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NO3013169T3 - - Google Patents

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Publication number
NO3013169T3
NO3013169T3 NO14802136A NO14802136A NO3013169T3 NO 3013169 T3 NO3013169 T3 NO 3013169T3 NO 14802136 A NO14802136 A NO 14802136A NO 14802136 A NO14802136 A NO 14802136A NO 3013169 T3 NO3013169 T3 NO 3013169T3
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NO
Norway
Application number
NO14802136A
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Publication date
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Publication of NO3013169T3 publication Critical patent/NO3013169T3/no

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
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    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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EA201591727A1 (ru) 2016-05-31
KR102059545B1 (ko) 2019-12-26
AU2014233657B2 (en) 2016-08-04
BR112015020008B1 (pt) 2021-05-11
HK1212692A1 (zh) 2016-06-17
US20170260207A1 (en) 2017-09-14
HUE035932T2 (en) 2018-05-28
AR095312A1 (es) 2015-10-07
CY1119707T1 (el) 2018-06-27
EP2970216A1 (en) 2016-01-20
SI2970216T1 (en) 2018-01-31
GT201500294A (es) 2018-11-27
KR20150133214A (ko) 2015-11-27
MX2015012290A (es) 2015-12-16
US10709712B2 (en) 2020-07-14
CN105143209A (zh) 2015-12-09
PH12015502116B1 (en) 2016-01-25
JP2020143117A (ja) 2020-09-10
AU2014233657A1 (en) 2015-08-27
CA2899967A1 (en) 2014-09-25
PL2970216T3 (pl) 2018-04-30
US20160038504A1 (en) 2016-02-11
MA38398A1 (fr) 2018-02-28
JP6360879B2 (ja) 2018-07-18
TN2015000332A1 (en) 2017-01-03
US20140275003A1 (en) 2014-09-18
WO2014151616A1 (en) 2014-09-25
ES2657900T3 (es) 2018-03-07
TWI662025B (zh) 2019-06-11
HRP20180158T1 (hr) 2018-03-09
JP7088983B2 (ja) 2022-06-21
NZ710835A (en) 2016-08-26
CN108467369B (zh) 2021-08-20
JOP20140104B1 (ar) 2021-08-17
EA028194B1 (ru) 2017-10-31
LT2970216T (lt) 2018-01-10
AP2015008632A0 (en) 2015-08-31
DOP2015000241A (es) 2015-12-15
CN105143209B (zh) 2018-03-13
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US9242969B2 (en) 2016-01-26
NI201500120A (es) 2015-11-18
ECSP15042895A (es) 2019-08-30
CR20150487A (es) 2016-01-29
DK2970216T3 (da) 2018-01-29
CU20150118A7 (es) 2016-03-31
CA2899967C (en) 2022-01-18
JP2018150319A (ja) 2018-09-27
BR112015020008A2 (pt) 2017-07-18
JP6738369B2 (ja) 2020-08-12
CL2015002151A1 (es) 2015-12-18
JP2016517417A (ja) 2016-06-16
IL241165B (en) 2019-03-31
PE20160875A1 (es) 2016-09-08
US9694016B2 (en) 2017-07-04
US20190175606A1 (en) 2019-06-13
SG11201506196SA (en) 2015-09-29
UY35398A (es) 2014-10-31
MA38398B1 (fr) 2018-09-28
TW201443021A (zh) 2014-11-16
ZA201505438B (en) 2016-03-30
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