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TN2010000333A1 - Bicyclic derivativesof azabicyclic carboxamides, preparation thereof and therapeutic use thereof - Google Patents

Bicyclic derivativesof azabicyclic carboxamides, preparation thereof and therapeutic use thereof

Info

Publication number
TN2010000333A1
TN2010000333A1 TNP2010000333A TN2010000333A TN2010000333A1 TN 2010000333 A1 TN2010000333 A1 TN 2010000333A1 TN P2010000333 A TNP2010000333 A TN P2010000333A TN 2010000333 A TN2010000333 A TN 2010000333A TN 2010000333 A1 TN2010000333 A1 TN 2010000333A1
Authority
TN
Tunisia
Prior art keywords
preparation
therapeutic use
heteroaryl
derivativesof
azabicyclic
Prior art date
Application number
TNP2010000333A
Other languages
French (fr)
Inventor
Laurent Dubois
Yannick Evanno
Catherine Gille
Andre Malanda
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/FR2009/000051 external-priority patent/WO2009112677A2/en
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of TN2010000333A1 publication Critical patent/TN2010000333A1/en

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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The invention relates to the compounds of general formula (1) in which X1, X2, X3 and X4 are, independently of one another, a nitrogen atom or a C-Ri group; W is an oxygen or sulphur atom; n is equal to 0, 1, 2 or 3; Y is an optionally substituted aryl or heteroaryl; A is the group of formula: (II), Z1, Z2, Z3 and Z4 are, independently of one another, a nitrogen atom or a C-R2 group; Ra and Rb form, together with the carbon atoms which bear them, either a partially unsaturated cycloalkyl, or an aryl; or a heterocycle, or a heteroaryl with 5 to 7 ring members comprising from one to three heteroatoms selected from O, S or N; it being possible for this cycloalkyl, this aryl, this heterocycle or this heteroaryl to be substituted with one or more substituents R3; in the form of a base or of an addition salt with an acid, and also in the form of a hydrate or of a solvate. Process for the preparation thereof and therapeutic use.
TNP2010000333A 2009-01-20 2010-07-19 Bicyclic derivativesof azabicyclic carboxamides, preparation thereof and therapeutic use thereof TN2010000333A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/FR2009/000051 WO2009112677A2 (en) 2008-01-22 2009-01-20 Bicyclic derivatives of azabicyclic carboxamides, preparation thereof and therapeutic use thereof

Publications (1)

Publication Number Publication Date
TN2010000333A1 true TN2010000333A1 (en) 2011-12-29

Family

ID=55024465

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2010000333A TN2010000333A1 (en) 2009-01-20 2010-07-19 Bicyclic derivativesof azabicyclic carboxamides, preparation thereof and therapeutic use thereof

Country Status (1)

Country Link
TN (1) TN2010000333A1 (en)

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