YU48396A - Zwitterionic forms of trovaphloxacine,process for preparation thereof and their pharmaceutical compositions - Google Patents
Zwitterionic forms of trovaphloxacine,process for preparation thereof and their pharmaceutical compositionsInfo
- Publication number
- YU48396A YU48396A YU48396A YU48396A YU48396A YU 48396 A YU48396 A YU 48396A YU 48396 A YU48396 A YU 48396A YU 48396 A YU48396 A YU 48396A YU 48396 A YU48396 A YU 48396A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- preparation
- pharmaceutical compositions
- trovaphloxacine
- zwitterionic forms
- zwitterionic
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Physical Water Treatments (AREA)
- Processing Of Solid Wastes (AREA)
Abstract
Zviterjonski oblik trovafloksacina koji ima formulu koji je izabran iz grupe koju čine njegovi nehigroskopni polimerf PI, higroskopni polimorf PII i pentahidrat, kao i postupci za njihovo dobijanje. Pronalazak se dalje odnosi na farmaceutske kompozicije koje obuhvataju jedinjenja pronalaska za lečenje bakterijskih infekcija kod sisara.A zwitterionic form of trovafloxacin having a formula selected from the group consisting of its non-hygroscopic polymorph PI, hygroscopic polymorph PII and pentahydrate, as well as methods for their preparation. The invention further relates to pharmaceutical compositions comprising the compounds of the invention for the treatment of bacterial infections in mammals.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US297595P | 1995-08-29 | 1995-08-29 |
Publications (1)
Publication Number | Publication Date |
---|---|
YU48396A true YU48396A (en) | 1998-12-23 |
Family
ID=21703460
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
YU48396A YU48396A (en) | 1995-08-29 | 1996-08-28 | Zwitterionic forms of trovaphloxacine,process for preparation thereof and their pharmaceutical compositions |
Country Status (30)
Country | Link |
---|---|
EP (1) | EP0850060A1 (en) |
JP (1) | JP3188476B2 (en) |
KR (1) | KR100343909B1 (en) |
CN (1) | CN1190889A (en) |
AP (1) | AP636A (en) |
AR (1) | AR003985A1 (en) |
AU (1) | AU704115B2 (en) |
BR (1) | BR9609998A (en) |
CA (1) | CA2229786C (en) |
CO (1) | CO4480739A1 (en) |
CZ (1) | CZ56698A3 (en) |
DZ (1) | DZ2087A1 (en) |
GT (1) | GT199600072A (en) |
HR (1) | HRP960395B1 (en) |
HU (1) | HUP9900170A3 (en) |
IL (1) | IL122651A (en) |
MA (1) | MA23966A1 (en) |
MY (1) | MY113874A (en) |
NO (1) | NO309814B1 (en) |
NZ (1) | NZ312199A (en) |
OA (1) | OA10669A (en) |
PE (1) | PE12598A1 (en) |
PL (1) | PL325170A1 (en) |
RU (1) | RU2144921C1 (en) |
SK (1) | SK23898A3 (en) |
TN (1) | TNSN96109A1 (en) |
TR (1) | TR199800339T1 (en) |
WO (1) | WO1997007800A1 (en) |
YU (1) | YU48396A (en) |
ZA (1) | ZA967282B (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
HN1998000106A (en) | 1997-08-01 | 1999-01-08 | Pfizer Prod Inc | PARENTERAL COMPOSITIONS OF ALATROFLAXACINO |
US7019142B2 (en) | 1998-01-16 | 2006-03-28 | Pfizer Inc. | Process for preparing naphthyridones and intermediates |
PA8466701A1 (en) | 1998-01-21 | 2000-09-29 | Pfizer Prod Inc | TROVAFLOXACINO MESYLATE TABLET |
US6114531A (en) * | 1998-07-28 | 2000-09-05 | Pfizer Inc. | Process for preparing quinolone and naphthyridone carboxylic acids |
HN1999000141A (en) * | 1998-09-03 | 2000-06-19 | Pfizer Prod Inc | PROCEDURE FOR PREPARING SALTS OF TROVAFLOXACIN FOR ADDITION OF ACIDS. |
US6239141B1 (en) | 1999-06-04 | 2001-05-29 | Pfizer Inc. | Trovafloxacin oral suspensions |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5164402A (en) * | 1989-08-16 | 1992-11-17 | Pfizer Inc | Azabicyclo quinolone and naphthyridinone carboxylic acids |
-
1996
- 1996-07-29 NZ NZ312199A patent/NZ312199A/en unknown
- 1996-07-29 CN CN96195624A patent/CN1190889A/en active Pending
- 1996-07-29 IL IL12265196A patent/IL122651A/en not_active IP Right Cessation
- 1996-07-29 CZ CZ98566A patent/CZ56698A3/en unknown
- 1996-07-29 WO PCT/IB1996/000756 patent/WO1997007800A1/en not_active Application Discontinuation
- 1996-07-29 CA CA002229786A patent/CA2229786C/en not_active Expired - Fee Related
- 1996-07-29 EP EP96923020A patent/EP0850060A1/en not_active Withdrawn
- 1996-07-29 TR TR1998/00339T patent/TR199800339T1/en unknown
- 1996-07-29 HU HU9900170A patent/HUP9900170A3/en unknown
- 1996-07-29 RU RU98103873/04A patent/RU2144921C1/en not_active IP Right Cessation
- 1996-07-29 SK SK238-98A patent/SK23898A3/en unknown
- 1996-07-29 AU AU63676/96A patent/AU704115B2/en not_active Ceased
- 1996-07-29 JP JP50343697A patent/JP3188476B2/en not_active Expired - Fee Related
- 1996-07-29 PL PL96325170A patent/PL325170A1/en unknown
- 1996-07-29 KR KR10-1998-0701468A patent/KR100343909B1/en not_active IP Right Cessation
- 1996-07-29 BR BR9609998A patent/BR9609998A/en unknown
- 1996-08-23 GT GT199600072A patent/GT199600072A/en unknown
- 1996-08-26 PE PE1996000633A patent/PE12598A1/en not_active Application Discontinuation
- 1996-08-26 AR ARP960104121A patent/AR003985A1/en unknown
- 1996-08-28 DZ DZ960131A patent/DZ2087A1/en active
- 1996-08-28 TN TNTNSN96109A patent/TNSN96109A1/en unknown
- 1996-08-28 ZA ZA9607282A patent/ZA967282B/en unknown
- 1996-08-28 YU YU48396A patent/YU48396A/en unknown
- 1996-08-28 MY MYPI96003579A patent/MY113874A/en unknown
- 1996-08-28 MA MA24344A patent/MA23966A1/en unknown
- 1996-08-29 AP APAP/P/1996/000853A patent/AP636A/en active
- 1996-08-29 CO CO96046149A patent/CO4480739A1/en unknown
- 1996-08-29 HR HR960395A patent/HRP960395B1/en not_active IP Right Cessation
-
1998
- 1998-02-27 NO NO980862A patent/NO309814B1/en not_active Application Discontinuation
- 1998-02-27 OA OA9800026A patent/OA10669A/en unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
YU16501A (en) | 4-carboxyamino-2-substituted-1,2,3,4-tetrahydroquinolines as cetp inhibitors | |
YU18101A (en) | 4-amino-supstituted-2-substituted-1,2,3,4-tetrahydroquinolines as cetp inhibitors | |
FI98460B (en) | Process for the preparation of a therapeutically useful 4H-1-benzopyran-4-one derivative or a salt thereof and an intermediate useful in the process | |
ME00558A (en) | Pyrazole derivatives for treating hiv | |
DE69634045D1 (en) | ANTITHROMBOTIC DIAMINE | |
HN1998000074A (en) | DERIVATIVES FROM MACROLIDES C-4 SUBSTITUTED | |
CY1111693T1 (en) | ANTIQUE FACTORS | |
AR038955A1 (en) | PIRIMIDINONE AND PIRIDONA SUBSTITUTED COMPOUNDS AND METHODS FOR USE | |
BR0111263A (en) | 2-Aminocarbonyl-9h-purine derivatives | |
FI20115753A (en) | Pharmaceutical compositions for the treatment of diseases caused by IL-6 production | |
BR0112395A (en) | Benzothiazole Derivatives | |
EA200501098A1 (en) | ANTIBACTERIAL AGENTS | |
UA44254C2 (en) | DERIVATIVES OF 4- (SUBSTITUTED PHENYLAMINO) QINAZOLINE, METHOD OF THEIR PREPARATION, METHOD OF TREATMENT AND PHARMACEUTICAL COMPOSITION | |
HUP0401538A2 (en) | Novel derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and pharmaceutical compositions containing same | |
DK0462812T3 (en) | Pyran derivatives as inhibitors of 5-lipoxygenase | |
MEP9309A (en) | Novel oligosaccharides, preparation method and pharmaceutical compositions containing the same | |
YU33401A (en) | 13-membered azalides and their use as antibiotic agents | |
ATE268337T1 (en) | C11-CARBAMATES OF ANTIBACTERIAL MACROLIDS | |
DK1057828T3 (en) | Oral trovafloxacin suspensions | |
YU48396A (en) | Zwitterionic forms of trovaphloxacine,process for preparation thereof and their pharmaceutical compositions | |
YU42098A (en) | The use of olanzapine | |
YU37597A (en) | New pyranosid derivatives | |
ES2076838T3 (en) | NEW DERIVATIVE OF ISOINDOLINONE, ITS PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS THAT CONTAIN IT. | |
ATE271062T1 (en) | MACROLIDE ANTIBIOTICS | |
YU48296A (en) | Polymorphs of the pro-drug 6-n-(l-ala-l-ala)-trovaphloxacyne processes for the preparation thereof and their pharmaceutical comositions |