Nothing Special   »   [go: up one dir, main page]

IT8067465A0 - Acidi 4 ammino 3 chinolincarbossili ci e loro esteri particolarmente utili come antisecretivi ed antiulcera - Google Patents

Acidi 4 ammino 3 chinolincarbossili ci e loro esteri particolarmente utili come antisecretivi ed antiulcera

Info

Publication number
IT8067465A0
IT8067465A0 IT8067465A IT6746580A IT8067465A0 IT 8067465 A0 IT8067465 A0 IT 8067465A0 IT 8067465 A IT8067465 A IT 8067465A IT 6746580 A IT6746580 A IT 6746580A IT 8067465 A0 IT8067465 A0 IT 8067465A0
Authority
IT
Italy
Prior art keywords
quinolincarboxy
antiulcera
antisecretives
acids
amino
Prior art date
Application number
IT8067465A
Other languages
English (en)
Other versions
IT1133079B (it
Inventor
Harry Randall Munson Jr
Reevis Stancil Alphin
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of IT8067465A0 publication Critical patent/IT8067465A0/it
Application granted granted Critical
Publication of IT1133079B publication Critical patent/IT1133079B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IT67465/80A 1979-03-26 1980-03-26 Acidi 4 ammino & chinolincarbossilici e loro esteri particolarmente utili come antisecreitivi ed antiulcera IT1133079B (it)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2398179A 1979-03-26 1979-03-26
US06/127,153 US4343804A (en) 1979-03-26 1980-03-04 4-Amino-3-quinolinecarboxylic acids and esters-antisecretory anti-ulcer compounds

Publications (2)

Publication Number Publication Date
IT8067465A0 true IT8067465A0 (it) 1980-03-26
IT1133079B IT1133079B (it) 1986-07-09

Family

ID=26697875

Family Applications (1)

Application Number Title Priority Date Filing Date
IT67465/80A IT1133079B (it) 1979-03-26 1980-03-26 Acidi 4 ammino & chinolincarbossilici e loro esteri particolarmente utili come antisecreitivi ed antiulcera

Country Status (31)

Country Link
US (1) US4343804A (it)
JP (1) JPH02117663A (it)
AR (1) AR230268A1 (it)
AT (1) AT372373B (it)
AU (1) AU528388B2 (it)
BR (1) BR8001779A (it)
CA (1) CA1147338A (it)
CH (1) CH644105A5 (it)
DE (1) DE3011490A1 (it)
DK (1) DK156056C (it)
EG (1) EG15009A (it)
ES (1) ES8103048A1 (it)
FI (1) FI77452C (it)
FR (1) FR2452485B1 (it)
GB (1) GB2047244B (it)
GR (1) GR68006B (it)
HK (1) HK67983A (it)
IE (1) IE49577B1 (it)
IL (1) IL59628A (it)
IN (1) IN151446B (it)
IT (1) IT1133079B (it)
MX (1) MX6264E (it)
NL (1) NL8001752A (it)
NO (1) NO153927C (it)
NZ (1) NZ193252A (it)
PH (1) PH16416A (it)
PL (1) PL125030B1 (it)
PT (1) PT71008B (it)
SE (1) SE435837B (it)
SG (1) SG33683G (it)
YU (1) YU41702B (it)

Families Citing this family (43)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8610981D0 (en) * 1986-05-06 1986-06-11 Ici America Inc Quinoline amides
GB8621425D0 (en) * 1986-09-05 1986-10-15 Smith Kline French Lab Compounds
GB8804445D0 (en) * 1988-02-25 1988-03-23 Smithkline Beckman Intercredit Compounds
GB8804446D0 (en) * 1988-02-25 1988-03-23 Smithkline Beckman Intercredit Compounds
GB8804448D0 (en) * 1988-02-25 1988-03-23 Smithkline Beckman Intercredit Compounds
GB8804444D0 (en) * 1988-02-25 1988-03-23 Smithkline Beckman Intercredit Compounds
GB8804443D0 (en) * 1988-02-25 1988-03-23 Smithkline Beckman Intercredit Compounds
GB8804447D0 (en) * 1988-02-25 1988-03-23 Smithkline Beckman Intercredit Compounds
US5432182A (en) * 1989-02-23 1995-07-11 Smithkline Beecham Intercredit B.V. Compounds substituted quinoline derivatives
CA2011086A1 (en) * 1989-03-17 1990-09-17 Karl-Heinz Geiss 2-alkyl-4-arylmethylaminoquinolines, the use thereof and drugs prepared therefrom
DE3917233A1 (de) * 1989-05-26 1990-11-29 Basf Ag 8-substituierte 4-(heterocyclylmethylamino)-chinoline, ihre verwendung und daraus hergestellte arzneimittel
GB8918265D0 (en) * 1989-08-10 1989-09-20 Smithkline Beckman Intercredit Compounds
US5362743A (en) * 1993-03-09 1994-11-08 Pfizer Inc. Aminoquinoline derivatives
IS4164A (is) * 1993-06-11 1994-12-12 Ab Astra Efnasambönd sem hindra flæði magasýru
US5556863A (en) * 1993-06-11 1996-09-17 Astra Aktiebolag Compound for gastric acid secretion inhibition
HU222178B1 (hu) * 1993-08-10 2003-04-28 James Black Foundation Ltd. Gasztrin és CCK-receptor ligandumok, eljárás előállításukra és ezeket tartalmazó gyógyászati készítmények
US5650415A (en) * 1995-06-07 1997-07-22 Sugen, Inc. Quinoline compounds
KR0169813B1 (ko) * 1995-07-12 1999-01-15 김종인 4-아미노-3-아실나프티리딘 유도체
US5760041A (en) * 1996-02-05 1998-06-02 American Cyanamid Company 4-aminoquinazoline EGFR Inhibitors
US6875769B2 (en) * 1996-05-23 2005-04-05 Pfizer Inc. Substituted6,6-hetero-bicyclicderivatives
US5929080A (en) * 1997-05-06 1999-07-27 American Cyanamid Company Method of treating polycystic kidney disease
US6251912B1 (en) 1997-08-01 2001-06-26 American Cyanamid Company Substituted quinazoline derivatives
US6323209B1 (en) 1997-11-06 2001-11-27 American Cyanamid Company Method of treating or inhibiting colonic polyps
CA2344168C (en) 1998-09-29 2011-04-05 American Cyanamid Company Substituted 3-cyanoquinolines as protein tyrosine kinases inhibitors
CN1217936C (zh) * 1999-12-28 2005-09-07 卫材株式会社 含有磺酰胺的杂环化合物
US6521618B2 (en) * 2000-03-28 2003-02-18 Wyeth 3-cyanoquinolines, 3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors
US6576644B2 (en) * 2000-09-06 2003-06-10 Bristol-Myers Squibb Co. Quinoline inhibitors of cGMP phosphodiesterase
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
MXPA05007485A (es) 2003-01-14 2006-01-30 Arena Pharm Inc Derivados de arilo y heteroarilo 1,2,3-trisubstituidos como moduladores del metabolismo y la profilaxis y tratamiento de trastornos relacionados con ello tales como diabetes e hiperglicemia.
WO2004080967A1 (en) 2003-03-10 2004-09-23 Altana Pharma Ag Novel process for the preparation of roflumilast
WO2005007658A2 (en) * 2003-07-14 2005-01-27 Arena Pharmaceuticals, Inc. Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
WO2006097456A1 (en) * 2005-03-16 2006-09-21 Nycomed Gmbh Taste masked dosage form containing roflumilast
WO2011022216A1 (en) * 2009-08-17 2011-02-24 High Point Pharmaceuticals, Llc Substituted pyridine derivatives, pharmaceutical compositions, and methods of use to treat oxidative stress
SG10201906876PA (en) 2010-01-27 2019-09-27 Arena Pharm Inc Processes for the preparation of (r)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid and salts thereof
BR112013008100A2 (pt) 2010-09-22 2016-08-09 Arena Pharm Inc "moduladores do receptor de gpr19 e o tratamento de distúrbios relacionados a eles."
PT3242666T (pt) 2015-01-06 2024-12-09 Arena Pharm Inc Composto para utilização no tratamento de patologias relacionadas com o recetor s1p1
AU2016284162A1 (en) 2015-06-22 2018-02-01 Arena Pharmaceuticals, Inc. Crystalline L-arginine salt of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta[b]indol-3-yl)acetic acid(Compound1) for use in SIP1 receptor-associated disorders
CA3043298A1 (en) * 2016-11-11 2018-05-17 Bayer Animal Health Gmbh Anthelmintic quinoline-3-carboxamide derivatives
CA3053418A1 (en) 2017-02-16 2018-08-23 Arena Pharmaceuticals, Inc. Compounds and methods for treatment of primary biliary cholangitis
WO2019084271A1 (en) * 2017-10-25 2019-05-02 Children's Medical Center Corporation PAPD5 INHIBITORS AND METHODS OF USE
SG11202010024UA (en) 2018-05-09 2020-11-27 Bayer Animal Health Gmbh New quinoline derivatives
CN112601516A (zh) 2018-06-06 2021-04-02 艾尼纳制药公司 治疗与s1p1受体相关的病况的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3470186A (en) * 1967-06-02 1969-09-30 American Cyanamid Co Substituted 4-anilino-3-quinolinecarboxylic acids and esters
JPS4838712A (it) * 1971-09-18 1973-06-07

Also Published As

Publication number Publication date
AR230268A1 (es) 1984-03-01
GB2047244A (en) 1980-11-26
YU41702B (en) 1987-12-31
CH644105A5 (fr) 1984-07-13
FR2452485A1 (fr) 1980-10-24
FR2452485B1 (fr) 1986-09-12
SG33683G (en) 1985-03-29
FI77452B (fi) 1988-11-30
HK67983A (en) 1983-12-23
DK128380A (da) 1980-09-27
AU528388B2 (en) 1983-04-28
IE49577B1 (en) 1985-10-30
PL222993A1 (it) 1981-01-30
SE8002292L (sv) 1980-09-27
DE3011490A1 (de) 1981-03-12
NO153927C (no) 1986-06-18
PT71008A (en) 1980-04-01
PT71008B (en) 1981-06-25
FI800910A (fi) 1980-09-27
SE435837B (sv) 1984-10-22
PL125030B1 (en) 1983-03-31
GR68006B (it) 1981-10-26
IL59628A (en) 1983-06-15
IT1133079B (it) 1986-07-09
PH16416A (en) 1983-09-29
GB2047244B (en) 1983-02-23
BR8001779A (pt) 1980-11-18
ATA156480A (de) 1983-02-15
FI77452C (fi) 1989-03-10
AT372373B (de) 1983-09-26
YU84480A (en) 1983-10-31
MX6264E (es) 1985-02-19
NL8001752A (nl) 1980-09-30
NO153927B (no) 1986-03-10
DK156056B (da) 1989-06-19
ES489887A0 (es) 1981-02-16
EG15009A (en) 1985-03-31
NO800858L (no) 1980-09-29
IN151446B (it) 1983-04-23
IL59628A0 (en) 1980-06-30
NZ193252A (en) 1984-04-27
DK156056C (da) 1989-11-06
DE3011490C2 (it) 1988-12-22
US4343804A (en) 1982-08-10
AU5684880A (en) 1980-10-02
IE800605L (en) 1980-09-26
JPH02117663A (ja) 1990-05-02
CA1147338A (en) 1983-05-31
ES8103048A1 (es) 1981-02-16

Similar Documents

Publication Publication Date Title
IT8067465A0 (it) Acidi 4 ammino 3 chinolincarbossili ci e loro esteri particolarmente utili come antisecretivi ed antiulcera
IT7868449A0 (it) Aminoacidi ciclici particolarmente utili per medicamenti e procedimento per la loro preparazione
IT8547651A0 (it) Procedimento per produrre acidi carbossilici sostituiti utili come agenti acilanti e loro derivati
IT1078869B (it) Procedimento per la produzione di acidi ed esteri ciclopropancarbossilici
IT1194632B (it) Acidi n-(idrossimetil)-amminoalcan-difosfonici e loro impiego come stabilizzanti
IT7948950A0 (it) Acidi lattamo-n-acetici e loro ammidi procedimento per prepararli e composizioni terapeutiche che licontengono
IT1098980B (it) Procedimento per la produzione di acidi carbossilici e/o di loro esteri
IT1146744B (it) Acidi 2 ammino 3 idrossi fenil metel fenilacetici loro esteri ed ammidi particolarmente utili come antiinfiammatori
IT1221767B (it) Acidi propenilamminotiazolilcefalosporanici 3-(sostituiti)e loro esteri
IT1065478B (it) Processo per la preparazione di acido 5 cianvalerianico e suoi esteri
BR8004778A (pt) Processo para a preparacao de esteres de acidos n-metil-o-pirazol(4)il-carbamicos,composicoes praguicidas e sua aplicacao
IT1133039B (it) Acidi alcossibenzofuran carbossilici e loro sali ed esteri utili come agenti ipolipidemici e procedimento per la loro prpparazione
IT8267152A0 (it) Acidi 2 ammino 3 alogenobenzoilmetilfenilacetici loro esteri e sali e composizioni farmaceutiche contenenti tali composti
IT1126477B (it) Processo per la preparazione di acidi aril-ed eteroarilesadienoici
IT7849635A0 (it) Di-e tri-fluorometil ammino acidi ed ammine composizioni e procedimento per la loro preparazione
IT1076780B (it) Esteri benzilici ed esteri analoghi di acidi 6,11-diidrodibenz parentesi quadra aperta b,e parentesi quadra chiusa-ossepin-acetici
IT1075420B (it) Processo per la preparazione di esteri benzilici ad azione pesticida e prodotti ottenuti
IT1100581B (it) Procedimento per la fabbricazione di esteri easici di acidi idrossicicicloesancarbossilici sostituti
IT1094565B (it) Acidi 5-solfamoilortanilici e processo per la loro preparazione
IT8348492A0 (it) Furfurilammidi di acidi fenossifenossialcanoici utili come erbicidi selettivi
IT1113428B (it) Acidi esaidro-1-mercaptoacil-1h-azepin-2-carbossilici e loro esteri
IT1186768B (it) Acilammino idrossialcanoil ammino ed immino acidi ed esteri
IT1118756B (it) Acidi paracarbonilfenossi carbossici particolarmente utili come medicamenti e procedimento per la loro preparazione
IT1135000B (it) Colorformiati di esteri alchilici di acidi c-alchil-tartronici e loro processo di preparazione
IT7941020A0 (it) Acidi 2 xantonossi 2 metilpropioni ci loro esteri e loro sali caratterizzati da attivita ipolipemizzante