Nothing Special   »   [go: up one dir, main page]

1.9 A crystal structure of interleukin 6: implications for a novel mode of receptor dimerization and signaling

EMBO J. 1997 Mar 3;16(5):989-97. doi: 10.1093/emboj/16.5.989.

Abstract

Interleukin 6 (IL-6) has many biological activities in vivo, and deregulation has been implicated in many disease processes. IL-6, a 185 amino acid polypeptide was refolded, purified and crystallized. The crystals diffracted to beyond 1.9 A and the structure was solved using single isomorphous replacement. The X-ray structure of IL-6 is composed of a four helix bundle linked by loops and an additional mini-helix. 157 out of 185 residues are well defined in the final structure, with 18 N-terminal and 8 A-B loop amino acids displaying no interpretable electron density. The three-dimensional structure has been used to construct a model of IL-6 interacting with the IL-6 receptor (alpha-chain) and gp130 (beta-chain) that gives new insight into the process of molecular recognition and signaling. Based on this model, we predict a fourth binding site on IL-6, a low affinity IL-6-IL-6 interaction, which may be necessary for the sequential assembly of a functional hexameric IL-6 receptor complex.

MeSH terms

  • Antigens, CD / chemistry*
  • Antigens, CD / metabolism
  • Binding Sites
  • Crystallization
  • Crystallography, X-Ray
  • Dimerization
  • Disulfides / chemistry
  • Escherichia coli / genetics
  • Gene Expression / genetics
  • Granulocyte Colony-Stimulating Factor / chemistry
  • Human Growth Hormone / chemistry
  • Humans
  • Hydrogen Bonding
  • Interleukin-6 / chemistry*
  • Interleukin-6 / metabolism
  • Models, Molecular
  • Protein Binding
  • Protein Conformation
  • Protein Folding
  • Protein Structure, Tertiary
  • Receptors, Interleukin / chemistry*
  • Receptors, Interleukin / metabolism
  • Receptors, Interleukin-6
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / isolation & purification
  • Recombinant Proteins / metabolism
  • Water / chemistry
  • Water / metabolism

Substances

  • Antigens, CD
  • Disulfides
  • Interleukin-6
  • Receptors, Interleukin
  • Receptors, Interleukin-6
  • Recombinant Proteins
  • Water
  • Human Growth Hormone
  • Granulocyte Colony-Stimulating Factor