UA92047C2 - Carbonylamino pyrrolopyrazoles, potent kinase inhibitors - Google Patents
Carbonylamino pyrrolopyrazoles, potent kinase inhibitorsInfo
- Publication number
- UA92047C2 UA92047C2 UAA200807387A UAA200807387A UA92047C2 UA 92047 C2 UA92047 C2 UA 92047C2 UA A200807387 A UAA200807387 A UA A200807387A UA A200807387 A UAA200807387 A UA A200807387A UA 92047 C2 UA92047 C2 UA 92047C2
- Authority
- UA
- Ukraine
- Prior art keywords
- kinase inhibitors
- pyrrolopyrazoles
- carbonylamino
- potent kinase
- compounds
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Carbonyiamino Pyirolopyrazole compounds of formula (I), compositions including these compounds and methods of their use are provided. Preferred compounds of formula (I) have activity as protein kinase inhibitors, including as inhibitors of PAK4. EMBED ISISServer I
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US75334905P | 2005-12-21 | 2005-12-21 | |
US86493206P | 2006-11-08 | 2006-11-08 | |
PCT/IB2006/003646 WO2007072153A2 (en) | 2005-12-21 | 2006-12-12 | Carbonylamino pyrrolopyrazoles, potent kinase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
UA92047C2 true UA92047C2 (en) | 2010-09-27 |
Family
ID=40247953
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA200807387A UA92047C2 (en) | 2005-12-21 | 2006-12-12 | Carbonylamino pyrrolopyrazoles, potent kinase inhibitors |
Country Status (5)
Country | Link |
---|---|
CN (1) | CN101346382B (en) |
SI (1) | SI1979356T1 (en) |
TN (1) | TNSN08274A1 (en) |
UA (1) | UA92047C2 (en) |
ZA (1) | ZA200804667B (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN113234081A (en) * | 2021-05-27 | 2021-08-10 | 东南大学 | Preparation method of pyrrolopyrazole derivative and DMDPEDA as urea |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UA81790C2 (en) * | 2002-12-19 | 2008-02-11 | Фармация Италия С.П.А. | Substituted derivatives of pyrolopyrazol as kinaze inhibitors |
-
2006
- 2006-12-12 UA UAA200807387A patent/UA92047C2/en unknown
- 2006-12-12 SI SI200631657T patent/SI1979356T1/en unknown
- 2006-12-12 CN CN2006800486846A patent/CN101346382B/en not_active Expired - Fee Related
-
2008
- 2008-05-29 ZA ZA200804667A patent/ZA200804667B/en unknown
- 2008-06-20 TN TNP2008000274A patent/TNSN08274A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
ZA200804667B (en) | 2010-05-26 |
TNSN08274A1 (en) | 2009-10-30 |
SI1979356T1 (en) | 2013-11-29 |
CN101346382A (en) | 2009-01-14 |
CN101346382B (en) | 2011-07-06 |
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