PT68102B - Process for the preparation of alpha-fluoromethyl-alpha-amino alkanoic acids - Google Patents

Process for the preparation of alpha-fluoromethyl-alpha-amino alkanoic acids

Info

Publication number: PT68102B
Authority: PT; Portugal
Prior art keywords: alpha; fluoromethyl; preparation; alkanoic acids; amino alkanoic
Prior art date: 1977-06-01

Application number

PT68102A

Other languages

Portuguese (pt)

Other versions

PT68102A (en

Original Assignee

Merck & Co Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-06-01

Filing date

1978-05-30

Publication date

1982-06-08

1977-06-01 Priority claimed from US05/802,391 external-priority patent/US4325961A/en

1978-05-30 Application filed by Merck & Co Inc filed Critical Merck & Co Inc

1978-06-01 Publication of PT68102A publication Critical patent/PT68102A/en

1982-06-08 Publication of PT68102B publication Critical patent/PT68102B/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)

PT68102A 1977-06-01 1978-05-30 Process for the preparation of alpha-fluoromethyl-alpha-amino alkanoic acids PT68102B (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US80238977A	1977-06-01	1977-06-01
US05/802,391 US4325961A (en)	1977-06-01	1977-06-01	Fluorinated amino acids

Publications (2)

Publication Number	Publication Date
PT68102A PT68102A (en)	1978-06-01
PT68102B true PT68102B (en)	1982-06-08

Family

ID=27122442

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT68102A PT68102B (en)	1977-06-01	1978-05-30	Process for the preparation of alpha-fluoromethyl-alpha-amino alkanoic acids

Country Status (26)

Country	Link
JP (1)	JPS5416423A (en)
AR (1)	AR223463A1 (en)
AT (1)	AT360509B (en)
AU (1)	AU518479B2 (en)
CA (1)	CA1120040A (en)
CH (1)	CH639639A5 (en)
DD (1)	DD138651A5 (en)
DE (1)	DE2824116A1 (en)
DK (1)	DK149841C (en)
ES (1)	ES470296A1 (en)
FI (1)	FI66840C (en)
FR (1)	FR2392958A1 (en)
GB (1)	GB1602525A (en)
GR (1)	GR64495B (en)
HK (1)	HK18184A (en)
HU (1)	HU181911B (en)
IE (1)	IE46983B1 (en)
IT (1)	IT1104709B (en)
LU (1)	LU79750A1 (en)
NL (1)	NL190485C (en)
NO (1)	NO147382C (en)
NZ (1)	NZ187377A (en)
PL (1)	PL115731B1 (en)
PT (1)	PT68102B (en)
SE (1)	SE7806440L (en)
YU (1)	YU129178A (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1091661A (en) *	1977-07-11	1980-12-16	Philippe Bey	.alpha.-HALOMETHYL DERIVATIVES OF .alpha.-AMINO ACIDS
IL59481A0 (en) *	1977-07-11	1980-05-30	Merrell Toraude & Co	-halomethyl amino acids
ZA783273B (en) *	1977-07-11	1979-06-27	Merrell Toraude & Co	A-halomethyl amino acids
US4315095A (en) *	1977-07-28	1982-02-09	Merrell Toraude Et Compagnie	α-Halomethyl derivatives of amino acids
DE2965364D1 (en) *	1978-07-24	1983-06-16	Merck & Co Inc	Alpha-difluoromethyl amino acids and pharmaceutical composition containing the same
IE49522B1 (en) *	1979-04-26	1985-10-16	Merrell Toraude & Co	Alpha-halomethylaminoacids
NZ194347A (en) *	1979-07-26	1982-11-23	Merrell Toraude & Co	Fluorinated alkenylamines intermediate alkenyl fluorinated methyl ketimine magnesium halides and preparation of certain amino alkanoic acids
ZA813018B (en) *	1980-05-09	1982-05-26	Merrell Toraude & Co	Fluoromethylated tyrosine methyl ester
PH16634A (en) *	1980-06-16	1983-12-05	Merrell Dow Pharma	Method of inhibiting the growth of protozoa
US4421767A (en) *	1981-06-01	1983-12-20	Merrell Toraude Et Compagnie	Compounds and methods for treating depression
GB9325368D0 (en) *	1993-12-10	1994-02-16	Univ Bristol	Organic compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3046300A (en) *	1960-10-21	1962-07-24	Merck & Co Inc	alpha-trifluoromethyloxyphenylalanines

1978
- 1978-05-25 FR FR7815567A patent/FR2392958A1/en active Granted
- 1978-05-25 NZ NZ187377A patent/NZ187377A/en unknown
- 1978-05-25 GR GR56328A patent/GR64495B/en unknown
- 1978-05-26 FI FI781674A patent/FI66840C/en not_active IP Right Cessation
- 1978-05-26 AR AR272336A patent/AR223463A1/en active
- 1978-05-29 AU AU36586/78A patent/AU518479B2/en not_active Expired
- 1978-05-29 CA CA000304318A patent/CA1120040A/en not_active Expired
- 1978-05-29 ES ES470296A patent/ES470296A1/en not_active Expired
- 1978-05-30 DD DD78205669A patent/DD138651A5/en unknown
- 1978-05-30 IE IE1078/78A patent/IE46983B1/en unknown
- 1978-05-30 PT PT68102A patent/PT68102B/en unknown
- 1978-05-30 YU YU01291/78A patent/YU129178A/en unknown
- 1978-05-30 GB GB24330/78A patent/GB1602525A/en not_active Expired
- 1978-05-30 DK DK237978A patent/DK149841C/en not_active IP Right Cessation
- 1978-05-30 AT AT393278A patent/AT360509B/en not_active IP Right Cessation
- 1978-05-30 HU HU78ME2169A patent/HU181911B/en unknown
- 1978-05-31 IT IT49637/78A patent/IT1104709B/en active
- 1978-05-31 NO NO781892A patent/NO147382C/en unknown
- 1978-05-31 CH CH597978A patent/CH639639A5/en not_active IP Right Cessation
- 1978-05-31 PL PL1978207242A patent/PL115731B1/en unknown
- 1978-06-01 DE DE19782824116 patent/DE2824116A1/en active Granted
- 1978-06-01 LU LU79750A patent/LU79750A1/en unknown
- 1978-06-01 NL NLAANVRAGE7805981,A patent/NL190485C/en not_active IP Right Cessation
- 1978-06-01 JP JP6501678A patent/JPS5416423A/en active Granted
- 1978-06-01 SE SE7806440A patent/SE7806440L/en unknown
1984
- 1984-03-01 HK HK181/84A patent/HK18184A/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
LU79750A1 (en)	1979-02-02
DK149841B (en)	1986-10-13
FR2392958A1 (en)	1978-12-29
NO147382B (en)	1982-12-20
NZ187377A (en)	1981-05-15
PL207242A1 (en)	1979-04-23
GR64495B (en)	1980-03-31
FI66840B (en)	1984-08-31
ATA393278A (en)	1980-06-15
PL115731B1 (en)	1981-04-30
ES470296A1 (en)	1979-09-16
DE2824116A1 (en)	1978-12-14
PT68102A (en)	1978-06-01
DE2824116C2 (en)	1989-04-27
NO781892L (en)	1978-12-04
IT1104709B (en)	1985-10-28
NL190485C (en)	1994-03-16
FI66840C (en)	1984-12-10
SE7806440L (en)	1978-12-02
GB1602525A (en)	1981-11-11
CA1120040A (en)	1982-03-16
AR223463A1 (en)	1981-08-31
NO147382C (en)	1983-03-30
AU3658678A (en)	1979-12-06
NL7805981A (en)	1978-12-05
JPS5416423A (en)	1979-02-07
HU181911B (en)	1983-11-28
DD138651A5 (en)	1979-11-14
DK149841C (en)	1987-04-21
HK18184A (en)	1984-03-09
CH639639A5 (en)	1983-11-30
FI781674A (en)	1978-12-02
FR2392958B1 (en)	1980-10-24
DK237978A (en)	1979-01-19
IT7849637A0 (en)	1978-05-31
NL190485B (en)	1993-10-18
YU129178A (en)	1983-01-21
IE46983B1 (en)	1983-11-16
JPS641474B2 (en)	1989-01-11
AU518479B2 (en)	1981-10-01
AT360509B (en)	1981-01-12
IE781078L (en)	1978-12-01

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