KR20010014183A - 술폰아미드 화합물 및 그의 의약 용도 - Google Patents
술폰아미드 화합물 및 그의 의약 용도Info
- Publication number
- KR20010014183A KR20010014183A KR19997012258A KR19997012258A KR20010014183A KR 20010014183 A KR20010014183 A KR 20010014183A KR 19997012258 A KR19997012258 A KR 19997012258A KR 19997012258 A KR19997012258 A KR 19997012258A KR 20010014183 A KR20010014183 A KR 20010014183A
- Authority
- KR
- South Korea
- Prior art keywords
- optionally substituted
- sulfonamide compounds
- alkylene
- medicinal use
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
- C07D241/50—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to ring nitrogen atoms
- C07D241/52—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
- C07D239/96—Two oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/16—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems
- C07D249/18—Benzotriazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP20829597 | 1997-06-27 | ||
| JP11471898 | 1998-04-24 | ||
| PCT/JP1998/002877 WO1999000372A1 (en) | 1997-06-27 | 1998-06-24 | Sulfonamide compounds and medicinal use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20010014183A true KR20010014183A (ko) | 2001-02-26 |
Family
ID=26453401
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR19997012258A KR20010014183A (ko) | 1997-06-27 | 1998-06-24 | 술폰아미드 화합물 및 그의 의약 용도 |
Country Status (12)
| Country | Link |
|---|---|
| US (3) | US6348474B1 (ko) |
| EP (1) | EP0995742A4 (ko) |
| KR (1) | KR20010014183A (ko) |
| CN (1) | CN1268942A (ko) |
| AU (1) | AU745081B2 (ko) |
| BR (1) | BR9810456A (ko) |
| CA (1) | CA2295239A1 (ko) |
| IL (1) | IL133575A0 (ko) |
| RU (1) | RU2199532C2 (ko) |
| TW (1) | TW426666B (ko) |
| WO (1) | WO1999000372A1 (ko) |
| ZA (1) | ZA985618B (ko) |
Families Citing this family (83)
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|---|---|---|---|---|
| KR20010014183A (ko) * | 1997-06-27 | 2001-02-26 | Fujisawa Pharmaceutical Co | 술폰아미드 화합물 및 그의 의약 용도 |
| ATE413386T1 (de) * | 1998-01-29 | 2008-11-15 | Amgen Inc | Ppar-gamma modulatoren |
| CA2327397A1 (en) * | 1998-04-06 | 1999-10-14 | Fujisawa Pharmaceutical Co., Ltd. | Indole derivatives |
| PE20000942A1 (es) * | 1998-07-31 | 2000-09-28 | Lilly Co Eli | Derivados de amida, carbamato y urea |
| EP1136492A4 (en) * | 1998-12-04 | 2002-03-27 | Fujisawa Pharmaceutical Co | SULFAMIDE COMPOUNDS AND USES THEREOF AS MEDICAMENTS |
| US6869950B1 (en) | 1998-12-24 | 2005-03-22 | Fujisawa Pharmaceutical Co., Ltd. | Benzimidazole derivatives |
| IL143802A0 (en) | 1998-12-24 | 2002-04-21 | Fujisawa Pharmaceutical Co | Imidazole derivatives and pharmaceutical compositions containing the same |
| GB9904103D0 (en) * | 1999-02-24 | 1999-04-14 | Zeneca Ltd | Quinoline derivatives |
| US7041691B1 (en) | 1999-06-30 | 2006-05-09 | Amgen Inc. | Compounds for the modulation of PPARγ activity |
| US6653332B2 (en) | 2000-05-03 | 2003-11-25 | Tularik Inc. | Combination therapeutic compositions and method of use |
| US20030171399A1 (en) * | 2000-06-28 | 2003-09-11 | Tularik Inc. | Quinolinyl and benzothiazolyl modulators |
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| SE0102299D0 (sv) | 2001-06-26 | 2001-06-26 | Astrazeneca Ab | Compounds |
| SE0102764D0 (sv) * | 2001-08-17 | 2001-08-17 | Astrazeneca Ab | Compounds |
| GB0226930D0 (en) | 2002-11-19 | 2002-12-24 | Astrazeneca Ab | Chemical compounds |
| WO2005021537A1 (en) | 2003-08-21 | 2005-03-10 | Osi Pharmaceuticals, Inc. | N-substituted pyrazolyl-amidyl-benzimidazolyl c-kit inhibitors |
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| RU2009121756A (ru) * | 2006-12-21 | 2011-01-27 | Астразенека Аб (Se) | Новое кристаллическое соединение, полезное в качестве активатора глюкокиназы (glk) |
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| DK2247580T3 (en) | 2008-03-05 | 2015-10-05 | Merck Patent Gmbh | Quinoxalinone derivatives AS INSULINSEKRETIONSSTIMULATORER, METHODS FOR OBTAINING THEREOF AND USE THEREOF FOR THE TREATMENT OF DIABETES |
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| EP2593427B1 (en) | 2010-07-12 | 2014-12-24 | Pfizer Limited | Sulfonamide derivatives as nav1.7 inhibitors for the treatment of pain |
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| WO2012105594A1 (ja) | 2011-02-01 | 2012-08-09 | 協和発酵キリン株式会社 | 縮環複素環誘導体 |
| MY159058A (en) * | 2011-02-25 | 2016-12-15 | Merck Sharp & Dohme | Novel cyclic azabenzimidazole derivatives useful as anti-diabetic agent |
| EP3495366A1 (en) * | 2011-07-15 | 2019-06-12 | Shionogi & Co., Ltd | Azabenzimidazole derivative having ampk-activating activity |
| JP2013028559A (ja) * | 2011-07-28 | 2013-02-07 | Nippon Light Metal Co Ltd | ３−クロロ−４−メチル安息香酸イソプロピル及びその製造方法 |
| JP5965484B2 (ja) | 2012-07-27 | 2016-08-03 | 佐藤製薬株式会社 | ジフルオロメチレン化合物 |
| TW201410677A (zh) | 2012-07-31 | 2014-03-16 | Kyowa Hakko Kirin Co Ltd | 縮環雜環化合物 |
| LT2925757T (lt) | 2012-11-19 | 2017-12-27 | Novartis Ag | Junginiai ir kompozicijos, skirti parazitinių ligų gydymui |
| US8871754B2 (en) | 2012-11-19 | 2014-10-28 | Irm Llc | Compounds and compositions for the treatment of parasitic diseases |
| TWI731317B (zh) * | 2013-12-10 | 2021-06-21 | 美商健臻公司 | 原肌球蛋白相關之激酶（ｔｒｋ）抑制劑 |
| KR102561692B1 (ko) | 2014-12-18 | 2023-07-28 | 젠자임 코포레이션 | 트로포미오신-관련 키나제(trk) 억제제의 약제학적 제형 |
| PE20180573A1 (es) * | 2015-07-20 | 2018-04-04 | Genzyme Corp | Inhibidores del receptor del factor estimulador de colonias 1 (csf-1r) |
| TW201831471A (zh) * | 2017-02-24 | 2018-09-01 | 盧森堡商艾伯維公司 | 囊腫纖化症跨膜傳導調節蛋白的調節劑及其使用方法 |
| DE102017123282A1 (de) * | 2017-10-06 | 2019-04-11 | Henkel Ag & Co. Kgaa | Hydrolyselabile Silylenolether von Riechstoffketonen oder -aldehyden |
| JP2024500919A (ja) | 2020-12-23 | 2024-01-10 | ジェンザイム・コーポレーション | 重水素化コロニー刺激因子－１受容体（ｃｓｆ－１ｒ）阻害剤 |
| CN114732816B (zh) * | 2022-03-03 | 2023-08-15 | 南方医科大学南方医院 | 2-芳基-1,3二氢苯并咪唑衍生物在制备治疗肾癌药物中的用途 |
| CN115154466B (zh) * | 2022-06-06 | 2023-08-15 | 南方医科大学南方医院 | 2-芳基-1,3二氢苯并咪唑衍生物在制备治疗糖尿病肾病药物中的用途 |
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| IS2334B (is) | 1992-09-08 | 2008-02-15 | Vertex Pharmaceuticals Inc., (A Massachusetts Corporation) | Aspartyl próteasi hemjari af nýjum flokki súlfonamíða |
| ATE165823T1 (de) | 1993-06-22 | 1998-05-15 | Knoll Ag | Isochinolin-derivate mit therapeutischer wirkung |
| US5599811A (en) * | 1995-02-21 | 1997-02-04 | Warner-Lambert Company | Benzothiazine dioxides as endothelin antagonists |
| FR2733233B1 (fr) | 1995-04-20 | 1997-05-30 | Roussel Uclaf | Nouveaux derives de quinoleine, leur procede de preparation, les nouveaux intermediaires obtenus, leur application a titre de medicaments et les compositions pharmaceutiques les renfermant |
| AU722514B2 (en) | 1995-12-28 | 2000-08-03 | Fujisawa Pharmaceutical Co., Ltd. | Benzimidazole derivatives |
| JP2000511533A (ja) * | 1996-05-20 | 2000-09-05 | メルク エンド カンパニー インコーポレーテッド | ゴナドトロピン放出ホルモン拮抗薬 |
| WO1998008818A1 (en) * | 1996-08-26 | 1998-03-05 | Genetics Institute, Inc. | Inhibitors of phospholipase enzymes |
| FR2756284B1 (fr) | 1996-11-26 | 2000-04-28 | Adir | Nouveaux derives du benzopyrane, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| US6242474B1 (en) * | 1997-06-27 | 2001-06-05 | Fujisawa Pharmaceutical Co., Ltd. | Aromatic ring derivatives |
| KR20010014183A (ko) * | 1997-06-27 | 2001-02-26 | Fujisawa Pharmaceutical Co | 술폰아미드 화합물 및 그의 의약 용도 |
| TW453999B (en) * | 1997-06-27 | 2001-09-11 | Fujisawa Pharmaceutical Co | Benzimidazole derivatives |
| EP1136492A4 (en) * | 1998-12-04 | 2002-03-27 | Fujisawa Pharmaceutical Co | SULFAMIDE COMPOUNDS AND USES THEREOF AS MEDICAMENTS |
-
1998
- 1998-06-24 KR KR19997012258A patent/KR20010014183A/ko not_active Application Discontinuation
- 1998-06-24 RU RU2000101813/04A patent/RU2199532C2/ru not_active IP Right Cessation
- 1998-06-24 US US09/446,110 patent/US6348474B1/en not_active Expired - Fee Related
- 1998-06-24 CN CN98808571A patent/CN1268942A/zh active Pending
- 1998-06-24 BR BR9810456-0A patent/BR9810456A/pt not_active IP Right Cessation
- 1998-06-24 AU AU79345/98A patent/AU745081B2/en not_active Ceased
- 1998-06-24 WO PCT/JP1998/002877 patent/WO1999000372A1/ja not_active Application Discontinuation
- 1998-06-24 EP EP98929715A patent/EP0995742A4/en not_active Withdrawn
- 1998-06-24 CA CA002295239A patent/CA2295239A1/en not_active Abandoned
- 1998-06-24 IL IL13357598A patent/IL133575A0/xx unknown
- 1998-06-25 TW TW087110245A patent/TW426666B/zh not_active IP Right Cessation
- 1998-06-26 ZA ZA985618A patent/ZA985618B/xx unknown
-
2002
- 2002-01-17 US US10/047,093 patent/US6911469B2/en not_active Expired - Fee Related
-
2004
- 2004-03-30 US US10/811,989 patent/US20040180947A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US6348474B1 (en) | 2002-02-19 |
| US6911469B2 (en) | 2005-06-28 |
| EP0995742A4 (en) | 2004-08-25 |
| US20040180947A1 (en) | 2004-09-16 |
| US20020099212A1 (en) | 2002-07-25 |
| TW426666B (en) | 2001-03-21 |
| RU2199532C2 (ru) | 2003-02-27 |
| AU745081B2 (en) | 2002-03-14 |
| IL133575A0 (en) | 2001-04-30 |
| BR9810456A (pt) | 2001-09-25 |
| WO1999000372A1 (en) | 1999-01-07 |
| CN1268942A (zh) | 2000-10-04 |
| AU7934598A (en) | 1999-01-19 |
| ZA985618B (en) | 1999-01-19 |
| EP0995742A1 (en) | 2000-04-26 |
| CA2295239A1 (en) | 1999-01-07 |
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