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HK1223270A1 - 長效螺異惡唑啉製劑 - Google Patents

長效螺異惡唑啉製劑

Info

Publication number
HK1223270A1
HK1223270A1 HK16111350.3A HK16111350A HK1223270A1 HK 1223270 A1 HK1223270 A1 HK 1223270A1 HK 16111350 A HK16111350 A HK 16111350A HK 1223270 A1 HK1223270 A1 HK 1223270A1
Authority
HK
Hong Kong
Prior art keywords
long
acting
spiro
isoxazoline
composition
Prior art date
Application number
HK16111350.3A
Other languages
English (en)
Inventor
Todd P. Foster
Laibin Luo
Original Assignee
硕腾服务有限责任公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 硕腾服务有限责任公司 filed Critical 硕腾服务有限责任公司
Publication of HK1223270A1 publication Critical patent/HK1223270A1/zh

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1641Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647Polyesters, e.g. poly(lactide-co-glycolide)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Inorganic Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
HK16111350.3A 2013-09-30 2014-09-26 長效螺異惡唑啉製劑 HK1223270A1 (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361884467P 2013-09-30 2013-09-30
US61/884,467 2013-09-30
PCT/US2014/057588 WO2015048371A1 (en) 2013-09-30 2014-09-26 Long-acting spiro-isoxazoline formulations

Publications (1)

Publication Number Publication Date
HK1223270A1 true HK1223270A1 (zh) 2017-07-28

Family

ID=51794952

Family Applications (1)

Application Number Title Priority Date Filing Date
HK16111350.3A HK1223270A1 (zh) 2013-09-30 2014-09-26 長效螺異惡唑啉製劑

Country Status (10)

Country Link
US (1) US10350196B2 (zh)
EP (1) EP3052080B1 (zh)
JP (1) JP6209272B2 (zh)
CN (1) CN105579029B (zh)
AU (1) AU2014324837B2 (zh)
BR (1) BR112016006182B1 (zh)
CA (1) CA2924537C (zh)
HK (1) HK1223270A1 (zh)
MX (1) MX374480B (zh)
WO (1) WO2015048371A1 (zh)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110327468B (zh) 2013-12-20 2023-04-28 英特维特国际股份有限公司 异噁唑啉组合物及其在预防或治疗动物的寄生虫侵袭中的用途
EA036272B1 (ru) * 2015-04-08 2020-10-21 БЁРИНГЕР ИНГЕЛЬХАЙМ ЭНИМАЛ ХЕЛТ ЮЭсЭй ИНК. Инъецируемые препараты замедленного высвобождения, содержащие изоксазолиновое действующее вещество, способы и применение
PL3313400T3 (pl) 2015-06-23 2022-07-25 Intervet International B.V. Roztwór izoksazoliny zawierający witaminę e do stosowania z odkażoną wodą pitną
UY37137A (es) * 2016-02-24 2017-09-29 Merial Inc Compuestos antiparasitarios de isoxazolina, formulaciones inyectables de acción prolongada que los comprenden, métodos y usos de los mismos
IL297676B2 (en) 2016-03-25 2023-12-01 Intra Cellular Therapies Inc A sustained-release or delayed-release pharmaceutical composition comprising a deuterated compound
WO2017201134A1 (en) * 2016-05-20 2017-11-23 Avista Pharma Solutions, Inc. Synthetic process and novel intermediates
WO2018071233A1 (en) 2016-10-12 2018-04-19 Intra-Cellular Therapies, Inc. Amorphous solid dispersions
RU2022103663A (ru) 2017-03-24 2022-04-07 Интра-Селлулар Терапиз, Инк. Новые композиции и способы
BR112020008853A2 (pt) 2017-11-07 2020-10-13 Intervet International B.V. composições farmacêuticas injetáveis de isoxazolina e seu uso contra infestação parasitária
PE20210170A1 (es) 2017-11-07 2021-01-29 Intervet Int Bv Proceso para preparar particulas de isoxazolina de gran tamano
EP3723483A1 (en) 2017-12-12 2020-10-21 Intervet International B.V. Implantable isoxazoline pharmaceutical compositions and uses thereof
AR113997A1 (es) 2017-12-21 2020-07-08 Intervet Int Bv Composiciones antiparasitarias para unción dorsal continua
CN110787661A (zh) * 2018-08-01 2020-02-14 台鉅生技股份有限公司 聚合物-胶原蛋白复合膜及其制造方法
US12144808B2 (en) 2018-08-29 2024-11-19 Intra-Cellular Therapies, Inc. Compositions and methods
CN109053751A (zh) * 2018-08-30 2018-12-21 成都海博锐药业有限公司 具有螺环结构的fxr调节剂
WO2020047407A1 (en) 2018-08-31 2020-03-05 Intra-Cellular Therapies, Inc. Novel methods
CN118873536A (zh) 2018-08-31 2024-11-01 细胞内治疗公司 新方法
MX2021013429A (es) 2019-05-03 2021-12-10 Intervet Int Bv Composiciones farmaceuticas inyectables y usos de las mismas.
US20230310386A1 (en) 2020-05-20 2023-10-05 Intervet Inc. Injectable pharmaceutical compositions and uses thereof
CA3185969A1 (en) 2020-07-24 2022-01-27 Jean Marie Defauw Process for making an isoxazoline compound and intermediate thereof

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE744162A (fr) 1969-01-16 1970-06-15 Fuji Photo Film Co Ltd Procede d'encapsulage
JPS523342B2 (zh) 1972-01-26 1977-01-27
US4389330A (en) 1980-10-06 1983-06-21 Stolle Research And Development Corporation Microencapsulation process
JPS6098823A (ja) 1983-11-02 1985-06-01 株式会社東芝 電力変換装置
US6136838A (en) 1998-03-19 2000-10-24 Merck & Co., Inc. Sulfurpentafluorophenylpyrazoles for controlling ectoparasitic infestations
US6726918B1 (en) 2000-07-05 2004-04-27 Oculex Pharmaceuticals, Inc. Methods for treating inflammation-mediated conditions of the eye
GB2386066A (en) * 2002-02-28 2003-09-10 Norbrook Lab Ltd Long-acting parasiticidal composition with improved bioavailability comprising a salicylanilide, a further anti-parasitic compound & a polymeric species
US7589057B2 (en) 2004-04-30 2009-09-15 Allergan, Inc. Oil-in-water method for making alpha-2 agonist polymeric drug delivery systems
US8362086B2 (en) * 2005-08-19 2013-01-29 Merial Limited Long acting injectable formulations
TW200846029A (en) * 2007-02-09 2008-12-01 Wyeth Corp High dose, long-acting ectoparasiticide for extended control
WO2012001083A2 (en) * 2010-06-29 2012-01-05 Ceva Sante Animale Sa Novel eprinomectin injectable compositions
JP5806743B2 (ja) * 2011-03-10 2015-11-10 ゾエティス・エルエルシー 抗寄生虫薬としてのスピロ環式イソオキサゾリン誘導体
BRPI1103229B1 (pt) * 2011-07-18 2020-10-06 Universidade Federal Do Rio De Janeiro Composições farmacêuticas microparticuladas contendo antiparasitários para terapia subcutânea prolongada, uso das ditas composições farmacêuticas para a produção de um medicamento e método de tratamento de parasitoses

Also Published As

Publication number Publication date
CA2924537C (en) 2018-01-16
CN105579029A (zh) 2016-05-11
BR112016006182A2 (pt) 2017-08-01
AU2014324837B2 (en) 2019-01-17
JP2016536272A (ja) 2016-11-24
CN105579029B (zh) 2019-03-05
US20160235720A1 (en) 2016-08-18
MX374480B (es) 2025-03-06
US10350196B2 (en) 2019-07-16
WO2015048371A1 (en) 2015-04-02
BR112016006182A8 (pt) 2020-02-18
EP3052080B1 (en) 2025-06-25
EP3052080A1 (en) 2016-08-10
AU2014324837A1 (en) 2016-03-17
JP6209272B2 (ja) 2017-10-04
CA2924537A1 (en) 2015-04-02
MX2016004035A (es) 2016-06-02
BR112016006182B1 (pt) 2023-01-10

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