TR200201145T2 - Hidromisin türevleri - Google Patents
Hidromisin türevleriInfo
- Publication number
- TR200201145T2 TR200201145T2 TR2002/01145T TR200201145T TR200201145T2 TR 200201145 T2 TR200201145 T2 TR 200201145T2 TR 2002/01145 T TR2002/01145 T TR 2002/01145T TR 200201145 T TR200201145 T TR 200201145T TR 200201145 T2 TR200201145 T2 TR 200201145T2
- Authority
- TR
- Turkey
- Prior art keywords
- hydromycin
- derivatives
- relates
- compounds
- prodrugs
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Biotechnology (AREA)
- Veterinary Medicine (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Mevcut bulus formül (1'e ait bilesiklerle ve bunlarin farmasötik açidan kabul gören tuzlari, ön ilaçlar ve solvatlari ile ilgilidir; buradaki X,Y,V,W ,W ,Z ve Z , burada tanimlandigi gibidir. Bulus, yukaridaki bilesikleri ihtiva eden farmasötik kompozisyonlarla ve yukaridaki bilesiklerin uygulanmasi suretiyle bakteriyel ve protozoal enfeksiyonlarin tedavi edilmesine yönelik metotlarla da ilgilidir.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US16258199P | 1999-10-29 | 1999-10-29 |
Publications (1)
Publication Number | Publication Date |
---|---|
TR200201145T2 true TR200201145T2 (tr) | 2002-09-23 |
Family
ID=22586256
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2002/01145T TR200201145T2 (tr) | 1999-10-29 | 2000-10-09 | Hidromisin türevleri |
Country Status (32)
Country | Link |
---|---|
US (1) | US6562792B1 (tr) |
EP (1) | EP1224197A1 (tr) |
JP (1) | JP2003512473A (tr) |
KR (1) | KR20020063885A (tr) |
CN (1) | CN1382150A (tr) |
AP (1) | AP2002002494A0 (tr) |
AR (1) | AR023282A1 (tr) |
AU (1) | AU7549400A (tr) |
BG (1) | BG106727A (tr) |
BR (1) | BR0015153A (tr) |
CA (1) | CA2389191A1 (tr) |
CO (1) | CO5261498A1 (tr) |
CZ (1) | CZ20021355A3 (tr) |
EA (1) | EA200200292A1 (tr) |
EE (1) | EE200200228A (tr) |
GT (1) | GT200000185A (tr) |
HK (1) | HK1049672A1 (tr) |
HU (1) | HUP0203525A3 (tr) |
IL (1) | IL148577A0 (tr) |
IS (1) | IS6311A (tr) |
MA (1) | MA26838A1 (tr) |
MX (1) | MXPA02004360A (tr) |
NO (1) | NO20021850D0 (tr) |
OA (1) | OA12081A (tr) |
PA (1) | PA8505801A1 (tr) |
PE (1) | PE20010763A1 (tr) |
PL (1) | PL357083A1 (tr) |
SK (1) | SK5472002A3 (tr) |
SV (1) | SV2002000211A (tr) |
TN (1) | TNSN00211A1 (tr) |
TR (1) | TR200201145T2 (tr) |
WO (1) | WO2001030795A1 (tr) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SK16612002A3 (sk) | 2000-06-02 | 2004-04-06 | Pfizer Products Inc. | Deriváty hygromycínu A na použitie na liečenie bakteriálnych a protozoálnych infekcií |
US6653481B2 (en) * | 2000-12-29 | 2003-11-25 | Synthon Bv | Process for making amlodipine |
US7923439B2 (en) * | 2008-10-15 | 2011-04-12 | Tyco Healthcare Group Lp | Hydroxamate compositions |
EP3840743A4 (en) * | 2018-08-20 | 2022-08-17 | Northeastern University | Hygromycin a compounds and methods of treating spirochete diseases |
CR20220316A (es) | 2019-12-06 | 2022-10-07 | Vertex Pharma | Tetrahidrofuranos sustituidos como moduladores de canales de sodio |
WO2022256622A1 (en) | 2021-06-04 | 2022-12-08 | Vertex Pharmaceuticals Incorporated | N-(hydroxyalkyl (hetero)aryl) tetrahydrofuran carboxamides as modulators of sodium channels |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100418167B1 (ko) * | 1998-12-02 | 2004-02-11 | 화이자 프로덕츠 인크. | 항균제로서의 하이그로마이신 a 유도체 |
-
2000
- 2000-10-09 BR BR0015153-0A patent/BR0015153A/pt not_active IP Right Cessation
- 2000-10-09 AU AU75494/00A patent/AU7549400A/en not_active Abandoned
- 2000-10-09 CA CA002389191A patent/CA2389191A1/en not_active Abandoned
- 2000-10-09 SK SK547-2002A patent/SK5472002A3/sk not_active Application Discontinuation
- 2000-10-09 PL PL00357083A patent/PL357083A1/xx not_active Application Discontinuation
- 2000-10-09 WO PCT/IB2000/001461 patent/WO2001030795A1/en not_active Application Discontinuation
- 2000-10-09 HU HU0203525A patent/HUP0203525A3/hu unknown
- 2000-10-09 AP APAP/P/2002/002494A patent/AP2002002494A0/en unknown
- 2000-10-09 TR TR2002/01145T patent/TR200201145T2/tr unknown
- 2000-10-09 MX MXPA02004360A patent/MXPA02004360A/es active IP Right Grant
- 2000-10-09 EP EP00964572A patent/EP1224197A1/en not_active Withdrawn
- 2000-10-09 IL IL14857700A patent/IL148577A0/xx unknown
- 2000-10-09 EA EA200200292A patent/EA200200292A1/ru unknown
- 2000-10-09 OA OA1200200129A patent/OA12081A/en unknown
- 2000-10-09 CZ CZ20021355A patent/CZ20021355A3/cs unknown
- 2000-10-09 JP JP2001533146A patent/JP2003512473A/ja active Pending
- 2000-10-09 KR KR1020027005533A patent/KR20020063885A/ko not_active Application Discontinuation
- 2000-10-09 EE EEP200200228A patent/EE200200228A/xx unknown
- 2000-10-09 CN CN00814843A patent/CN1382150A/zh active Pending
- 2000-10-20 US US09/693,118 patent/US6562792B1/en not_active Expired - Fee Related
- 2000-10-25 CO CO00081374A patent/CO5261498A1/es not_active Application Discontinuation
- 2000-10-25 GT GT200000185A patent/GT200000185A/es unknown
- 2000-10-26 PA PA20008505801A patent/PA8505801A1/es unknown
- 2000-10-26 PE PE2000001146A patent/PE20010763A1/es not_active Application Discontinuation
- 2000-10-27 TN TNTNSN00211A patent/TNSN00211A1/fr unknown
- 2000-10-27 SV SV2000000211A patent/SV2002000211A/es unknown
- 2000-10-27 AR ARP000105698A patent/AR023282A1/es not_active Application Discontinuation
-
2002
- 2002-03-19 IS IS6311A patent/IS6311A/is unknown
- 2002-04-19 NO NO20021850A patent/NO20021850D0/no not_active Application Discontinuation
- 2002-04-22 MA MA26613A patent/MA26838A1/fr unknown
- 2002-05-20 BG BG106727A patent/BG106727A/bg unknown
-
2003
- 2003-03-14 HK HK03101860.2A patent/HK1049672A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
GT200000185A (es) | 2002-04-18 |
NO20021850L (no) | 2002-04-19 |
OA12081A (en) | 2006-05-04 |
EE200200228A (et) | 2003-06-16 |
AR023282A1 (es) | 2002-09-04 |
IS6311A (is) | 2002-03-19 |
HUP0203525A3 (en) | 2003-08-28 |
JP2003512473A (ja) | 2003-04-02 |
CN1382150A (zh) | 2002-11-27 |
SV2002000211A (es) | 2002-07-16 |
TNSN00211A1 (fr) | 2005-11-10 |
AP2002002494A0 (en) | 2002-06-30 |
PA8505801A1 (es) | 2002-08-26 |
IL148577A0 (en) | 2002-09-12 |
PE20010763A1 (es) | 2001-07-25 |
PL357083A1 (en) | 2004-07-12 |
MA26838A1 (fr) | 2004-12-20 |
US6562792B1 (en) | 2003-05-13 |
EA200200292A1 (ru) | 2002-10-31 |
KR20020063885A (ko) | 2002-08-05 |
CZ20021355A3 (cs) | 2002-11-13 |
CA2389191A1 (en) | 2001-05-03 |
BR0015153A (pt) | 2002-07-16 |
HUP0203525A2 (hu) | 2003-02-28 |
HK1049672A1 (zh) | 2003-05-23 |
WO2001030795A1 (en) | 2001-05-03 |
SK5472002A3 (en) | 2003-02-04 |
EP1224197A1 (en) | 2002-07-24 |
AU7549400A (en) | 2001-05-08 |
BG106727A (bg) | 2003-01-31 |
NO20021850D0 (no) | 2002-04-19 |
CO5261498A1 (es) | 2003-03-31 |
MXPA02004360A (es) | 2002-11-07 |
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