HU9500418D0 - Process for producing 3-{2-[4-(6-fluoro-benzo[d]isoxazol-3-yl)piperidine-1-il]-ethyl}-2-methyl-6,7,8,9-tetrahydro-4h-pyrido[1,2-a]pyrimidine-4-one - Google Patents

Process for producing 3-{2-[4-(6-fluoro-benzo[d]isoxazol-3-yl)piperidine-1-il]-ethyl}-2-methyl-6,7,8,9-tetrahydro-4h-pyrido[1,2-a]pyrimidine-4-one

Info

Publication number: HU9500418D0
Authority: HU; Hungary
Prior art keywords: isoxazol; pyrido; benzo; tetrahydro; piperidine
Prior art date: 1994-02-11

Application number

HU9500418A

Other languages

Hungarian (hu)

Other versions

HU222110B1 (en

HUT70169A (en

Inventor

Olondriz Francisco Marquillas

Barjoan Pere Dalmases

Clotet Joan Huguet

Rovira Ana Bosch

Castillo Nieto Juan Carlos Del

Ges Jose Maria Caldero

Original Assignee

Vita Invest Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-02-11

Filing date

1995-02-10

Publication date

1995-03-28

1995-02-10 Application filed by Vita Invest Sa filed Critical Vita Invest Sa

1995-03-28 Publication of HU9500418D0 publication Critical patent/HU9500418D0/en

1995-09-28 Publication of HUT70169A publication Critical patent/HUT70169A/en

2003-04-28 Publication of HU222110B1 publication Critical patent/HU222110B1/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

HU9500418A 1994-02-11 1995-02-10 Process for producing 3-{2-[4-(6-fluoro-benzo[d]isoxazol-3-yl)piperidine-1-il]-ethyl}-2-methyl-6,7,8,9-tetrahydro-4h-pyrido[1,2-a]pyrimidine-4-one and intermediates HU222110B1 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
ES09400252A ES2074966B1 (en)	1994-02-11	1994-02-11	PROCEDURE FOR OBTAINING 3- (2- (4- (6-FLUORO-BENZO (D) ISOXAZOL-3-IL) PIPERIDIN-1-IL) -ETIL) -2-METHYL-6,7,8,9- TETRAHIDRO-4H-PIRIDO- (1,2-A) PIRIMIDIN-4-ONA.

Publications (3)

Publication Number	Publication Date
HU9500418D0 true HU9500418D0 (en)	1995-03-28
HUT70169A HUT70169A (en)	1995-09-28
HU222110B1 HU222110B1 (en)	2003-04-28

Family

ID=8285178

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HU9500418A HU222110B1 (en)	1994-02-11	1995-02-10	Process for producing 3-{2-[4-(6-fluoro-benzo[d]isoxazol-3-yl)piperidine-1-il]-ethyl}-2-methyl-6,7,8,9-tetrahydro-4h-pyrido[1,2-a]pyrimidine-4-one and intermediates

Country Status (14)

Country	Link
KR (1)	KR100221108B1 (en)
AT (1)	AT405401B (en)
CZ (1)	CZ286398B6 (en)
EG (1)	EG20877A (en)
ES (1)	ES2074966B1 (en)
FI (1)	FI110000B (en)
GR (1)	GR1002344B (en)
HU (1)	HU222110B1 (en)
IS (1)	IS1766B (en)
NO (1)	NO306022B1 (en)
PL (1)	PL181420B1 (en)
PT (1)	PT101654B (en)
RU (1)	RU2123004C1 (en)
SK (1)	SK281752B6 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2101646B1 (en) *	1995-04-12	1998-04-01	Ferrer Int	NEW COMPOUND DERIVED FROM CHROMENE.
ES2144355B1 (en) *	1997-12-30	2001-01-01	Ferrer Int	COMPOUNDS DERIVED FROM THE CHROME.
EP1280804B1 (en) *	2000-05-05	2004-04-14	RPG Life Sciences Limited	A process for the preparation of anti-psychotic 3- 2- 4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4h-pyrido 1,2,-a]pyrimidin-4-one
EP1982980A1 (en)	2000-08-14	2008-10-22	Teva Pharmaceutical Industries Ltd.	Crystalline form of risperidone
KR20040034996A (en)	2002-10-18	2004-04-29	한미약품 주식회사	Improved method for the preparation of risperidone
CN100390146C (en)	2002-11-13	2008-05-28	斯索恩有限公司	Process for making risperidone and intermediates therefor
BRPI0809837A2 (en) *	2007-04-19	2014-11-11	Youxin Li	"COMPOSITION FOR TREATING MENTAL DISORDERS, BALANCE OF COMPOSITE FOR TREATING MENTAL DISORDERS, PHARMACEUTICAL COMPOSITION AND USE OF COMPOSITE FOR TREATING MENTAL DISORDERS"

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4352811A (en) *	1981-11-12	1982-10-05	Hoechst-Roussel Pharmaceuticals Inc.	3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4804663A (en) *	1985-03-27	1989-02-14	Janssen Pharmaceutica N.V.	3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) *	1987-07-13	1990-12-25	Hoechst-Roussel Pharmaceuticals Inc.	N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

1994
- 1994-02-11 ES ES09400252A patent/ES2074966B1/en not_active Expired - Fee Related
1995
- 1995-02-01 GR GR950100035A patent/GR1002344B/en not_active IP Right Cessation
- 1995-02-07 SK SK156-95A patent/SK281752B6/en not_active IP Right Cessation
- 1995-02-08 CZ CZ1995329A patent/CZ286398B6/en not_active IP Right Cessation
- 1995-02-08 IS IS4259A patent/IS1766B/en unknown
- 1995-02-09 PT PT101654A patent/PT101654B/en active IP Right Grant
- 1995-02-09 NO NO950501A patent/NO306022B1/en not_active IP Right Cessation
- 1995-02-09 EG EG11595A patent/EG20877A/en active
- 1995-02-10 FI FI950579A patent/FI110000B/en not_active IP Right Cessation
- 1995-02-10 RU RU95101859/04A patent/RU2123004C1/en not_active IP Right Cessation
- 1995-02-10 HU HU9500418A patent/HU222110B1/en not_active IP Right Cessation
- 1995-02-10 AT AT0024995A patent/AT405401B/en not_active IP Right Cessation
- 1995-02-10 PL PL95307200A patent/PL181420B1/en not_active IP Right Cessation
- 1995-02-11 KR KR1019950002516A patent/KR100221108B1/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
FI110000B (en)	2002-11-15
HU222110B1 (en)	2003-04-28
FI950579A0 (en)	1995-02-10
CZ286398B6 (en)	2000-04-12
NO950501D0 (en)	1995-02-09
KR950032196A (en)	1995-12-20
ES2074966A1 (en)	1995-09-16
HUT70169A (en)	1995-09-28
PL181420B1 (en)	2001-07-31
ES2074966B1 (en)	1996-06-16
FI950579A (en)	1995-08-12
GR1002344B (en)	1996-05-24
SK281752B6 (en)	2001-07-10
RU95101859A (en)	1997-03-20
KR100221108B1 (en)	1999-09-15
PL307200A1 (en)	1995-08-21
ATA24995A (en)	1998-12-15
PT101654A (en)	1995-09-12
PT101654B (en)	2002-01-30
NO950501L (en)	1995-08-14
NO306022B1 (en)	1999-09-06
IS1766B (en)	2001-03-15
CZ32995A3 (en)	1995-09-13
EG20877A (en)	2000-05-31
AT405401B (en)	1999-08-25
IS4259A (en)	1995-08-12
SK15695A3 (en)	1995-10-11
RU2123004C1 (en)	1998-12-10

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Legal Events

Date	Code	Title	Description
2003-04-28	HFG4	Patent granted, date of granting	Effective date: 20030312
2003-04-28	HPC4	Succession in title of patentee	Owner name: LABORATORIOS VITA S.A., ES
2005-06-28	HPC4	Succession in title of patentee	Owner name: VITA CIENTIFICA, ES
2007-12-28	GB9A	Succession in title	Owner name: INKE, S.A., ES Free format text: FORMER OWNER(S): LABORATORIOS VITA S.A., ES; VITA-INVEST S.A., ES; VITA CIENTIFICA, ES
2011-11-28	MM4A	Lapse of definitive patent protection due to non-payment of fees