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ID30393A - Senyawa tienopirimidina, pembuatan dan penggunaannya - Google Patents

Senyawa tienopirimidina, pembuatan dan penggunaannya

Info

Publication number
ID30393A
ID30393A IDW00200102298A ID20012298A ID30393A ID 30393 A ID30393 A ID 30393A ID W00200102298 A IDW00200102298 A ID W00200102298A ID 20012298 A ID20012298 A ID 20012298A ID 30393 A ID30393 A ID 30393A
Authority
ID
Indonesia
Prior art keywords
tienopirimidina
compounds
making
tienopirimidina compounds
Prior art date
Application number
IDW00200102298A
Other languages
English (en)
Inventor
Shuichi Furuya
Nobuhiro Suzuki
Nobuo Choh
Yoshi Nara
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of ID30393A publication Critical patent/ID30393A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/02Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A61P5/04Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
IDW00200102298A 1999-03-24 2000-03-23 Senyawa tienopirimidina, pembuatan dan penggunaannya ID30393A (id)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP7937199 1999-03-24
JP2000018019 2000-01-25

Publications (1)

Publication Number Publication Date
ID30393A true ID30393A (id) 2001-11-29

Family

ID=26420391

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW00200102298A ID30393A (id) 1999-03-24 2000-03-23 Senyawa tienopirimidina, pembuatan dan penggunaannya

Country Status (28)

Country Link
US (1) US6340686B1 (id)
EP (1) EP1163244B1 (id)
JP (1) JP3240293B2 (id)
KR (2) KR100533483B1 (id)
CN (1) CN1349536A (id)
AR (1) AR023152A1 (id)
AT (1) ATE261449T1 (id)
AU (1) AU764019B2 (id)
BR (1) BR0009297A (id)
CA (1) CA2368108C (id)
CZ (1) CZ294747B6 (id)
DE (1) DE60008862T2 (id)
DK (1) DK1163244T3 (id)
ES (1) ES2212992T3 (id)
HK (1) HK1042495B (id)
HU (1) HUP0200550A3 (id)
ID (1) ID30393A (id)
IL (1) IL145549A (id)
MX (1) MXPA01009566A (id)
MY (1) MY124726A (id)
NO (1) NO20014603L (id)
NZ (1) NZ514737A (id)
OA (1) OA11920A (id)
PL (1) PL351202A1 (id)
PT (1) PT1163244E (id)
SK (1) SK13552001A3 (id)
TW (1) TWI225863B (id)
WO (1) WO2000056739A1 (id)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
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US6828415B2 (en) * 1993-02-19 2004-12-07 Zentaris Gmbh Oligopeptide lyophilisate, their preparation and use
CN1173977C (zh) * 2000-02-29 2004-11-03 武田药品工业株式会社 制备噻吩并嘧啶衍生物的方法
AU2001248760A1 (en) * 2000-04-13 2001-10-30 Takeda Chemical Industries Ltd. Preventives/remedies for alzheimer's disease
AU2001264264A1 (en) * 2000-06-14 2001-12-24 Takeda Chemical Industries Ltd. Sustained release compositions
AU2001288102A1 (en) * 2000-09-22 2002-04-02 Takeda Chemical Industries Ltd. Solid preparations
WO2002043766A1 (fr) * 2000-11-29 2002-06-06 Takeda Chemical Industries, Ltd. Compositions medicinales et leur procede de preparation
WO2002047722A1 (fr) * 2000-12-15 2002-06-20 Takeda Chemical Industries, Ltd. Compositions medicinales agoniste ou antagoniste de la gonadoliberine non peptidyl, methode de production et utilisation desdites compositions
WO2002078669A1 (fr) * 2001-03-30 2002-10-10 Takeda Chemical Industries, Ltd. Solutions medicinales
JP2005504034A (ja) 2001-08-02 2005-02-10 ニューロクライン バイオサイエンシーズ, インコーポレイテッド ゴナドトロピン放出性ホルモンレセプターアンタゴニストとしてのピリジノン誘導体およびピリダジノン誘導体
US6673796B2 (en) 2001-08-02 2004-01-06 Neurocrine Biosciences, Inc. Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
AU2002324586B2 (en) 2001-08-02 2008-04-24 Neurocrine Biosciences, Inc. 1,3,5-triazine-2,4,6-triones, preparation and use as gonadotropin-releasing hormone receptor antagonists
EP1411945A1 (en) 2001-08-02 2004-04-28 Neurocrine Biosciences, Inc. Substituted pyridin-4-ones and their use as gonadotropin-releasing hormone receptor antagonists
JP2005500356A (ja) 2001-08-02 2005-01-06 ニューロクライン バイオサイエンシーズ, インコーポレイテッド ゴナドトロピン放出ホルモンレセプターアンタゴニスト
WO2003064429A1 (fr) 2002-01-30 2003-08-07 Takeda Chemical Industries, Ltd. Thienopyrimidines, procedes de fabrication et d'utilisation correspondants
WO2003086464A1 (fr) 2002-04-12 2003-10-23 Takeda Pharmaceutical Company Limited. Agents pour prevenir/traiter les bouffees de chaleur
ES2298545T3 (es) * 2002-08-21 2008-05-16 Astrazeneca Ab Compuestos de tieno-pirrol como antagonistas de la hormona liberadora de gonadotropina.
DK1591446T3 (da) 2003-01-29 2013-06-10 Takeda Pharmaceutical Thienopyrimidinforbindelser og anvendelse deraf.
GB0307777D0 (en) 2003-04-04 2003-05-07 Medical Res Council Conjugate compounds
US20060083017A1 (en) * 2004-10-18 2006-04-20 Bwt Propety, Inc. Solid-state lighting apparatus for navigational aids
NZ566038A (en) * 2005-07-22 2011-06-30 Takeda Pharmaceutical The use of thieno(2,3-d)pyrimidine-2,4-dione derivatives which are gonadotropin releasing hormone (GnRH) antagonists as premature ovulation preventive agent
EP2329823A4 (en) 2008-09-03 2013-04-03 Takeda Pharmaceutical METHOD FOR IMPROVING CAPACITY OF PREPARATION TO BE ABSORBED AND PREPARATION WHICH CAPACITY TO BE ABSORBED IS IMPROVED
BR112014021331B1 (pt) * 2012-02-28 2020-12-15 Tiumbio Co., Ltd Antagonistas do receptor do hormônio liberador de gonadotropina, composição farmacêutica compreendendo os mesmos e uso desses
CA2881132C (en) 2012-09-28 2020-11-24 Takeda Pharmaceutical Company Limited Production method of thienopyrimidine derivative
LT3263110T (lt) 2015-02-26 2023-07-10 Takeda Pharmaceutical Company Limited Tabletė, apimanti metoksikarbamido darinį ir manitolio daleles
WO2018060501A2 (en) 2016-09-30 2018-04-05 Myovant Sciences Gmbh Methods of treating uterine fibroids and endometriosis
MX2019003733A (es) 2016-09-30 2019-09-26 Myovant Sciences Gmbh Tratamiento de cancer de prostata.
KR101973074B1 (ko) * 2018-11-30 2019-04-26 주식회사 티움바이오 퓨로피리미딘 화합물의 염 및 결정형, 및 이를 포함하는 약학적 조성물
CN111943960B (zh) * 2019-07-29 2022-02-15 广东东阳光药业有限公司 取代的嘧啶二酮类化合物及其用途
CN111574534B (zh) * 2020-05-25 2021-06-04 东莞市东阳光新药研发有限公司 苯基取代的噻吩并[2,3-d]嘧啶-2,4(1H,3H)-二酮类化合物及其用途
CN111925379B (zh) * 2020-07-31 2022-02-15 广东东阳光药业有限公司 含氮杂芳基取代的嘧啶二酮类化合物及其用途
CN111909168B (zh) * 2020-07-31 2022-02-01 广东东阳光药业有限公司 含氮杂环基取代的嘧啶二酮类化合物及其用途
CN113754679B (zh) * 2020-09-09 2023-04-07 广东东阳光药业有限公司 取代的嘧啶二酮类化合物及其用途
CN112047957B (zh) * 2020-09-09 2022-02-01 广东东阳光药业有限公司 取代的嘧啶二酮类化合物及其用途
CN113563363B (zh) * 2020-12-30 2022-06-28 上海博志研新药物技术有限公司 瑞卢戈利中间体、其制备方法及瑞卢戈利的制备方法
CN115260211B (zh) * 2021-04-29 2024-02-06 长春金赛药业有限责任公司 含噻吩稠环类衍生物、药物组合物及其制备方法和应用
CN113717149A (zh) * 2021-09-29 2021-11-30 成都伊诺达博医药科技有限公司 一种瑞卢戈利关键中间体及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW449600B (en) * 1994-04-19 2001-08-11 Takeda Chemical Industries Ltd Condensed-ring thiophene derivatives, their production and use
UY23948A1 (es) * 1995-02-08 2001-10-25 Takeda Chemical Industries Ltd Derivados de anillos condensados de tiofeno su producción y uso.
US5627786A (en) * 1995-02-10 1997-05-06 Micron Quantum Devices, Inc. Parallel processing redundancy scheme for faster access times and lower die area
WO1996028405A1 (fr) * 1995-03-10 1996-09-19 Nitto Chemical Industry Co., Ltd. Procede de production de derives de 1,2-ethanediol

Also Published As

Publication number Publication date
EP1163244A1 (en) 2001-12-19
NZ514737A (en) 2003-10-31
CZ294747B6 (cs) 2005-03-16
NO20014603L (no) 2001-11-26
ES2212992T3 (es) 2004-08-16
MY124726A (en) 2006-06-30
PL351202A1 (en) 2003-03-24
DK1163244T3 (da) 2004-07-12
HUP0200550A3 (en) 2004-07-28
CN1349536A (zh) 2002-05-15
AR023152A1 (es) 2002-09-04
ATE261449T1 (de) 2004-03-15
CA2368108A1 (en) 2000-09-28
HUP0200550A2 (en) 2002-06-29
KR20010015920A (ko) 2001-02-26
HK1042495A1 (en) 2002-08-16
SK13552001A3 (sk) 2002-03-05
WO2000056739A1 (en) 2000-09-28
CZ20013419A3 (cs) 2002-02-13
TWI225863B (en) 2005-01-01
DE60008862T2 (de) 2005-01-27
BR0009297A (pt) 2001-12-18
HK1042495B (zh) 2004-10-08
IL145549A0 (en) 2002-06-30
PT1163244E (pt) 2004-07-30
AU3326200A (en) 2000-10-09
US6340686B1 (en) 2002-01-22
KR20010090430A (ko) 2001-10-18
DE60008862D1 (de) 2004-04-15
KR100370981B1 (ko) 2003-02-06
EP1163244B1 (en) 2004-03-10
OA11920A (en) 2006-04-12
NO20014603D0 (no) 2001-09-21
AU764019B2 (en) 2003-08-07
JP3240293B2 (ja) 2001-12-17
KR100533483B1 (ko) 2005-12-05
MXPA01009566A (es) 2002-05-14
JP2001278884A (ja) 2001-10-10
CA2368108C (en) 2009-12-22
IL145549A (en) 2005-11-20

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