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OA10843A - Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma - Google Patents

Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma Download PDF

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Publication number
OA10843A
OA10843A OA9800148A OA9800148A OA10843A OA 10843 A OA10843 A OA 10843A OA 9800148 A OA9800148 A OA 9800148A OA 9800148 A OA9800148 A OA 9800148A OA 10843 A OA10843 A OA 10843A
Authority
OA
OAPI
Prior art keywords
phenyl
methyl
ethoxy
propionic acid
phenylamino
Prior art date
Application number
OA9800148A
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English (en)
Inventor
Timothy Mark Willson
Istvan Kaldor
David Norman Deaton
Jeffrey Edmond Cobb
Matthew Jude Sharp
Greg Alan Erickson
Robert A Mook Jr
Brad Richard Henke
Jon Loren Collins
Marcus Brackeen
John Mark O'callaghan
Grady Evan Boswell
Original Assignee
Glaxo Group Ltd
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10789571&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=OA10843(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of OA10843A publication Critical patent/OA10843A/en

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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OA9800148A 1996-02-28 1998-08-25 Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma OA10843A (en)

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