NO176098C - Analogifremgangsmåte for fremstilling av 2-substituerte N,N'-ditrimetoksybenzoyl-piperaziner - Google Patents

Analogifremgangsmåte for fremstilling av 2-substituerte N,N'-ditrimetoksybenzoyl-piperaziner

Info

Publication number: NO176098C
Authority: NO; Norway
Prior art keywords: ditrimethoxybenzoyl; piperazines; substituted; preparation; analogous process
Prior art date: 1989-04-15

Application number

NO901631A

Other languages

English (en)

Other versions

NO901631D0 (no

NO901631L (no

NO176098B (no

Inventor

Pierre Braquet

Eduardo Pirotzky

Jean-Jacques Godfroid

Francoise Heymans

Original Assignee

Sod Conseils Rech Applic

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1989-04-15

Filing date

1990-04-10

Publication date

1995-02-01

1990-04-10 Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic

1990-04-10 Publication of NO901631D0 publication Critical patent/NO901631D0/no

1990-10-16 Publication of NO901631L publication Critical patent/NO901631L/no

1994-10-24 Publication of NO176098B publication Critical patent/NO176098B/no

1995-02-01 Publication of NO176098C publication Critical patent/NO176098C/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/04—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/12—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pulmonology (AREA)
Immunology (AREA)
Diabetes (AREA)
Hematology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

NO901631A 1989-04-15 1990-04-10 Analogifremgangsmåte for fremstilling av 2-substituerte N,N'-ditrimetoksybenzoyl-piperaziner NO176098C (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB898908587A GB8908587D0 (en)	1989-04-15	1989-04-15	New 2-substituted n,n'-ditrimethoxybenzoyl piperazines

Publications (4)

Publication Number	Publication Date
NO901631D0 NO901631D0 (no)	1990-04-10
NO901631L NO901631L (no)	1990-10-16
NO176098B NO176098B (no)	1994-10-24
NO176098C true NO176098C (no)	1995-02-01

Family

ID=10655129

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO901631A NO176098C (no)	1989-04-15	1990-04-10	Analogifremgangsmåte for fremstilling av 2-substituerte N,N'-ditrimetoksybenzoyl-piperaziner

Country Status (32)

Country	Link
US (1)	US5019576A (no)
JP (1)	JP2633709B2 (no)
KR (1)	KR900016178A (no)
AR (1)	AR247736A1 (no)
AT (1)	AT399337B (no)
AU (1)	AU631334B2 (no)
BE (1)	BE1007245A3 (no)
CA (1)	CA2014521C (no)
CH (1)	CH681301A5 (no)
DE (1)	DE4011925A1 (no)
DK (1)	DK91890A (no)
DZ (1)	DZ1407A1 (no)
ES (1)	ES2019554A6 (no)
FI (1)	FI92058C (no)
FR (2)	FR2645859B1 (no)
GB (2)	GB8908587D0 (no)
GR (1)	GR1000355B (no)
HK (1)	HK95092A (no)
IE (1)	IE65058B1 (no)
IN (1)	IN175799B (no)
IT (1)	IT1241631B (no)
LU (1)	LU87719A1 (no)
MA (1)	MA21805A1 (no)
NL (1)	NL9000798A (no)
NO (1)	NO176098C (no)
NZ (1)	NZ233250A (no)
OA (1)	OA09446A (no)
PT (1)	PT93736B (no)
SE (1)	SE505186C2 (no)
SG (1)	SG92092G (no)
TN (1)	TNSN90051A1 (no)
ZA (1)	ZA902566B (no)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5344830A (en) *	1992-12-10	1994-09-06	Merck & Co., Inc.	N,N-diacylpiperazine tachykinin antagonists
IL111730A (en) *	1993-11-29	1998-12-06	Fujisawa Pharmaceutical Co	Piperazine derivatives, processes for their preparation and pharmaceutical preparations containing them
US5883098A (en) *	1993-11-29	1999-03-16	Fujisawa Pharmaceutical Co., Ltd.	Piperazine derivatives
US5610165A (en) *	1994-02-17	1997-03-11	Merck & Co., Inc.	N-acylpiperidine tachykinin antagonists
MX9708416A (es) *	1995-05-02	1998-02-28	Schering Corp	Derivados de piperazino como antagonistas de neuroquininas.
US5795894A (en) *	1995-05-02	1998-08-18	Schering Corporation	Piperazino derivatives as neurokinn antagonists
BR9610277A (pt) *	1995-08-31	1999-07-06	Schering Corp	Derivados de piperazino como antagonistas de neurowuinina
US5892039A (en) *	1995-08-31	1999-04-06	Schering Corporation	Piperazino derivatives as neurokinin antagonists
US5869488A (en) *	1996-05-01	1999-02-09	Schering Corporation	Piperazino derivatives as neurokinin antagonists
FR2780649B1 (fr) *	1998-07-06	2001-03-09	Univ Paris Vii Denis Diderot	Derives de la piperazine pour l'inhibition de la replication du virus de l'immunodeficience humaine

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1243991A (en) *	1968-06-10	1971-08-25	Ici Ltd	Piperidine, morpholine and piperazine derivatives
FR2209560A1 (en) *	1972-12-07	1974-07-05	Degussa	N-(Trialkoxyaroyl)-ethylenediamine derivs - useful as cardioactive medicaments, exhibit anti-ischaemic activity comparable to nitroglycerin
IL85700A0 (en) *	1987-03-24	1988-08-31	Takeda Chemical Industries Ltd	1,4-disubstituted piperazine compounds,their production and use
EP0318235A3 (en) *	1987-11-25	1991-05-02	Takeda Chemical Industries, Ltd.	Paf antagonist, 1,4-disubstituted piperazine compounds and production thereof
KR900018073A (ko) *	1988-05-23	1990-12-20	추후보충	피페라진 화합물
GB8823775D0 (en) *	1988-10-11	1988-11-16	Scras	New 2-carbonyl substituted n n'-di-(trimethoxybenzoyl)piperazines
GB8823776D0 (en) *	1988-10-11	1988-11-16	Scras	New 2-methoxycarbonyl sustituted n n'-di-(trimethoxybenzoyl)piperazines
US4997836A (en) *	1988-11-11	1991-03-05	Takeda Chemical Industries, Ltd.	Trisubstituted piperazine compounds, their production and use

1989
- 1989-04-15 GB GB898908587A patent/GB8908587D0/en active Pending
1990
- 1990-04-03 ZA ZA902566A patent/ZA902566B/xx unknown
- 1990-04-04 GB GB9007612A patent/GB2230262B/en not_active Expired - Fee Related
- 1990-04-05 NL NL9000798A patent/NL9000798A/nl not_active Application Discontinuation
- 1990-04-05 IN IN140DE1990D patent/IN175799B/en unknown
- 1990-04-06 GR GR900100270A patent/GR1000355B/el unknown
- 1990-04-06 SE SE9001269A patent/SE505186C2/sv not_active IP Right Cessation
- 1990-04-09 NZ NZ233250A patent/NZ233250A/en unknown
- 1990-04-09 US US07/506,421 patent/US5019576A/en not_active Expired - Lifetime
- 1990-04-10 CH CH1206/90A patent/CH681301A5/fr not_active IP Right Cessation
- 1990-04-10 MA MA22064A patent/MA21805A1/fr unknown
- 1990-04-10 AR AR90316593A patent/AR247736A1/es active
- 1990-04-10 NO NO901631A patent/NO176098C/no unknown
- 1990-04-10 LU LU87719A patent/LU87719A1/fr unknown
- 1990-04-11 BE BE9000408A patent/BE1007245A3/fr not_active IP Right Cessation
- 1990-04-11 PT PT93736A patent/PT93736B/pt not_active IP Right Cessation
- 1990-04-11 AT AT0086690A patent/AT399337B/de not_active IP Right Cessation
- 1990-04-11 DK DK091890A patent/DK91890A/da unknown
- 1990-04-11 ES ES9001056A patent/ES2019554A6/es not_active Expired - Fee Related
- 1990-04-11 DZ DZ900066A patent/DZ1407A1/fr active
- 1990-04-11 IE IE131490A patent/IE65058B1/en not_active IP Right Cessation
- 1990-04-12 CA CA002014521A patent/CA2014521C/en not_active Expired - Fee Related
- 1990-04-12 TN TNTNSN90051A patent/TNSN90051A1/fr unknown
- 1990-04-12 DE DE4011925A patent/DE4011925A1/de not_active Ceased
- 1990-04-12 OA OA59775A patent/OA09446A/xx unknown
- 1990-04-12 IT IT20020A patent/IT1241631B/it active IP Right Grant
- 1990-04-12 FI FI901883A patent/FI92058C/fi not_active IP Right Cessation
- 1990-04-13 JP JP2096620A patent/JP2633709B2/ja not_active Expired - Lifetime
- 1990-04-13 FR FR909004798A patent/FR2645859B1/fr not_active Expired - Fee Related
- 1990-04-13 FR FR909004797A patent/FR2645743B1/fr not_active Expired - Fee Related
- 1990-04-14 KR KR1019900005198A patent/KR900016178A/ko not_active Application Discontinuation
- 1990-04-17 AU AU53261/90A patent/AU631334B2/en not_active Ceased
1992
- 1992-09-11 SG SG920/92A patent/SG92092G/en unknown
- 1992-11-26 HK HK950/92A patent/HK95092A/xx not_active IP Right Cessation

Also Published As

Publication number	Publication date
CH681301A5 (no)	1993-02-26
DK91890D0 (da)	1990-04-11
GR900100270A (en)	1991-09-27
CA2014521A1 (en)	1990-10-15
BE1007245A3 (fr)	1995-05-02
SG92092G (en)	1992-12-04
NO901631D0 (no)	1990-04-10
OA09446A (fr)	1992-10-15
FR2645859B1 (fr)	1992-06-05
NL9000798A (nl)	1990-11-01
ES2019554A6 (es)	1991-06-16
JPH02292266A (ja)	1990-12-03
NO901631L (no)	1990-10-16
CA2014521C (en)	1997-09-09
KR900016178A (ko)	1990-11-12
SE505186C2 (sv)	1997-07-14
FR2645859A1 (fr)	1990-10-19
FR2645743B1 (fr)	1992-06-05
GB9007612D0 (en)	1990-05-30
FI901883A0 (fi)	1990-04-12
FI92058C (fi)	1994-09-26
AT399337B (de)	1995-04-25
ATA86690A (de)	1994-09-15
SE9001269D0 (sv)	1990-04-06
MA21805A1 (fr)	1990-12-31
FR2645743A1 (fr)	1990-10-19
AU631334B2 (en)	1992-11-19
AR247736A1 (es)	1995-03-31
IT1241631B (it)	1994-01-25
FI92058B (fi)	1994-06-15
LU87719A1 (fr)	1990-07-24
DZ1407A1 (fr)	2004-09-13
US5019576A (en)	1991-05-28
TNSN90051A1 (fr)	1991-03-05
GR1000355B (el)	1992-06-25
IE65058B1 (en)	1995-10-04
PT93736B (pt)	1996-09-30
SE9001269L (sv)	1990-10-16
IN175799B (no)	1995-08-26
IE901314L (en)	1990-10-15
IT9020020A0 (it)	1990-04-12
NO176098B (no)	1994-10-24
GB8908587D0 (en)	1989-06-01
JP2633709B2 (ja)	1997-07-23
GB2230262B (en)	1992-02-26
ZA902566B (en)	1991-01-30
DK91890A (da)	1990-10-16
AU5326190A (en)	1990-11-01
GB2230262A (en)	1990-10-17
DE4011925A1 (de)	1990-10-18
HK95092A (en)	1992-12-04
IT9020020A1 (it)	1991-10-12
NZ233250A (en)	1991-03-26
PT93736A (pt)	1990-11-20

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FI891338A (fi)	1989-09-25	Parannus menetelmään 2',3'-dideoksi-2',3'-didehydronukleosidien valmistamiseksi
FI894546A (fi)	1990-03-28	Menetelmä uusien 2'-halogeenimetylideeni-, 2'-etenylideeni- ja 2'-etynyyliadenosiinijohdannaisten valmistamiseksi
NO176098C (no)	1995-02-01	Analogifremgangsmåte for fremstilling av 2-substituerte N,N'-ditrimetoksybenzoyl-piperaziner
FI895662A0 (fi)	1989-11-27	Menetelmä 3,4-difluorisubstituoidun benseenin valmistamiseksi
FR2630735B1 (fr)	1990-09-14	Procede de preparations d'halogenophenols
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PT86623A (pt)	1988-02-01	Process for the preparation of derivatives of 3-aryl-5-alkylthio-4h-1,2,4-triazoles
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FI93363C (fi)	1995-03-27	Uusi menetelmä 2-diatso-3-trisubstituoitujen silyylioksi-3-butenoaattien valmistamiseksi
FR2666581B1 (fr)	1993-05-28	Procede de preparation d'acetate de tocopherol.
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