RU94045866A - Применение бисфенилалкилпиперазинов для лечения расстройств, вызванных злоупотреблением веществами, способ лечения - Google Patents
Применение бисфенилалкилпиперазинов для лечения расстройств, вызванных злоупотреблением веществами, способ леченияInfo
- Publication number
- RU94045866A RU94045866A RU94045866/14A RU94045866A RU94045866A RU 94045866 A RU94045866 A RU 94045866A RU 94045866/14 A RU94045866/14 A RU 94045866/14A RU 94045866 A RU94045866 A RU 94045866A RU 94045866 A RU94045866 A RU 94045866A
- Authority
- RU
- Russia
- Prior art keywords
- treatment
- phenylalkylpiperazines
- bis
- substance abuse
- substance
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/43—Enzymes; Proenzymes; Derivatives thereof
- A61K38/46—Hydrolases (3)
- A61K38/48—Hydrolases (3) acting on peptide bonds (3.4)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Addiction (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
- Compounds Of Unknown Constitution (AREA)
Abstract
Способ для ослабления или профилактики абстинентного синдрома, являющегося результатом чрезмерного употребления лекарственного средства или вещества злоупотребления и/или для подавления зависимости от лекарств или веществ зависимости, который включает применение эффективного количества бисфенилалкилпиперазинов и их фармацевтически приемлемых солей, полученных в результате присоединения кислоты.
Claims (1)
- Способ для ослабления или профилактики абстинентного синдрома, являющегося результатом чрезмерного употребления лекарственного средства или вещества злоупотребления и/или для подавления зависимости от лекарств или веществ зависимости, который включает применение эффективного количества бисфенилалкилпиперазинов и их фармацевтически приемлемых солей, полученных в результате присоединения кислоты.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE9201239-2 | 1992-04-21 | ||
SE9201239A SE9201239D0 (sv) | 1992-04-21 | 1992-04-21 | Agents for treating substance abuse disorders |
PCT/SE1993/000339 WO1993020821A1 (en) | 1992-04-21 | 1993-04-19 | Agents for treating substance abuse disorders |
Publications (2)
Publication Number | Publication Date |
---|---|
RU94045866A true RU94045866A (ru) | 1996-10-20 |
RU2126254C1 RU2126254C1 (ru) | 1999-02-20 |
Family
ID=20386004
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU94045866A RU2126254C1 (ru) | 1992-04-21 | 1993-04-19 | Применение бисфенилалкилпиперазинов для лечения расстройств, вызванных злоупотреблением веществами, и способ лечения |
Country Status (26)
Country | Link |
---|---|
US (1) | US5565455A (ru) |
EP (1) | EP0637242B1 (ru) |
JP (1) | JP3245642B2 (ru) |
KR (1) | KR100321319B1 (ru) |
AT (1) | ATE184484T1 (ru) |
AU (1) | AU659941B2 (ru) |
BG (1) | BG62154B1 (ru) |
BR (1) | BR9306361A (ru) |
CA (1) | CA2118512C (ru) |
CZ (1) | CZ281296B6 (ru) |
DE (1) | DE69326459T2 (ru) |
DK (1) | DK0637242T3 (ru) |
EE (1) | EE02974B1 (ru) |
ES (1) | ES2139007T3 (ru) |
GR (1) | GR3032030T3 (ru) |
HU (1) | HU223463B1 (ru) |
IL (1) | IL105449A (ru) |
NO (2) | NO308827B1 (ru) |
PH (1) | PH31051A (ru) |
RO (1) | RO117150B1 (ru) |
RU (1) | RU2126254C1 (ru) |
SE (1) | SE9201239D0 (ru) |
SK (1) | SK279940B6 (ru) |
UA (1) | UA27884C2 (ru) |
WO (1) | WO1993020821A1 (ru) |
ZA (1) | ZA932757B (ru) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5316759A (en) * | 1986-03-17 | 1994-05-31 | Robert J. Schaap | Agonist-antagonist combination to reduce the use of nicotine and other drugs |
SE9201956D0 (sv) * | 1992-06-25 | 1992-06-25 | Kabi Pharmacia Ab | Novel nicotinicacid esters |
SE9601708D0 (sv) | 1996-05-06 | 1996-05-06 | Pharmacia Ab | Pyridyl- and pyrimidyl-piperazines in the treatment of substance abuse disorders |
AU744539B2 (en) | 1997-10-27 | 2002-02-28 | Neurosearch A/S | Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors |
US6632823B1 (en) * | 1997-12-22 | 2003-10-14 | Merck & Co., Inc. | Substituted pyridine compounds useful as modulators of acetylcholine receptors |
US6344222B1 (en) | 1998-09-03 | 2002-02-05 | Jsr Llc | Medicated chewing gum delivery system for nicotine |
US6358060B2 (en) | 1998-09-03 | 2002-03-19 | Jsr Llc | Two-stage transmucosal medicine delivery system for symptom relief |
US6090780A (en) * | 1999-04-07 | 2000-07-18 | Chandon Prasad | Histidyl-proline diketopiperazine and method of use |
PT1551372T (pt) | 2002-09-20 | 2018-07-23 | Alpharma Pharmaceuticals Llc | Subunidade de sequestração e composições e métodos relacionados |
KR101486228B1 (ko) | 2006-06-19 | 2015-01-26 | 알파마 파머슈티컬스 엘엘씨 | 약제학적 조성물 |
US8642016B2 (en) | 2006-07-21 | 2014-02-04 | Jsrnti, Llc | Medicinal delivery system, and related methods |
US8623418B2 (en) | 2007-12-17 | 2014-01-07 | Alpharma Pharmaceuticals Llc | Pharmaceutical composition |
BRPI1003506B1 (pt) | 2010-09-24 | 2019-12-03 | Ache Int Bvi Ltd | composto alquil-piperazino-fenil-4(3h)quinazolinonas e uso do composto alquil-piperazino-fenil-4(3h)quinazolinonas associado aos receptores serotoninérgicos 5-ht1a e 5-ht2a |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2958694A (en) * | 1959-06-22 | 1960-11-01 | Janssen Paul Adriaan Jan | 1-(aroylalkyl)-4-(2'-pyridyl) piperazines |
US2985657A (en) * | 1959-10-12 | 1961-05-23 | Paul A J Janssen | 1-(aroylalkyl)-4-heterocyclylpiperazines |
US2979508A (en) * | 1959-10-12 | 1961-04-11 | Paul A J Janssen | Heterocyclic derivatives of 1-phenyl-omega-(piperazine) alkanols |
NO154582C (no) * | 1978-10-20 | 1986-11-05 | Ferrosan Ab | Analogifremgangsmaate for fremstilling av terapeutisk aktive difenyl-dibutylpiperazinkarboksamider. |
US4605655A (en) * | 1984-03-06 | 1986-08-12 | Bristol-Myers Company | Antipsychotic 1-fluorophenylbutyl-4-(2-pyrimidinyl)piperazine derivatives |
US4766215A (en) * | 1987-02-27 | 1988-08-23 | American Home Products Corporation | Histamine H1 -receptor antagonists |
SE8701375D0 (sv) * | 1987-04-02 | 1987-04-02 | Leo Ab | Novel pyridyl- and pyrimidyl derivatives |
US5217987A (en) * | 1989-10-30 | 1993-06-08 | Berger Stephen P | Dopamine uptake inhibitors in reducing substance abuse and/or craving |
SE9100860D0 (sv) * | 1991-03-22 | 1991-03-22 | Kabi Pharmacia Ab | New use |
-
1992
- 1992-04-21 SE SE9201239A patent/SE9201239D0/xx unknown
-
1993
- 1993-04-19 HU HU9403020A patent/HU223463B1/hu not_active IP Right Cessation
- 1993-04-19 UA UA94105949A patent/UA27884C2/uk unknown
- 1993-04-19 BR BR9306361A patent/BR9306361A/pt not_active Application Discontinuation
- 1993-04-19 US US08/325,212 patent/US5565455A/en not_active Expired - Lifetime
- 1993-04-19 IL IL105449A patent/IL105449A/en not_active IP Right Cessation
- 1993-04-19 DE DE69326459T patent/DE69326459T2/de not_active Expired - Fee Related
- 1993-04-19 SK SK1269-94A patent/SK279940B6/sk not_active IP Right Cessation
- 1993-04-19 AT AT93911554T patent/ATE184484T1/de not_active IP Right Cessation
- 1993-04-19 EP EP93911554A patent/EP0637242B1/en not_active Expired - Lifetime
- 1993-04-19 CZ CZ942606A patent/CZ281296B6/cs not_active IP Right Cessation
- 1993-04-19 WO PCT/SE1993/000339 patent/WO1993020821A1/en active IP Right Grant
- 1993-04-19 DK DK93911554T patent/DK0637242T3/da active
- 1993-04-19 RU RU94045866A patent/RU2126254C1/ru active
- 1993-04-19 JP JP51825193A patent/JP3245642B2/ja not_active Expired - Fee Related
- 1993-04-19 RO RO94-01692A patent/RO117150B1/ro unknown
- 1993-04-19 ES ES93911554T patent/ES2139007T3/es not_active Expired - Lifetime
- 1993-04-19 AU AU40437/93A patent/AU659941B2/en not_active Ceased
- 1993-04-19 CA CA002118512A patent/CA2118512C/en not_active Expired - Fee Related
- 1993-04-20 ZA ZA932757A patent/ZA932757B/xx unknown
- 1993-04-21 PH PH46084A patent/PH31051A/en unknown
-
1994
- 1994-10-19 BG BG99129A patent/BG62154B1/bg unknown
- 1994-10-20 NO NO943977A patent/NO308827B1/no not_active IP Right Cessation
- 1994-10-21 KR KR1019940703758A patent/KR100321319B1/ko not_active IP Right Cessation
- 1994-11-17 EE EE9400398A patent/EE02974B1/xx not_active IP Right Cessation
-
1999
- 1999-12-02 GR GR990403117T patent/GR3032030T3/el unknown
-
2000
- 2000-08-21 NO NO20004169A patent/NO318461B1/no not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
RU94041223A (ru) | Средство для лечения мотонейроновых заболеваний | |
SE9802073D0 (sv) | New use | |
GEP20002298B (en) | Benzimidazole Derivatives, Method of Their Production, Pharmaceutical Composition Containing the Same and Method for Its Treatment | |
GEP20033131B (en) | Azabicycloalkanes as CCR5 Modulators, Pharmaceutical Compositions Containing the Same and Their Use for Treatment and Prevention of Diseases Caused by CCR5 Activity | |
RU94045866A (ru) | Применение бисфенилалкилпиперазинов для лечения расстройств, вызванных злоупотреблением веществами, способ лечения | |
DE69731610D1 (de) | Orale verabreichung wirksamer mengen von hyaluronsäure | |
KR880011197A (ko) | 위장장해를 치료하기 위한 조성물 및 방법 | |
MY111260A (en) | Pharmaceutical composition for the treatment of nicotine dependence | |
KR910019618A (ko) | 발기부전증 치료용 제약 조성물 | |
DE69733089D1 (de) | Behandlung der osteoarthritis durch verabreichung von poly-n-acetyl-d-glucosamin | |
ATE15596T1 (de) | Pharmazeutische mittel. | |
RU95105973A (ru) | Способ снижения тяжести токсоплазмоза, фармацевтическая композиция, применение производных рифамицина для получения лекарственных препаратов для лечения токсоплазмоза | |
RU95101385A (ru) | Продукты, содержащие g-csf и tnf связующие протеина | |
CA2270955A1 (en) | Pharmaceutical composition containing morphinan derivative for treating drug dependence | |
KR950016760A (ko) | 치질 치료제 | |
CA2156481A1 (en) | 5-ht2 receptor antagonist compositions useful in treating venous conditions | |
ATE356637T1 (de) | Supramolekulare komplexe enthaltende arzneimittel | |
KR920000326A (ko) | 사람에 있어서 몰핀 및 동족체의 진통 효과에 대한 내성 발생을 방지하기 위한 gm₁모노시알로강글리오사이드 및 이의 내부 에스테르 유도체의 용도 | |
KR960706341A (ko) | 유기 인 콜린스테라아제 억제제에 의해 야기되는 중독의 예방 및 예비 치료를 위한 약제 제형(pharmaceutical formulation for preventing or pre-treating poisoning by organophosphoric cholinesterase inhibitors) | |
RU2209064C2 (ru) | Новое применение в медицинских целях | |
RU98101105A (ru) | Новое применение в медицинских целях | |
CA2394471A1 (en) | External preparation for treating pruritus | |
KR900701278A (ko) | 바이러스 감염 치료용 담즙산 | |
RU94032792A (ru) | Применение 5нтiа - антагонистов для прекращения использования табака | |
IE790157L (en) | Therapeutic agents |