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FR2424919A1 - SUBSTITUTE QUINOLEINECARBOXYLIC ACID AND ITS DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS - Google Patents

SUBSTITUTE QUINOLEINECARBOXYLIC ACID AND ITS DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS

Info

Publication number
FR2424919A1
FR2424919A1 FR7813217A FR7813217A FR2424919A1 FR 2424919 A1 FR2424919 A1 FR 2424919A1 FR 7813217 A FR7813217 A FR 7813217A FR 7813217 A FR7813217 A FR 7813217A FR 2424919 A1 FR2424919 A1 FR 2424919A1
Authority
FR
France
Prior art keywords
acid
derivatives
quinoleinecarboxylic
substitute
antibacterial agents
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7813217A
Other languages
French (fr)
Other versions
FR2424919B1 (en
Inventor
Tsutomu Irikura
Seigo Suzue
Akiro Ito
Hiroshi Koga
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kyorin Pharmaceutical Co Ltd
Original Assignee
Kyorin Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kyorin Pharmaceutical Co Ltd filed Critical Kyorin Pharmaceutical Co Ltd
Priority to FR7813217A priority Critical patent/FR2424919B1/en
Publication of FR2424919A1 publication Critical patent/FR2424919A1/en
Application granted granted Critical
Publication of FR2424919B1 publication Critical patent/FR2424919B1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

ACIDE QUINOLEINECARBOXYLIQUE SUBSTITUE ET SES DERIVES, AINSI QUE LEURS UTILISATIONS. CET ACIDE EST L'ACIDE 1-ETHYL-6-FLUORO-7-(4-METHYL-1-PIPERAZINYL)-4-OXO-1,4-DIHYDROQUINOLEINE-3-CARBOXYLIQUE AYANT LA FORMULE: (CF DESSIN DANS BOPI) LES DERIVES UTILES DE CET ACIDE SONT LES SELS D'ADDITION AVEC LES ACIDES, LES SELS ALCALINS ET LES HYDRATES. LA PRESENTE INVENTION EST PARTICULIEREMENT UTILE POUR FOURNIR UN ACIDE QUINOLEINECARBOXYLIQUE SUBSTITUE, AINSI QUE SES DERIVES, EMPLOYES COMME AGENTS ANTIBACTERIENS PUISSANTS.SUBSTITUTE QUINOLEINECARBOXYLIC ACID AND ITS DERIVATIVES AND THEIR USES. THIS ACID IS 1-ETHYL-6-FLUORO-7- (4-METHYL-1-PIPERAZINYL) -4-OXO-1,4-DIHYDROQUINOLEINE-3-CARBOXYLIC ACID WITH THE FORMULA: (DRAWING IN BOPI) USEFUL DERIVATIVES OF THIS ACID ARE ADDITIONAL SALTS WITH ACIDS, ALKALINE SALTS AND HYDRATES. THE PRESENT INVENTION IS PARTICULARLY USEFUL FOR PROVIDING A SUBSTITUTE QUINOLEINECARBOXYLIC ACID, AS WELL AS ITS DERIVATIVES, USED AS POWERFUL ANTIBACTERIAL AGENTS.

FR7813217A 1978-05-03 1978-05-03 SUBSTITUTED QUINOLEINECARBOXYLIC ACID AND DERIVATIVES THEREOF AND THEIR USE AS ANTIBACTERIAL AGENTS Expired FR2424919B1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR7813217A FR2424919B1 (en) 1978-05-03 1978-05-03 SUBSTITUTED QUINOLEINECARBOXYLIC ACID AND DERIVATIVES THEREOF AND THEIR USE AS ANTIBACTERIAL AGENTS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7813217A FR2424919B1 (en) 1978-05-03 1978-05-03 SUBSTITUTED QUINOLEINECARBOXYLIC ACID AND DERIVATIVES THEREOF AND THEIR USE AS ANTIBACTERIAL AGENTS

Publications (2)

Publication Number Publication Date
FR2424919A1 true FR2424919A1 (en) 1979-11-30
FR2424919B1 FR2424919B1 (en) 1980-10-31

Family

ID=9207900

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7813217A Expired FR2424919B1 (en) 1978-05-03 1978-05-03 SUBSTITUTED QUINOLEINECARBOXYLIC ACID AND DERIVATIVES THEREOF AND THEIR USE AS ANTIBACTERIAL AGENTS

Country Status (1)

Country Link
FR (1) FR2424919B1 (en)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2403339A1 (en) * 1977-09-20 1979-04-13 Bellon Labor Sa Roger 6-Halo-7-tert. amino-4-oxo-quinoline carboxylic acid derivs. - broad spectrum antibacterials and growth promoters for animals
EP0181521A1 (en) * 1984-10-19 1986-05-21 Otsuka Pharmaceutical Co., Ltd. Antimicrobial 1-substituted Phenyl-4-oxoquinoline-3-carboxylic acid compounds
WO1987003595A1 (en) 1985-12-09 1987-06-18 Chinoin Gyógyszer és Vegyészeti Termékek Gyára Rt. Norfloxacin intermediate
US4684648A (en) * 1985-05-10 1987-08-04 Otsuka Pharmaceutical Company Limited Antimicrobial 1-substituted phenyl-4-oxoquinoline-3-carboxylic acid compounds and compositions thereof
US4755513A (en) * 1985-01-30 1988-07-05 Otsuka Pharmaceutical Company, Limited Antimicrobial 1-substituted phenyl-4-oxoquinoline-3-carboxylic acid compounds
EP0351889A1 (en) 1985-12-09 1990-01-24 CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. Process for the preparation of a quinoline carboxylic acid

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2210413A1 (en) * 1972-12-18 1974-07-12 Dainippon Pharmaceutical Co

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2210413A1 (en) * 1972-12-18 1974-07-12 Dainippon Pharmaceutical Co

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2403339A1 (en) * 1977-09-20 1979-04-13 Bellon Labor Sa Roger 6-Halo-7-tert. amino-4-oxo-quinoline carboxylic acid derivs. - broad spectrum antibacterials and growth promoters for animals
FR2498931A1 (en) * 1977-09-20 1982-08-06 Bellon Labor Sa Roger MEDICAMENT CONSISTING OF THE ACID ETHYL-1 FLUORO-6 PIPERAZINYL-7-OXO-4-DIHYDRO-1,4 QUINOLIN-3-CARBOXYLIC AND ITS SALTS OF ADDITION OF NON-TOXIC ACIDS PHARMACEUTICALLY ACCEPTABLE
EP0181521A1 (en) * 1984-10-19 1986-05-21 Otsuka Pharmaceutical Co., Ltd. Antimicrobial 1-substituted Phenyl-4-oxoquinoline-3-carboxylic acid compounds
US4755513A (en) * 1985-01-30 1988-07-05 Otsuka Pharmaceutical Company, Limited Antimicrobial 1-substituted phenyl-4-oxoquinoline-3-carboxylic acid compounds
US4684648A (en) * 1985-05-10 1987-08-04 Otsuka Pharmaceutical Company Limited Antimicrobial 1-substituted phenyl-4-oxoquinoline-3-carboxylic acid compounds and compositions thereof
WO1987003595A1 (en) 1985-12-09 1987-06-18 Chinoin Gyógyszer és Vegyészeti Termékek Gyára Rt. Norfloxacin intermediate
EP0351889A1 (en) 1985-12-09 1990-01-24 CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. Process for the preparation of a quinoline carboxylic acid

Also Published As

Publication number Publication date
FR2424919B1 (en) 1980-10-31

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