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YU48396A - Zwitterionic forms of trovaphloxacine,process for preparation thereof and their pharmaceutical compositions - Google Patents

Zwitterionic forms of trovaphloxacine,process for preparation thereof and their pharmaceutical compositions

Info

Publication number
YU48396A
YU48396A YU48396A YU48396A YU48396A YU 48396 A YU48396 A YU 48396A YU 48396 A YU48396 A YU 48396A YU 48396 A YU48396 A YU 48396A YU 48396 A YU48396 A YU 48396A
Authority
YU
Yugoslavia
Prior art keywords
preparation
pharmaceutical compositions
trovaphloxacine
zwitterionic forms
zwitterionic
Prior art date
Application number
YU48396A
Other languages
Serbo-Croatian (sh)
Inventor
John Meldrum Allen Douglas
Bruning Joseph David
Norris Timothy
Original Assignee
Pfizer Inc Delaware
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc Delaware filed Critical Pfizer Inc Delaware
Publication of YU48396A publication Critical patent/YU48396A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Physical Water Treatments (AREA)
  • Processing Of Solid Wastes (AREA)

Abstract

Zviterjonski oblik trovafloksacina koji ima formulu koji je izabran iz grupe koju čine njegovi nehigroskopni polimerf PI, higroskopni polimorf PII i pentahidrat, kao i postupci za njihovo dobijanje. Pronalazak se dalje odnosi na farmaceutske kompozicije koje obuhvataju jedinjenja pronalaska za lečenje bakterijskih infekcija kod sisara.A zwitterionic form of trovafloxacin having a formula selected from the group consisting of its non-hygroscopic polymorph PI, hygroscopic polymorph PII and pentahydrate, as well as methods for their preparation. The invention further relates to pharmaceutical compositions comprising the compounds of the invention for the treatment of bacterial infections in mammals.

YU48396A 1995-08-29 1996-08-28 Zwitterionic forms of trovaphloxacine,process for preparation thereof and their pharmaceutical compositions YU48396A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US297595P 1995-08-29 1995-08-29

Publications (1)

Publication Number Publication Date
YU48396A true YU48396A (en) 1998-12-23

Family

ID=21703460

Family Applications (1)

Application Number Title Priority Date Filing Date
YU48396A YU48396A (en) 1995-08-29 1996-08-28 Zwitterionic forms of trovaphloxacine,process for preparation thereof and their pharmaceutical compositions

Country Status (30)

Country Link
EP (1) EP0850060A1 (en)
JP (1) JP3188476B2 (en)
KR (1) KR100343909B1 (en)
CN (1) CN1190889A (en)
AP (1) AP636A (en)
AR (1) AR003985A1 (en)
AU (1) AU704115B2 (en)
BR (1) BR9609998A (en)
CA (1) CA2229786C (en)
CO (1) CO4480739A1 (en)
CZ (1) CZ56698A3 (en)
DZ (1) DZ2087A1 (en)
GT (1) GT199600072A (en)
HR (1) HRP960395B1 (en)
HU (1) HUP9900170A3 (en)
IL (1) IL122651A (en)
MA (1) MA23966A1 (en)
MY (1) MY113874A (en)
NO (1) NO309814B1 (en)
NZ (1) NZ312199A (en)
OA (1) OA10669A (en)
PE (1) PE12598A1 (en)
PL (1) PL325170A1 (en)
RU (1) RU2144921C1 (en)
SK (1) SK23898A3 (en)
TN (1) TNSN96109A1 (en)
TR (1) TR199800339T1 (en)
WO (1) WO1997007800A1 (en)
YU (1) YU48396A (en)
ZA (1) ZA967282B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1998000106A (en) 1997-08-01 1999-01-08 Pfizer Prod Inc PARENTERAL COMPOSITIONS OF ALATROFLAXACINO
US7019142B2 (en) 1998-01-16 2006-03-28 Pfizer Inc. Process for preparing naphthyridones and intermediates
PA8466701A1 (en) 1998-01-21 2000-09-29 Pfizer Prod Inc TROVAFLOXACINO MESYLATE TABLET
US6114531A (en) * 1998-07-28 2000-09-05 Pfizer Inc. Process for preparing quinolone and naphthyridone carboxylic acids
HN1999000141A (en) * 1998-09-03 2000-06-19 Pfizer Prod Inc PROCEDURE FOR PREPARING SALTS OF TROVAFLOXACIN FOR ADDITION OF ACIDS.
US6239141B1 (en) 1999-06-04 2001-05-29 Pfizer Inc. Trovafloxacin oral suspensions

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids

Also Published As

Publication number Publication date
CN1190889A (en) 1998-08-19
SK23898A3 (en) 1999-05-07
IL122651A (en) 2000-02-17
AU6367696A (en) 1997-03-19
KR100343909B1 (en) 2003-04-10
PE12598A1 (en) 1998-03-20
MX9801664A (en) 1998-08-30
GT199600072A (en) 1998-02-14
RU2144921C1 (en) 2000-01-27
AU704115B2 (en) 1999-04-15
ZA967282B (en) 1998-03-02
NO980862D0 (en) 1998-02-27
AP9600853A0 (en) 1996-10-31
BR9609998A (en) 1999-07-06
TR199800339T1 (en) 1998-06-22
CA2229786A1 (en) 1997-03-06
IL122651A0 (en) 1998-08-16
HRP960395A2 (en) 1998-06-30
JP3188476B2 (en) 2001-07-16
AR003985A1 (en) 1998-09-30
WO1997007800A1 (en) 1997-03-06
KR19990044232A (en) 1999-06-25
MA23966A1 (en) 1997-04-01
CA2229786C (en) 2002-02-19
AP636A (en) 1998-04-09
NO980862L (en) 1998-02-27
OA10669A (en) 2000-11-06
PL325170A1 (en) 1998-07-06
HUP9900170A3 (en) 1999-11-29
MY113874A (en) 2002-06-29
NZ312199A (en) 1999-06-29
DZ2087A1 (en) 2002-07-22
CO4480739A1 (en) 1997-07-09
JPH10511692A (en) 1998-11-10
EP0850060A1 (en) 1998-07-01
HRP960395B1 (en) 2001-12-31
NO309814B1 (en) 2001-04-02
CZ56698A3 (en) 1999-02-17
HUP9900170A2 (en) 1999-05-28
TNSN96109A1 (en) 2005-03-15

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