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HN2001000019A - Derivados de nicotinamida benzocondensada heterociclico utiles como inhibidores selectivos de las isozimas pde4. - Google Patents

Derivados de nicotinamida benzocondensada heterociclico utiles como inhibidores selectivos de las isozimas pde4.

Info

Publication number
HN2001000019A
HN2001000019A HN2001000019A HN2001000019A HN2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A HN 2001000019 A HN2001000019 A HN 2001000019A
Authority
HN
Honduras
Prior art keywords
pde4
isozimas
benzocondensada
heterociclico
nicotinamide
Prior art date
Application number
HN2001000019A
Other languages
English (en)
Inventor
Chambers Robert James
Marfat Anthony
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of HN2001000019A publication Critical patent/HN2001000019A/es

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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Abstract

LA PRESENTE INVENCION SE REFIERE TAMBIEN AL USO DE INHIBIDORES SELECTIVOS DE LAS PDE4 PARA UN MEJOR TRATAMIENTO TERAPEUTICO DE UNA SERIE DE ENFERMEDADES Y CONDICIONES INFLAMATORIAS, RESPIRATORIAS Y ALERGICAS, PERO ESPECIALMENTE PARA EL TRATAMIENTO DEL ASMA
HN2001000019A 2000-01-31 2001-06-30 Derivados de nicotinamida benzocondensada heterociclico utiles como inhibidores selectivos de las isozimas pde4. HN2001000019A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17928400P 2000-01-31 2000-01-31

Publications (1)

Publication Number Publication Date
HN2001000019A true HN2001000019A (es) 2001-09-06

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HN2001000019A HN2001000019A (es) 2000-01-31 2001-06-30 Derivados de nicotinamida benzocondensada heterociclico utiles como inhibidores selectivos de las isozimas pde4.

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US (1) US7354941B2 (es)
EP (1) EP1252158B1 (es)
JP (1) JP3917863B2 (es)
KR (1) KR20020072299A (es)
CN (1) CN1404481A (es)
AP (1) AP2002002589A0 (es)
AR (1) AR027337A1 (es)
AT (1) ATE293624T1 (es)
AU (1) AU2700201A (es)
BG (1) BG106852A (es)
BR (1) BR0107964A (es)
CA (1) CA2398182C (es)
CO (1) CO5261634A1 (es)
CZ (1) CZ20022410A3 (es)
DE (1) DE60110205T2 (es)
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EE (1) EE200200425A (es)
ES (1) ES2238415T3 (es)
GE (1) GEP20043302B (es)
GT (1) GT200100022A (es)
HN (1) HN2001000019A (es)
HU (1) HUP0204262A2 (es)
IL (1) IL150641A0 (es)
IS (1) IS6421A (es)
MA (1) MA26870A1 (es)
MX (1) MXPA02007419A (es)
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PT (1) PT1252158E (es)
SK (1) SK10142002A3 (es)
SV (1) SV2002000299A (es)
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UY (1) UY26569A1 (es)
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WO2000021509A2 (en) * 1998-10-15 2000-04-20 Imperial College Innovations Limited Methods of treatment
ATE292957T1 (de) * 2000-01-28 2005-04-15 Alza Corp Liposomen enthaltend eine eingeschlossene verbindung in übersattigter lösung
JP2004518629A (ja) 2000-09-18 2004-06-24 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 殺菌・殺カビ剤として使用するためのピリジニルアミド類およびイミド類
IL156412A0 (en) 2001-01-31 2004-01-04 Pfizer Prod Inc Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes
WO2002060896A1 (en) 2001-01-31 2002-08-08 Pfizer Products Inc. Ether derivatives useful as inhibitors of pde4 isozymes
US7250518B2 (en) 2001-01-31 2007-07-31 Pfizer Inc. Nicotinamide acids, amides, and their mimetics active as inhibitors of PDE4 isozymes
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