SA520411943B1 - تصنيع مركبات بنزيميدازول مستبدلة عند الموضع-2 - Google Patents
تصنيع مركبات بنزيميدازول مستبدلة عند الموضع-2Info
- Publication number
- SA520411943B1 SA520411943B1 SA520411943A SA520411943A SA520411943B1 SA 520411943 B1 SA520411943 B1 SA 520411943B1 SA 520411943 A SA520411943 A SA 520411943A SA 520411943 A SA520411943 A SA 520411943A SA 520411943 B1 SA520411943 B1 SA 520411943B1
- Authority
- SA
- Saudi Arabia
- Prior art keywords
- substituted benzimidazoles
- manufacture
- compositions
- aqueous system
- corrosion
- Prior art date
Links
- -1 2-Substituted Benzimidazoles Chemical class 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title 1
- 238000005260 corrosion Methods 0.000 abstract 2
- 230000007797 corrosion Effects 0.000 abstract 2
- 239000002184 metal Substances 0.000 abstract 2
- 229910052751 metal Inorganic materials 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000002739 metals Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000003880 polar aprotic solvent Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/08—Radicals containing only hydrogen and carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/12—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/18—Benzimidazoles; Hydrogenated benzimidazoles with aryl radicals directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C23—COATING METALLIC MATERIAL; COATING MATERIAL WITH METALLIC MATERIAL; CHEMICAL SURFACE TREATMENT; DIFFUSION TREATMENT OF METALLIC MATERIAL; COATING BY VACUUM EVAPORATION, BY SPUTTERING, BY ION IMPLANTATION OR BY CHEMICAL VAPOUR DEPOSITION, IN GENERAL; INHIBITING CORROSION OF METALLIC MATERIAL OR INCRUSTATION IN GENERAL
- C23F—NON-MECHANICAL REMOVAL OF METALLIC MATERIAL FROM SURFACE; INHIBITING CORROSION OF METALLIC MATERIAL OR INCRUSTATION IN GENERAL; MULTI-STEP PROCESSES FOR SURFACE TREATMENT OF METALLIC MATERIAL INVOLVING AT LEAST ONE PROCESS PROVIDED FOR IN CLASS C23 AND AT LEAST ONE PROCESS COVERED BY SUBCLASS C21D OR C22F OR CLASS C25
- C23F11/00—Inhibiting corrosion of metallic material by applying inhibitors to the surface in danger of corrosion or adding them to the corrosive agent
- C23F11/08—Inhibiting corrosion of metallic material by applying inhibitors to the surface in danger of corrosion or adding them to the corrosive agent in other liquids
- C23F11/10—Inhibiting corrosion of metallic material by applying inhibitors to the surface in danger of corrosion or adding them to the corrosive agent in other liquids using organic inhibitors
- C23F11/14—Nitrogen-containing compounds
- C23F11/149—Heterocyclic compounds containing nitrogen as hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Materials Engineering (AREA)
- Mechanical Engineering (AREA)
- Metallurgy (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Preventing Corrosion Or Incrustation Of Metals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
يتم الكشف عن مركبات بنزيميدازول مستبدلة عند الموضع-2 وطرق تحضيرها. يمكن أن تتضمن التركيبات مركب أو ملح منه، وحمض، ومذيب لا بروتوني قطبي polar aprotic solvent. يمكن استخدام التركيبات لتثبيط تآكل inhibit corrosion سطح معدني متلامس مع نظام مائي، وتوفير حماية معزَّزة ضد تآكل المعادن في النظام المائي. الصيغة (I)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201762585278P | 2017-11-13 | 2017-11-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
SA520411943B1 true SA520411943B1 (ar) | 2024-08-07 |
Family
ID=64572508
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SA520411943A SA520411943B1 (ar) | 2017-11-13 | 2020-05-11 | تصنيع مركبات بنزيميدازول مستبدلة عند الموضع-2 |
Country Status (12)
Country | Link |
---|---|
US (1) | US11053203B2 (ar) |
EP (1) | EP3710436A1 (ar) |
JP (1) | JP2021502401A (ar) |
KR (1) | KR102653426B1 (ar) |
CN (1) | CN111372924B (ar) |
AU (1) | AU2018366253B2 (ar) |
CA (1) | CA3082375A1 (ar) |
MX (1) | MX2020004901A (ar) |
SA (1) | SA520411943B1 (ar) |
SG (1) | SG11202004310YA (ar) |
TW (1) | TWI823873B (ar) |
WO (1) | WO2019094672A1 (ar) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2020176604A1 (en) | 2019-02-28 | 2020-09-03 | Ecolab Usa Inc. | Hydrogen sulfide scavengers for asphalt |
CN110776467A (zh) * | 2019-10-30 | 2020-02-11 | 西南石油大学 | 一种基于苯并咪唑衍生物的缓蚀剂及其制备方法和应用 |
EP4127268A1 (en) | 2020-03-27 | 2023-02-08 | Ecolab Usa Inc. | Galvanized metal corrosion inhibitor compositions and methods of use |
US20230053321A1 (en) * | 2021-08-02 | 2023-02-16 | Ecolab Usa Inc. | One-pot homogeneous process for the large scale manufacture of 2-substituted benzimidazoles |
US20230416128A1 (en) | 2022-06-23 | 2023-12-28 | Ecolab Usa Inc. | Method of Inhibiting Corrosion of a Metal in an Industrial Water System |
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DE1176659B (de) | 1960-12-27 | 1964-08-27 | Beiersdorf & Co A G P | Verfahren zur Herstellung von 1-(ª‰-Diaethyl-amino-aethyl)-2-(ª‡-hydroxy-p-methoxy-benzyl)-5-nitro-benzimidazol und seinem Hydrochlorid |
US3784517A (en) | 1972-06-27 | 1974-01-08 | Us Air Force | Preparation of polybenzimidazoles in the presence of a sulfone solvent |
US4001268A (en) | 1974-08-07 | 1977-01-04 | The United States Of America As Represented By The Secretary Of The Air Force | Substituted phenyl-benzimidazo compounds |
DE2900506A1 (de) | 1979-01-08 | 1980-07-17 | Basf Ag | Verfahren zur herstellung von 2-cyanmethylbenzimidazol |
SU819098A1 (ru) | 1979-01-17 | 1981-04-07 | Предприятие П/Я Р-6875 | Способ получени 2-метилбензимидазола |
SU1164232A1 (ru) | 1983-05-11 | 1985-06-30 | Ферганский политехнический институт | Способ получени 2-ацетиламинобензимидазола |
DE4305714A1 (de) | 1993-02-25 | 1994-09-01 | Hoechst Ag | Verfahren zur Herstellung von substituiertem und unsubstituiertem 2-(Cyanmethyl)benzimidazol |
DE19539114C1 (de) | 1995-10-20 | 1997-04-17 | Hoechst Ag | Verfahren zur Aufarbeitung von Benzimidazolone enthaltenden Reaktionsgemischen |
DE10201725A1 (de) | 2002-01-18 | 2003-08-14 | Boehringer Ingelheim Pharma | Verfahren zur Herstellung und Reinigung von 1,7'-Dimethyl-2'-propyl-2,5'-bi-1H-benzimidazol |
EP1814865A4 (en) | 2004-09-21 | 2009-09-02 | Wyeth Corp | BENZIMIDAZOL ACETIC ACIDS WITH CRTH2 RECEPTOR ANTAGONISM AND ITS APPLICATIONS |
WO2006132625A1 (en) * | 2005-06-03 | 2006-12-14 | Ppg Industries Ohio, Inc. | Composition for the vapor phase dehydrohalogenation of 1,1,2-trihaloethane to 1,1-dihaloethylene and methods for preparing and using such compositions |
DE102005034279A1 (de) | 2005-07-22 | 2007-01-25 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Herstellung von 1,7'-Dimethyl-2'-propyl-2,5'-bi-1H-benzimidazol |
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WO2009116089A2 (en) | 2008-03-14 | 2009-09-24 | Ipca Laboratories Limited | Novel intermediates and method for synthesis of 4'-[(1,4'-dimethyl-2'-propyl-[2,6'- bi-1hbenzimidazol]-l-yl)methyl]-1,1-biphenyl]-2-carboxylic acid. |
EP2280947B1 (de) | 2008-05-02 | 2014-11-26 | Boehringer Ingelheim International GmbH | Herstellung von 1,7´-dimethyl-2´-propyl-2,5´-bi-1h-benzimidazol |
CN101891689B (zh) | 2010-07-23 | 2012-04-18 | 江苏先声药物研究有限公司 | 盐酸γ-羟基苯达莫司汀的制备方法 |
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-
2018
- 2018-11-09 KR KR1020207014944A patent/KR102653426B1/ko active IP Right Grant
- 2018-11-09 CA CA3082375A patent/CA3082375A1/en active Pending
- 2018-11-09 US US16/185,304 patent/US11053203B2/en active Active
- 2018-11-09 JP JP2020526295A patent/JP2021502401A/ja active Pending
- 2018-11-09 EP EP18812476.2A patent/EP3710436A1/en active Pending
- 2018-11-09 AU AU2018366253A patent/AU2018366253B2/en active Active
- 2018-11-09 SG SG11202004310YA patent/SG11202004310YA/en unknown
- 2018-11-09 MX MX2020004901A patent/MX2020004901A/es unknown
- 2018-11-09 CN CN201880075983.1A patent/CN111372924B/zh active Active
- 2018-11-09 WO PCT/US2018/059947 patent/WO2019094672A1/en active Application Filing
- 2018-11-13 TW TW107140167A patent/TWI823873B/zh active
-
2020
- 2020-05-11 SA SA520411943A patent/SA520411943B1/ar unknown
Also Published As
Publication number | Publication date |
---|---|
AU2018366253A1 (en) | 2020-05-21 |
CN111372924B (zh) | 2023-09-19 |
KR102653426B1 (ko) | 2024-03-29 |
WO2019094672A1 (en) | 2019-05-16 |
RU2020119396A (ru) | 2021-12-15 |
CA3082375A1 (en) | 2019-05-16 |
US20190144395A1 (en) | 2019-05-16 |
JP2021502401A (ja) | 2021-01-28 |
KR20200087779A (ko) | 2020-07-21 |
TW201922715A (zh) | 2019-06-16 |
SG11202004310YA (en) | 2020-06-29 |
CN111372924A (zh) | 2020-07-03 |
MX2020004901A (es) | 2020-09-09 |
US11053203B2 (en) | 2021-07-06 |
BR112020009285A2 (pt) | 2020-10-27 |
AU2018366253B2 (en) | 2024-05-02 |
TWI823873B (zh) | 2023-12-01 |
EP3710436A1 (en) | 2020-09-23 |
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