LTIP915A - Catehol derivatives,methods for their preparation and pharmaceutical compositions containing them - Google Patents
Catehol derivatives,methods for their preparation and pharmaceutical compositions containing themInfo
- Publication number
- LTIP915A LTIP915A LTIP915A LTIP915A LTIP915A LT IP915 A LTIP915 A LT IP915A LT IP915 A LTIP915 A LT IP915A LT IP915 A LTIP915 A LT IP915A LT IP915 A LTIP915 A LT IP915A
- Authority
- LT
- Lithuania
- Prior art keywords
- catehol
- derivatives
- preparation
- methods
- pharmaceutical compositions
- Prior art date
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- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C07C205/21—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups having nitro groups and hydroxy groups bound to carbon atoms of six-membered aromatic rings having nitro groups and hydroxy groups bound to carbon atoms of the same non-condensed six-membered aromatic ring
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- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
- C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
- C07D319/24—[b,e]-condensed with two six-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FI864875A FI864875A0 (en) | 1986-11-28 | 1986-11-28 | NYA FARMAKOLOGISKT AKTIVA FOERENINGAR, DESSA INNEHAOLLANDE KOMPOSITIONER SAMT FOERFARANDE OCH MELLANPRODUKTER FOER ANVAENDNING VID FRAMSTAELLNING AV DESSA. |
Publications (2)
Publication Number | Publication Date |
---|---|
LTIP915A true LTIP915A (en) | 1995-03-27 |
LT3770B LT3770B (en) | 1996-03-25 |
Family
ID=8523579
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
LTIP915A LT3770B (en) | 1986-11-28 | 1993-08-31 | Catehol derivatives,methods for their preparation and pharmaceutical compositions containing them |
Country Status (12)
Country | Link |
---|---|
US (1) | US5112861A (en) |
KR (1) | KR960004771B1 (en) |
DD (1) | DD281375A5 (en) |
FI (2) | FI864875A0 (en) |
GB (1) | GB8712437D0 (en) |
HR (1) | HRP921250B1 (en) |
LT (1) | LT3770B (en) |
MX (1) | MX9524A (en) |
NO (1) | NO1999010I1 (en) |
PL (1) | PL154006B1 (en) |
SU (1) | SU1729291A3 (en) |
ZA (1) | ZA878953B (en) |
Families Citing this family (31)
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IL91382A (en) * | 1988-09-01 | 1995-06-29 | Orion Yhtymae Oy | Alkenyl or arylmethylene-substituted beta-diketones their preparation and pharmaceutical compositions containing them |
GB9113431D0 (en) * | 1991-06-20 | 1991-08-07 | Orion Yhytma Oy | Method for the preparation of 3,4-dihydroxy-5-nitrobenzaldehyde |
GB9626472D0 (en) | 1996-12-20 | 1997-02-05 | Aperia Anita C | New use of comt inhibitors |
US6506378B1 (en) | 1998-12-16 | 2003-01-14 | Arch Development Corporation | Vesicular monoamine transporter gene therapy in Parkinson's disease |
FI20000635A0 (en) * | 2000-03-17 | 2000-03-17 | Orion Yhtymae Oyj | Use of COMT inhibitors as an analgesic |
US7094427B2 (en) * | 2002-05-29 | 2006-08-22 | Impax Laboratories, Inc. | Combination immediate release controlled release levodopa/carbidopa dosage forms |
US20060013875A1 (en) * | 2002-05-29 | 2006-01-19 | Impax Laboratories, Inc. | Combination immediate release controlled release levodopa/carbidopa dosage forms |
JP2008515956A (en) * | 2004-10-12 | 2008-05-15 | ノボ ノルディスク アクティーゼルスカブ | 11.beta.-hydroxysteroid dehydrogenase type 1 active spiro compound |
US20070148238A1 (en) * | 2005-06-23 | 2007-06-28 | Spherics, Inc. | Dosage forms for movement disorder treatment |
EP1948190A2 (en) * | 2005-11-01 | 2008-07-30 | Transtech Pharma | Pharmaceutical use of substituted amides |
EP1945207A2 (en) * | 2005-11-01 | 2008-07-23 | Transtech Pharma, Inc. | Pharmaceutical use of substituted amides |
US20100168083A1 (en) * | 2006-03-21 | 2010-07-01 | Soren Ebdrup | Adamantane derivatives for the treatment of the metabolic syndrome |
KR20090014347A (en) | 2006-04-07 | 2009-02-10 | 하이 포인트 파마슈티칼스, 엘엘씨 | 11beta-HYDROXYSTEROID DEHYDROGENASE TYPE 1 ACTIVE COMPOUNDS |
JP2009539937A (en) * | 2006-06-16 | 2009-11-19 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | Pharmaceutical use of substituted piperidine carboxamides |
US20080131492A1 (en) * | 2006-06-23 | 2008-06-05 | Spherics, Inc. | Dosage forms for movement disorder treatment |
EP2044073A1 (en) * | 2006-07-13 | 2009-04-08 | High Point Pharmaceuticals, LLC | 11beta-hydroxysteroid dehydrogenase type 1 active compounds |
EP1878721A1 (en) * | 2006-07-13 | 2008-01-16 | Novo Nordisk A/S | 4-Piperidylbenzamides as 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors |
EP2063867A2 (en) * | 2006-12-22 | 2009-06-03 | Combinatorx, Incorporated | Pharmaceutical compositions for treatment of parkinson's disease and related disorders |
US8334305B2 (en) * | 2007-02-23 | 2012-12-18 | High Point Pharmaceuticals, Llc | N-adamantyl benzamides as inhibitors of 11-β-hydroxysteroid dehydrogenase |
US20110003856A1 (en) * | 2007-02-23 | 2011-01-06 | Soren Ebdrup | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
WO2008101885A1 (en) * | 2007-02-23 | 2008-08-28 | High Point Pharmaceuticals, Llc | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
AU2008219326B2 (en) | 2007-02-23 | 2012-12-13 | Vtv Therapeutics Llc | N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase |
MX2009009623A (en) * | 2007-03-09 | 2009-09-21 | High Point Pharmaceuticals Llc | Indole- and benzimidazole amides as hydroxysteroid dehydrogenase inhibitors. |
WO2008119017A1 (en) * | 2007-03-28 | 2008-10-02 | High Point Pharmaceuticals, Llc | 11beta-hsd1 active compounds |
CN101677562A (en) * | 2007-04-11 | 2010-03-24 | 高点制药有限责任公司 | Novel compounds |
CA2685036A1 (en) * | 2007-04-24 | 2008-11-06 | High Point Pharmaceuticals, Llc | Pharmaceutical use of substituted amides |
WO2009105140A2 (en) | 2007-12-11 | 2009-08-27 | Viamet Pharmaceuticals, Inc. | Metalloenzyme inhibitors using metal binding moieties in combination with targeting moieties |
AU2009316802B2 (en) * | 2008-11-21 | 2015-02-26 | Vtv Therapeutics Llc | Adamantyl benzamide compounds |
CA2926082C (en) | 2013-10-07 | 2022-06-14 | Impax Laboratories, Inc. | Muco-adhesive, controlled release formulations of levodopa and/or esters of levodopa and uses thereof |
EP3503883B1 (en) * | 2016-08-24 | 2022-05-04 | National Institute Of Biological Sciences, Beijing | Entacapone-related compounds to treat macular degeneration |
CN110225751A (en) * | 2016-08-24 | 2019-09-10 | 北京生命科学研究所 | For treating the compound relevant to Entacapone of damage |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB902586A (en) * | 1960-01-01 | 1962-08-01 | Shell Res Ltd | Herbicidal compositions and novel compounds for use therein |
GB1188364A (en) * | 1967-05-02 | 1970-04-15 | May & Baker Ltd | Quinoline Derivatives |
BE759266A (en) * | 1969-11-24 | 1971-05-24 | Hoffmann La Roche | PROCESS FOR THE PREPARATION OF INDOLE DERIVATIVES |
US3886285A (en) * | 1970-12-07 | 1975-05-27 | Reckitt & Colmann Prod Ltd | Pharmaceutical compositions containing substituted phenyl sulphoxides and sulphones and method of using same |
IE35838B1 (en) * | 1970-12-07 | 1976-06-09 | Reckitt & Colmann Prod Ltd | Pharmaceutical compositions |
CA1190223A (en) * | 1977-11-01 | 1985-07-09 | Anthony C. Richardson | Substrates for enzymes |
JPS5581832A (en) * | 1978-12-13 | 1980-06-20 | Sumitomo Chem Co Ltd | Preparation of p-hydroxybenzaldehyde derivatives |
FR2486523A1 (en) * | 1980-07-11 | 1982-01-15 | Rhone Poulenc Ind | PROCESS FOR THE PREPARATION OF POLYPHENOLS WHICH MAY INCLUDE ALDEHYDE GROUP |
JPS5890534A (en) * | 1981-11-25 | 1983-05-30 | Ono Pharmaceut Co Ltd | 2-aminophenol derivative, its production, and remedy containing the same as an active ingredient |
US4618627A (en) * | 1983-05-13 | 1986-10-21 | Yamanouchi Pharmaceutical Co., Ltd. | Catechol derivatives and pharmaceutical compositions thereof for inhibiting anaphylaxis (SRS-A) |
FR2557097B1 (en) * | 1983-12-22 | 1986-06-13 | Rhone Poulenc Spec Chim | PROCESS FOR THE PREPARATION OF HYDROXY AND / OR ALKOXY SUBSTITUTED BROMOBENZALDEHYDES |
FR2557098B1 (en) * | 1983-12-22 | 1986-06-13 | Rhone Poulenc Spec Chim | PROCESS FOR THE PREPARATION OF HYDROXY AND / OR ALKOXY BROMOBENZALDEHYDES SUBSTITUTED |
EP0155335A1 (en) * | 1984-03-21 | 1985-09-25 | LUDWIG HEUMANN & CO GMBH | Process for the preparation of 3,5-dimethoxy-4-alkoxy-benzaldehydes |
DK175069B1 (en) * | 1986-03-11 | 2004-05-24 | Hoffmann La Roche | Pyrocatechol derivatives |
GR871701B (en) * | 1986-11-07 | 1988-03-04 | Oreal | Method for preparing 5,6 - dihydrixyindol, and its 3 - alkylated derivative and intermediates |
US6712137B2 (en) | 2000-04-24 | 2004-03-30 | Shell Oil Company | In situ thermal processing of a coal formation to pyrolyze a selected percentage of hydrocarbon material |
-
1986
- 1986-11-28 FI FI864875A patent/FI864875A0/en not_active Application Discontinuation
-
1987
- 1987-05-27 GB GB878712437A patent/GB8712437D0/en active Pending
- 1987-11-27 KR KR87013396A patent/KR960004771B1/en active IP Right Review Request
- 1987-11-27 MX MX952487A patent/MX9524A/en unknown
- 1987-11-27 ZA ZA878953A patent/ZA878953B/en unknown
- 1987-11-27 FI FI875229A patent/FI93350C/en not_active IP Right Cessation
- 1987-11-27 PL PL1987283185A patent/PL154006B1/en unknown
- 1987-11-30 DD DD87309670A patent/DD281375A5/en not_active IP Right Cessation
-
1989
- 1989-01-23 SU SU894613317A patent/SU1729291A3/en active
-
1990
- 1990-09-25 US US07/587,791 patent/US5112861A/en not_active Expired - Lifetime
-
1992
- 1992-11-12 HR HR921250A patent/HRP921250B1/en not_active IP Right Cessation
-
1993
- 1993-08-31 LT LTIP915A patent/LT3770B/en not_active IP Right Cessation
-
1999
- 1999-06-10 NO NO1999010C patent/NO1999010I1/en unknown
Also Published As
Publication number | Publication date |
---|---|
MX9524A (en) | 1993-12-01 |
GB8712437D0 (en) | 1987-07-01 |
FI93350C (en) | 1995-03-27 |
HRP921250A2 (en) | 1998-06-30 |
HRP921250B1 (en) | 2000-06-30 |
KR960004771B1 (en) | 1996-04-13 |
KR880006170A (en) | 1988-07-21 |
DD281375A5 (en) | 1990-08-08 |
NO1999010I1 (en) | 1999-06-10 |
FI875229A (en) | 1988-05-29 |
FI93350B (en) | 1994-12-15 |
ZA878953B (en) | 1988-05-24 |
PL154006B1 (en) | 1991-06-28 |
SU1729291A3 (en) | 1992-04-23 |
FI875229A0 (en) | 1987-11-27 |
US5112861A (en) | 1992-05-12 |
FI864875A0 (en) | 1986-11-28 |
LT3770B (en) | 1996-03-25 |
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Legal Events
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SPCF | Filing an spc |
Free format text: PRODUCT NAME: N,N-DIETIL-2-CIANO-3-(3,4-DIHIDROKSI-5-NITROFENIL)AKRILAMIDAS (ENTACAPONE); REGISTRATION NO/DATE: EU/1/03/260/001, EU/1/03/260/002, EU/1/03/260/003, EU/1/03/260/004, EU/1/03/260/005, EU/1/03/260/006 20031017 Spc suppl protection certif: PA2004010 Filing date: 20041025 Expiry date: 20130831 |
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SPCR | Rejection of an spc |
Free format text: PRODUCT NAME: N,N-DIETIL-2-CIANO-3-(3,4-DIHIDROKSI-5-NITROFENIL)AKRILAMIDAS (ENTACAPONE); REGISTRATION NO/DATE: EU/1/03/260/001, EU/1/03/260/002, EU/1/03/260/003, EU/1/03/260/004, EU/1/03/260/005, EU/1/03/260/006 20031017 Spc suppl protection certif: PA2004010 Filing date: 20041025 Expiry date: 20130831 Effective date: 20050214 |
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MK9A | Expiry of a patent |
Effective date: 20130831 |