17 1996-05-17 Process for preparing 4-aryl-piperidine derivatives with a high yield of the desired enantiomer ZA963951B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK56395 1995-05-17

Publications (1)

Publication Number Publication Date
ZA963951B true ZA963951B (en) 1997-01-21

Family

ID=8094959

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA963951A ZA963951B (en) 1995-05-17 1996-05-17 Process for preparing 4-aryl-piperidine derivatives with a high yield of the desired enantiomer

Country Status (11)

Country Link
EP (1) EP0828735A1 (xx)
JP (1) JPH11505229A (xx)
CN (1) CN1068597C (xx)
AU (1) AU721257B2 (xx)
BR (1) BR9608471A (xx)
CA (1) CA2220963A1 (xx)
HU (1) HUP9900318A3 (xx)
IL (1) IL118294A0 (xx)
NZ (1) NZ307479A (xx)
WO (1) WO1996036636A1 (xx)
ZA (1) ZA963951B (xx)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9526645D0 (en) * 1995-12-28 1996-02-28 Chiroscience Ltd Stereoselective synthesis
ES2117557B1 (es) * 1996-02-29 1999-07-01 Ferrer Int Nuevo procedimiento de obtencion de (-)-trans -n-p-fluorobenzoilmetil-4-(p-fluorofenil)-3- ((3,4-(metilendioxi)fenoxi ) metil)-piperidina.
EP1394160A1 (en) 1996-06-13 2004-03-03 SUMIKA FINE CHEMICALS Co., Ltd. Process for preparing crystalline paroxetin hydrochloride
HU221921B1 (hu) * 1996-07-08 2003-02-28 Richter Gedeon Vegyészeti Gyár Rt. N-benzil-piperidin- és tetrahidropiridinszármazékok és eljárás azok előállítására
GB9623359D0 (en) * 1996-11-09 1997-01-08 Smithkline Beecham Plc Novel process
GB9700690D0 (en) 1997-01-15 1997-03-05 Smithkline Beecham Plc Novel process
GB9710004D0 (en) * 1997-05-17 1997-07-09 Knoll Ag Chemical process
CN1268889A (zh) 1997-05-29 2000-10-04 史密丝克莱恩比彻姆公司 新方法
JP2002503248A (ja) 1997-06-10 2002-01-29 シントン・ベスローテン・フェンノートシャップ ４−フェニルピペリジン化合物
CH689805A8 (fr) * 1998-07-02 2000-02-29 Smithkline Beecham Plc Méthanesulfonate de paroxétine, procédé pour sa préparation et compositions pharmaceutiques le contenant.
GB9826175D0 (en) * 1998-11-28 1999-01-20 Smithkline Beecham Plc Novel process
GB9828767D0 (en) * 1998-12-29 1999-02-17 Smithkline Beecham Plc Novel process
IT1308629B1 (it) * 1999-02-23 2002-01-09 Recordati Chem Pharm Processo per la produzione di paroxetina.
IT1313702B1 (it) * 1999-08-02 2002-09-09 Chemi Spa Processo per la preparazione di derivati 3-sostituiti di 4-fenil-piperidine.
WO2001032178A1 (en) * 1999-10-29 2001-05-10 Novo Nordisk A/S Use of 3,4-substituted piperidines
GB9930577D0 (en) * 1999-12-23 2000-02-16 Smithkline Beecham Plc Novel process
WO2001085688A1 (en) 2000-05-12 2001-11-15 Synthon B.V. TOSYLATE SALTS OF 4-(p-FLUOROPHENYL)-PIPERIDINE-3-CARBINOLS
WO2002006275A1 (en) * 2000-07-17 2002-01-24 Smithkline Beecham P.L.C. Novel processes for the preparation of 4-phenylpiperidine derivatives
GB0021147D0 (en) * 2000-08-30 2000-10-11 Knoll Ag Chemical process
GB0021145D0 (en) * 2000-08-30 2000-10-11 Knoll Ag Chemical process
WO2002028834A1 (en) * 2000-10-06 2002-04-11 Smithkline Beecham P.L.C. Process for the preparation of aryl-piperidine carbinols and intermediates thereof
ATE282594T1 (de) 2001-01-04 2004-12-15 Ferrer Int Verfahren zur herstellung von (+)-trans-4-p- fluorophenyl-3-hydroxymethyl-1-methylpiperidin
WO2015071831A1 (en) * 2013-11-18 2015-05-21 Piramal Enterprises Limited An improved process for minimising the formation of dehalogenated byproducts

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1422263A (en) * 1973-01-30 1976-01-21 Ferrosan As 4-phenyl-piperidine compounds
US4593036A (en) * 1984-02-07 1986-06-03 A/S Ferrosan (-)-Trans-4-(4-fluorophenyl)-3-[(4-methoxyphenoxy)methyl]-1-methylpiperidine useful as 5-HT potentiator
IE66332B1 (en) * 1986-11-03 1995-12-27 Novo Nordisk As Piperidine compounds and their preparation and use
DK715988D0 (da) * 1988-12-22 1988-12-22 Ferrosan As Etherifikation og dealkylering af piperidin-derivater samt intermediater

Also Published As

Publication number Publication date
AU721257B2 (en) 2000-06-29
HUP9900318A2 (hu) 1999-09-28
CA2220963A1 (en) 1996-11-21
AU5684596A (en) 1996-11-29
BR9608471A (pt) 1998-12-29
CN1184476A (zh) 1998-06-10
EP0828735A1 (en) 1998-03-18
WO1996036636A1 (en) 1996-11-21
NZ307479A (en) 1999-08-30
IL118294A0 (en) 1996-09-12
JPH11505229A (ja) 1999-05-18
HUP9900318A3 (en) 2001-09-28
CN1068597C (zh) 2001-07-18

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