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Higher acyclic nitrogen containing deoxy sugar derivatives: a new lead in the generation of antimycobacterial chemotherapeutics

Bioorg Med Chem. 2002 Jun;10(6):1695-702. doi: 10.1016/s0968-0896(02)00045-7.

Abstract

Syntheses of higher acyclic nitrogen containing deoxy sugar derivatives via nitroaldol reaction of different nitroalkanes with 2,3-dideoxy-alpha,beta-unsaturated aldehydo sugars obtained from glycals namely acetylated glucal and galactal and their in vitro antimycobacterial activity are presented.

MeSH terms

  • Acetylation
  • Antitubercular Agents / chemical synthesis*
  • Antitubercular Agents / chemistry
  • Antitubercular Agents / pharmacology*
  • Deoxy Sugars / chemistry*
  • Deoxy Sugars / pharmacology*
  • Hydrogenation
  • Microbial Sensitivity Tests
  • Molecular Structure
  • Mycobacterium tuberculosis / drug effects
  • Mycobacterium tuberculosis / growth & development
  • Nitrogen / analysis*
  • Structure-Activity Relationship

Substances

  • Antitubercular Agents
  • Deoxy Sugars
  • Nitrogen