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SG11201506918WA - Inhibitors of indoleamine 2,3-dioxygenase (ido) - Google Patents

Inhibitors of indoleamine 2,3-dioxygenase (ido)

Info

Publication number
SG11201506918WA
SG11201506918WA SG11201506918WA SG11201506918WA SG11201506918WA SG 11201506918W A SG11201506918W A SG 11201506918WA SG 11201506918W A SG11201506918W A SG 11201506918WA SG 11201506918W A SG11201506918W A SG 11201506918WA SG 11201506918W A SG11201506918W A SG 11201506918WA
Authority
SG
Singapore
Prior art keywords
indoleamine
ido
dioxygenase
inhibitors
Prior art date
Application number
SG11201506918WA
Inventor
James Aaron Balog
Audris Huang
Bin Chen
Libing Chen
Steven P Seitz
Amy C Hart
Jay A Markwalder
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of SG11201506918WA publication Critical patent/SG11201506918WA/en

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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
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    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
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    • A61K31/27—Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
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