HK1213181A1 - 雙環氧雜內酰胺激酶抑制劑 - Google Patents
雙環氧雜內酰胺激酶抑制劑Info
- Publication number
- HK1213181A1 HK1213181A1 HK16101135.6A HK16101135A HK1213181A1 HK 1213181 A1 HK1213181 A1 HK 1213181A1 HK 16101135 A HK16101135 A HK 16101135A HK 1213181 A1 HK1213181 A1 HK 1213181A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- kinase inhibitors
- oxa
- bicyclic
- lactam kinase
- lactam
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261706712P | 2012-09-27 | 2012-09-27 | |
| PCT/US2013/000225 WO2014051654A2 (en) | 2012-09-27 | 2013-09-27 | Bicyclic oxa-lactam kinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HK1213181A1 true HK1213181A1 (zh) | 2016-06-30 |
Family
ID=50389107
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HK16101135.6A HK1213181A1 (zh) | 2012-09-27 | 2016-02-01 | 雙環氧雜內酰胺激酶抑制劑 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US9469654B2 (zh) |
| EP (1) | EP2900243A4 (zh) |
| HK (1) | HK1213181A1 (zh) |
| WO (1) | WO2014051654A2 (zh) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2900243A4 (en) | 2012-09-27 | 2016-04-13 | Portola Pharm Inc | BICYCLIC OXA LACTAM KINASE HEMMER |
| BR112021018168B1 (pt) | 2019-03-21 | 2023-11-28 | Onxeo | Composição farmacêutica, combinação e kit compreendendo uma molécula dbait e um inibidor de quinase para o tratamento de câncer |
| CA3159348A1 (en) | 2019-11-08 | 2021-05-14 | Inserm (Institut National De La Sante Et De La Recherche Medicale) | Methods for the treatment of cancers that have acquired resistance to kinase inhibitors |
| WO2021148581A1 (en) | 2020-01-22 | 2021-07-29 | Onxeo | Novel dbait molecule and its use |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999016758A1 (en) * | 1997-10-27 | 1999-04-08 | Dr. Reddy's Research Foundation | Novel heterocyclic compounds and their use in medicine, process for their preparation and pharmaceutical compositions containing them |
| ZA200702688B (en) * | 2004-09-29 | 2008-06-25 | Portola Pharm Inc | Substituted 2H-1,3-benzoxazin-4-(3H)-ones |
| SG10201707798SA (en) * | 2008-12-08 | 2017-10-30 | Gilead Connecticut Inc | Imidazopyrazine syk inhibitors |
| EA201190062A1 (ru) | 2009-01-13 | 2012-02-28 | Глаксо Груп Лимитед | Производные пиримидинкарбоксамида в качестве ингибиторов syk-киназы |
| WO2011012883A1 (en) | 2009-07-29 | 2011-02-03 | Karus Therapeutics Limited | Benzo [e] [1, 3 ] oxazin-4-one derivatives as phosphoinositide 3-kinase inhibitors |
| MA33909B1 (fr) | 2009-12-23 | 2013-01-02 | Takeda Pharmaceutical | Pyrrolidinones accoles en tant d'inhibiteurs de syk |
| AU2011323484B2 (en) | 2010-11-01 | 2016-10-06 | Portola Pharmaceuticals, Inc. | Benzamides and nicotinamides as Syk modulators |
| EP2900243A4 (en) | 2012-09-27 | 2016-04-13 | Portola Pharm Inc | BICYCLIC OXA LACTAM KINASE HEMMER |
-
2013
- 2013-09-27 EP EP13840922.2A patent/EP2900243A4/en not_active Withdrawn
- 2013-09-27 WO PCT/US2013/000225 patent/WO2014051654A2/en active Application Filing
- 2013-09-27 US US14/432,162 patent/US9469654B2/en active Active
-
2016
- 2016-02-01 HK HK16101135.6A patent/HK1213181A1/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2014051654A2 (en) | 2014-04-03 |
| WO2014051654A3 (en) | 2014-05-22 |
| EP2900243A2 (en) | 2015-08-05 |
| US9469654B2 (en) | 2016-10-18 |
| US20150252056A1 (en) | 2015-09-10 |
| EP2900243A4 (en) | 2016-04-13 |
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