PT1150960E - Formas cristalinas polimorficas do celecoxib - Google Patents
Formas cristalinas polimorficas do celecoxibInfo
- Publication number
- PT1150960E PT1150960E PT00983865T PT00983865T PT1150960E PT 1150960 E PT1150960 E PT 1150960E PT 00983865 T PT00983865 T PT 00983865T PT 00983865 T PT00983865 T PT 00983865T PT 1150960 E PT1150960 E PT 1150960E
- Authority
- PT
- Portugal
- Prior art keywords
- polymoric
- celecoxib
- crystalline forms
- crystalline
- forms
- Prior art date
Links
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US16985699P | 1999-12-08 | 1999-12-08 |
Publications (1)
Publication Number | Publication Date |
---|---|
PT1150960E true PT1150960E (pt) | 2005-06-30 |
Family
ID=22617480
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT00983865T PT1150960E (pt) | 1999-12-08 | 2000-12-01 | Formas cristalinas polimorficas do celecoxib |
PT00982255T PT1150959E (pt) | 1999-12-08 | 2000-12-06 | Forma do celecoxib no estado sólido com biodisponibilidade acrescida |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT00982255T PT1150959E (pt) | 1999-12-08 | 2000-12-06 | Forma do celecoxib no estado sólido com biodisponibilidade acrescida |
Country Status (21)
Country | Link |
---|---|
KR (1) | KR100717570B1 (pt) |
CN (1) | CN1216869C (pt) |
AR (2) | AR027897A1 (pt) |
AU (1) | AU2041201A (pt) |
BG (1) | BG65239B1 (pt) |
CO (1) | CO5251445A1 (pt) |
CZ (1) | CZ20012875A3 (pt) |
EA (1) | EA200401397A1 (pt) |
EC (1) | ECSP003807A (pt) |
ES (1) | ES2236011T3 (pt) |
HU (1) | HUP0200580A3 (pt) |
MY (2) | MY128971A (pt) |
NZ (1) | NZ529933A (pt) |
OA (1) | OA11831A (pt) |
PE (1) | PE20010911A1 (pt) |
PT (2) | PT1150960E (pt) |
SV (1) | SV2002000235A (pt) |
TW (1) | TWI276435B (pt) |
WO (1) | WO2001041536A2 (pt) |
YU (1) | YU57801A (pt) |
ZA (2) | ZA200107146B (pt) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2002007721A2 (en) * | 2000-07-20 | 2002-01-31 | Lauras As | Use of cox-2 inhibitors for preventing immunodeficiency |
DE60233874D1 (de) | 2001-06-22 | 2009-11-12 | Pfizer Prod Inc | Pharmazeutische zusammensetzungen enthaltend dispersionen aus arzneistoffen und neutralen polymeren |
WO2004061433A1 (en) * | 2002-12-30 | 2004-07-22 | Transform Pharmaceuticals, Inc. | Pharmaceutical compositions with improved dissolution |
US7927613B2 (en) | 2002-02-15 | 2011-04-19 | University Of South Florida | Pharmaceutical co-crystal compositions |
WO2004026235A2 (en) * | 2002-09-20 | 2004-04-01 | Transform Pharmaceuticals, Inc. | Pharmaceutical compositions with improved dissolution |
US7790905B2 (en) | 2002-02-15 | 2010-09-07 | Mcneil-Ppc, Inc. | Pharmaceutical propylene glycol solvate compositions |
US7446107B2 (en) | 2002-02-15 | 2008-11-04 | Transform Pharmaceuticals, Inc. | Crystalline forms of conazoles and methods of making and using the same |
JP4906233B2 (ja) | 2002-03-01 | 2012-03-28 | ユニバーシティー オブ サウス フロリダ | 少なくとも1種の有効薬剤成分を含有する多構成要素固相 |
EP1505987A2 (en) * | 2002-05-13 | 2005-02-16 | Pharmacia Corporation | Stable amorphous celecoxib composite and process therefor |
AU2003243354A1 (en) | 2002-05-31 | 2003-12-19 | Transform Pharmaceuticals, Inc. | Novel conazole crystalline forms and related processes, pharmaceutical compositions and methods |
MXPA05000232A (es) * | 2002-06-21 | 2005-06-17 | Transform Pharmaceuticals Inc | Composiciones farmaceuticas con disolucion mejorada. |
US8183290B2 (en) | 2002-12-30 | 2012-05-22 | Mcneil-Ppc, Inc. | Pharmaceutically acceptable propylene glycol solvate of naproxen |
JP5021934B2 (ja) * | 2002-12-30 | 2012-09-12 | トランスフォーム・ファーマシューティカルズ・インコーポレイテッド | 改善された溶解性を有する医薬組成物 |
JP5438898B2 (ja) * | 2004-06-29 | 2014-03-12 | タケダ ファーマ アクティーゼルスカブ | 水不溶性薬剤の速放性医薬組成物の製造と、本発明の方法で得られた医薬組成物 |
GB0423103D0 (en) * | 2004-10-19 | 2004-11-17 | Boots Healthcare Int Ltd | Therapeutic agents |
CA2600822A1 (en) * | 2005-03-14 | 2006-09-21 | Nycomed Gmbh | Method for preventing cardiovascular diseases |
CN103462920A (zh) * | 2012-06-06 | 2013-12-25 | 南京亿华药业有限公司 | 一种口服环加氧酶-2抑制剂塞来昔布的组合物 |
CN103524416B (zh) * | 2013-10-29 | 2016-08-17 | 湖北华世通生物医药科技有限公司 | 一种塞来昔布新晶型a及其制备方法 |
CN103539739B (zh) * | 2013-10-30 | 2016-02-10 | 中美华世通生物医药科技(武汉)有限公司 | 一种塞来昔布新晶型b及其制备方法 |
CN103508958A (zh) * | 2013-10-30 | 2014-01-15 | 中美华世通生物医药科技(武汉)有限公司 | 一种塞来昔布新晶型c及其制备方法 |
KR101476096B1 (ko) * | 2014-03-28 | 2014-12-24 | 대원제약주식회사 | 용해도가 향상된 쎄레콕시브의 약제학적 조성물 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5474995A (en) * | 1993-06-24 | 1995-12-12 | Merck Frosst Canada, Inc. | Phenyl heterocycles as cox-2 inhibitors |
RO118291B1 (ro) * | 1993-11-30 | 2003-04-30 | Searle & Co | Derivati de pirazol 1,3,4,5 - tetrasubstituiti si compozitie farmaceutica care ii contine |
US5633272A (en) * | 1995-02-13 | 1997-05-27 | Talley; John J. | Substituted isoxazoles for the treatment of inflammation |
PT809636E (pt) * | 1995-02-13 | 2002-12-31 | Searle & Co | Isoxazoles substituidos utilizaveis para o tratamento de inflamacoes |
US5756529A (en) * | 1995-09-29 | 1998-05-26 | G.D. Searle & Co. | Substituted pyrazolyl benzenesulfonamides for use in veterinary therapies |
US5981576A (en) * | 1995-10-13 | 1999-11-09 | Merck Frosst Canada, Inc. | (Methylsulfonyl)phenyl-2-(5H)-furanones as COX-2 inhibitors |
EP0863134A1 (en) * | 1997-03-07 | 1998-09-09 | Merck Frosst Canada Inc. | 2-(3,5-difluorophenyl)-3-(4-(methyl-sulfonyl)phenyl)-2-cyclopenten-1-one useful as an inhibitor of cyclooxygenase-2 |
CA2328992A1 (en) * | 1998-04-27 | 1999-11-04 | Northwest Hospital | Nr-cam gene, nucleic acids and nucleic acid products for therapeutic and diagnostic uses for tumors |
-
2000
- 2000-12-01 CZ CZ20012875A patent/CZ20012875A3/cs unknown
- 2000-12-01 NZ NZ529933A patent/NZ529933A/en unknown
- 2000-12-01 PT PT00983865T patent/PT1150960E/pt unknown
- 2000-12-01 HU HU0200580A patent/HUP0200580A3/hu unknown
- 2000-12-01 YU YU57801A patent/YU57801A/sh unknown
- 2000-12-01 CN CN008060835A patent/CN1216869C/zh not_active Expired - Fee Related
- 2000-12-01 OA OA1200100210A patent/OA11831A/en unknown
- 2000-12-01 ES ES00983865T patent/ES2236011T3/es not_active Expired - Lifetime
- 2000-12-04 WO PCT/US2000/030180 patent/WO2001041536A2/en not_active Application Discontinuation
- 2000-12-04 AU AU20412/01A patent/AU2041201A/en not_active Withdrawn
- 2000-12-04 EC EC2000003807A patent/ECSP003807A/es unknown
- 2000-12-05 AR ARP000106473A patent/AR027897A1/es unknown
- 2000-12-06 MY MYPI20005730A patent/MY128971A/en unknown
- 2000-12-06 KR KR1020017010017A patent/KR100717570B1/ko not_active IP Right Cessation
- 2000-12-06 PE PE2000001299A patent/PE20010911A1/es not_active Application Discontinuation
- 2000-12-06 AR ARP000106475A patent/AR030039A1/es unknown
- 2000-12-06 EA EA200401397A patent/EA200401397A1/ru unknown
- 2000-12-06 MY MYPI20005733A patent/MY128366A/en unknown
- 2000-12-06 PT PT00982255T patent/PT1150959E/pt unknown
- 2000-12-08 SV SV2000000235A patent/SV2002000235A/es not_active Application Discontinuation
- 2000-12-11 CO CO00094077A patent/CO5251445A1/es not_active Application Discontinuation
-
2001
- 2001-05-18 TW TW089125991A patent/TWI276435B/zh not_active IP Right Cessation
- 2001-08-09 BG BG105808A patent/BG65239B1/bg unknown
- 2001-08-29 ZA ZA200107146A patent/ZA200107146B/xx unknown
- 2001-08-29 ZA ZA200107149A patent/ZA200107149B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
PT1150959E (pt) | 2008-04-21 |
ZA200107149B (en) | 2003-02-28 |
AR027897A1 (es) | 2003-04-16 |
ZA200107146B (en) | 2002-08-29 |
CN1411447A (zh) | 2003-04-16 |
AR030039A1 (es) | 2003-08-13 |
WO2001041536A2 (en) | 2001-06-14 |
KR100717570B1 (ko) | 2007-05-15 |
OA11831A (en) | 2005-08-23 |
ECSP003807A (es) | 2005-07-06 |
KR20020002386A (ko) | 2002-01-09 |
YU57801A (sh) | 2005-07-19 |
AU2041201A (en) | 2001-06-18 |
MY128971A (en) | 2007-03-30 |
SV2002000235A (es) | 2002-06-13 |
TWI276435B (en) | 2007-03-21 |
EA200401397A1 (ru) | 2005-08-25 |
PE20010911A1 (es) | 2001-09-10 |
HUP0200580A3 (en) | 2002-12-28 |
CZ20012875A3 (cs) | 2002-02-13 |
CO5251445A1 (es) | 2003-02-28 |
MY128366A (en) | 2007-01-31 |
HUP0200580A2 (hu) | 2002-11-28 |
BG105808A (en) | 2002-09-30 |
BG65239B1 (bg) | 2007-09-28 |
CN1216869C (zh) | 2005-08-31 |
NZ529933A (en) | 2005-06-24 |
ES2236011T3 (es) | 2005-07-16 |
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