FR2313046A1 - Derives acylamino de composes heterocycliques - Google Patents

Derives acylamino de composes heterocycliques

Info

Publication number: FR2313046A1
Authority: FR; France
Prior art keywords: heterocyclic compounds; acylamino derivatives; acylamino; derivatives; heterocyclic
Prior art date: 1975-06-05
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

FR7616973A

Other languages

English (en)

Other versions

FR2313046B1 (fr

Inventor

Roger Garrick Harrison

William Boffey Jamieson

William James Ross

John Christopher Saunders

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Lilly Industries Ltd

Original Assignee

Lilly Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1975-06-05

Filing date

1976-06-04

Publication date

1976-12-31

1976-06-04 Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd

1976-12-31 Publication of FR2313046A1 publication Critical patent/FR2313046A1/fr

1982-09-24 Application granted granted Critical

1982-09-24 Publication of FR2313046B1 publication Critical patent/FR2313046B1/fr

Status Granted legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
- C07D231/40—Acylated on said nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/88—Nitrogen atoms, e.g. allantoin
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/04—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
- C07D249/06—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles with aryl radicals directly attached to ring atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/14—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
- C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D257/04—Five-membered rings
- C07D257/06—Five-membered rings with nitrogen atoms directly attached to the ring carbon atom

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

FR7616973A 1975-06-05 1976-06-04 Derives acylamino de composes heterocycliques Granted FR2313046A1 (fr)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB24225/75A GB1547564A (en)	1975-06-05	1975-06-05	Acylated amino-heteroaryl compounds

Publications (2)

Publication Number	Publication Date
FR2313046A1 true FR2313046A1 (fr)	1976-12-31
FR2313046B1 FR2313046B1 (fr)	1982-09-24

Family

ID=10208295

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FR7616973A Granted FR2313046A1 (fr)	1975-06-05	1976-06-04	Derives acylamino de composes heterocycliques

Country Status (31)

Country	Link
US (2)	US4166123A (fr)
JP (1)	JPS51146465A (fr)
AR (2)	AR219280A1 (fr)
AT (1)	AT355562B (fr)
AU (1)	AU506564B2 (fr)
BE (1)	BE842578A (fr)
BG (2)	BG26515A3 (fr)
CA (1)	CA1081219A (fr)
CH (2)	CH618972A5 (fr)
CS (1)	CS219320B2 (fr)
DD (1)	DD125206A5 (fr)
DE (1)	DE2625227A1 (fr)
DK (1)	DK243576A (fr)
ES (2)	ES448477A1 (fr)
FR (1)	FR2313046A1 (fr)
GB (1)	GB1547564A (fr)
GR (1)	GR60336B (fr)
HU (1)	HU174190B (fr)
IE (1)	IE43579B1 (fr)
IL (1)	IL49691A (fr)
MX (1)	MX3638E (fr)
NL (1)	NL7606179A (fr)
NZ (1)	NZ181010A (fr)
PH (1)	PH14627A (fr)
PL (2)	PL101455B1 (fr)
PT (1)	PT65180B (fr)
RO (1)	RO70771A (fr)
SE (1)	SE431646B (fr)
SU (2)	SU648094A3 (fr)
YU (2)	YU137276A (fr)
ZA (1)	ZA763210B (fr)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0459887A1 (fr) *	1990-05-30	1991-12-04	Novapharme	Dérivés N-pyrazolyl-ortho-dialkyl-benzamide doués d'activité anticonvulsivante, procédé de préparation et composition pharmaceutique
US5258397A (en) *	1988-11-30	1993-11-02	Novapharme	3-Isoxazoyl derivatives endowed with anticonvulsant activity, procedure for their preparation and their pharmaceutical compositions
US5464860A (en) *	1988-11-30	1995-11-07	Novapharme	N(pyrazol-3-yl) benzamides and pharmaceutical compositions

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL7810634A (nl) *	1977-10-28	1979-05-02	May & Baker Ltd	Tetrazool-derivaten.
DK89480A (da) *	1979-03-02	1980-09-03	Glaxo Group Ltd	R fremgangsmaade til fremstilling af heterocycliske forbindelse
MA19269A1 (fr) *	1980-09-16	1982-04-01	Lilly Co Eli	Perfectionnement relatif a des derives de n-arylbenzamides .
US4801718A (en) *	1980-09-16	1989-01-31	Eli Lilly And Company	Thiaiazolyl benzamides
US5086184A (en) *	1980-09-16	1992-02-04	Dowelanco	N-heterocyclic benzamides
US4943634A (en) *	1980-09-16	1990-07-24	Eli Lilly And Company	N-heterocyclic benzamides
DE3100516A1 (de) *	1981-01-10	1982-08-12	C.H. Boehringer Sohn, 6507 Ingelheim	Pyridylaminobenzoesaeuren, ihre herstellung und verwendung
US5073566A (en) *	1989-11-30	1991-12-17	Eli Lilly And Company	Angiotensin ii antagonist 1,3-imidazoles and use thereas
US5612360A (en) *	1992-06-03	1997-03-18	Eli Lilly And Company	Angiotensin II antagonists
US5401851A (en) *	1992-06-03	1995-03-28	Eli Lilly And Company	Angiotensin II antagonists
AU5135998A (en) *	1996-12-03	1998-06-29	Banyu Pharmaceutical Co., Ltd.	Novel urea derivatives
DE69719544T2 (de) *	1996-12-12	2003-11-06	Banyu Pharmaceutical Co., Ltd.	Pyrazolderivate
WO1998025908A1 (fr) *	1996-12-13	1998-06-18	Banyu Pharmaceutical Co., Ltd.	Nouveaux derives d'aminopyrazole
EP0945440B1 (fr)	1996-12-16	2004-05-26	Banyu Pharmaceutical Co., Ltd.	Derives d'aminopyrazole
US6906069B1 (en)	1999-01-08	2005-06-14	Amgen Inc.	LXR modulators
AU2000235960A1 (en) *	2000-02-14	2001-08-27	Tularik, Inc.	Lxr modulators
US6673543B2 (en)	2000-04-05	2004-01-06	Tularik, Inc.	Solid phase synthesis of LXR ligands
WO2002023986A1 (fr) *	2000-08-25	2002-03-28	Sankyo Company, Limited	Derives de 4-acylaminopyrazole
JP4434745B2 (ja) *	2002-01-30	2010-03-17	アムジェンインコーポレイテッド	複素環式アリールスルホンアミドベンジル化合物
US7335779B2 (en) *	2002-03-08	2008-02-26	Quonova, Llc	Modulation of pathogenicity
KR100849021B1 (ko)	2007-06-19	2008-07-29	(주)더페이스샵코리아	카페익산 유도체 및 이를 함유하는 조성물
BR102020008433A2 (pt)	2020-04-28	2021-11-03	Universidade Federal Do Parana	Repelentes de artrópodes obtidos a partir da transformação química de ácido lático, lactatos ou outros derivados do ácido lático

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA698428A (en)		1964-11-24	W. Lynn John	Substituted triazole compounds and polymerization products thereof
US2467895A (en) *	1946-04-12	1949-04-19	American Cyanamid Co	Piperazine derivatives and method of preparing the same
US2953491A (en) *	1957-11-21	1960-09-20	American Cyanamid Co	Fungicide
US2914536A (en) *	1957-11-21	1959-11-24	American Cyanamid Co	Novel 3-acylamino triazoles
GB1111680A (en)	1965-12-01	1968-05-01	Shell Int Research	Improvements in or relating to ester-base compositions
US3457350A (en) *	1966-10-26	1969-07-22	American Cyanamid Co	Method of treating asthma
GB1497536A (en)	1973-12-17	1978-01-12	Lilly Industries Ltd	2-acylaminooxazoles methods for their preparation and their use

1975
- 1975-06-05 GB GB24225/75A patent/GB1547564A/en not_active Expired
1976
- 1976-05-31 NZ NZ181010A patent/NZ181010A/xx unknown
- 1976-05-31 IE IE1147/76A patent/IE43579B1/en unknown
- 1976-05-31 CA CA253,705A patent/CA1081219A/fr not_active Expired
- 1976-05-31 IL IL49691A patent/IL49691A/xx unknown
- 1976-06-01 AR AR263472A patent/AR219280A1/es active
- 1976-06-01 US US05/691,742 patent/US4166123A/en not_active Expired - Lifetime
- 1976-06-01 US US05/691,963 patent/US4089962A/en not_active Expired - Lifetime
- 1976-06-01 ZA ZA00763210A patent/ZA763210B/xx unknown
- 1976-06-01 RO RO7686316A patent/RO70771A/fr unknown
- 1976-06-01 GR GR50867A patent/GR60336B/el unknown
- 1976-06-02 DK DK243576A patent/DK243576A/da not_active Application Discontinuation
- 1976-06-02 CH CH691676A patent/CH618972A5/fr not_active IP Right Cessation
- 1976-06-02 ES ES448477A patent/ES448477A1/es not_active Expired
- 1976-06-02 SE SE7606225A patent/SE431646B/xx unknown
- 1976-06-03 YU YU01372/76A patent/YU137276A/xx unknown
- 1976-06-03 AU AU14618/76A patent/AU506564B2/en not_active Ceased
- 1976-06-03 PT PT65180A patent/PT65180B/pt unknown
- 1976-06-03 BE BE6045538A patent/BE842578A/fr not_active IP Right Cessation
- 1976-06-03 HU HU76LI292A patent/HU174190B/hu unknown
- 1976-06-04 MX MX76267U patent/MX3638E/es unknown
- 1976-06-04 DD DD193192A patent/DD125206A5/xx unknown
- 1976-06-04 PL PL1976196533A patent/PL101455B1/pl unknown
- 1976-06-04 BG BG033364A patent/BG26515A3/xx unknown
- 1976-06-04 SU SU762367202A patent/SU648094A3/ru active
- 1976-06-04 DE DE19762625227 patent/DE2625227A1/de not_active Withdrawn
- 1976-06-04 AT AT412376A patent/AT355562B/de not_active IP Right Cessation
- 1976-06-04 PL PL1976190125A patent/PL101468B1/pl unknown
- 1976-06-04 PH PH18537A patent/PH14627A/en unknown
- 1976-06-04 JP JP51066026A patent/JPS51146465A/ja active Pending
- 1976-06-04 CS CS763712A patent/CS219320B2/cs unknown
- 1976-06-04 FR FR7616973A patent/FR2313046A1/fr active Granted
- 1976-06-08 NL NL7606179A patent/NL7606179A/xx not_active Application Discontinuation
- 1976-06-09 YU YU01233/76A patent/YU123376A/xx unknown
- 1976-09-22 BG BG034256A patent/BG25211A3/xx unknown
1977
- 1977-04-07 SU SU772468107A patent/SU654168A3/ru active
- 1977-07-13 ES ES460711A patent/ES460711A1/es not_active Expired
- 1977-11-25 AR AR270117A patent/AR217662A1/es active
1980
- 1980-01-22 CH CH49980A patent/CH622254A5/fr not_active IP Right Cessation

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5258397A (en) *	1988-11-30	1993-11-02	Novapharme	3-Isoxazoyl derivatives endowed with anticonvulsant activity, procedure for their preparation and their pharmaceutical compositions
US5464860A (en) *	1988-11-30	1995-11-07	Novapharme	N(pyrazol-3-yl) benzamides and pharmaceutical compositions
EP0459887A1 (fr) *	1990-05-30	1991-12-04	Novapharme	Dérivés N-pyrazolyl-ortho-dialkyl-benzamide doués d'activité anticonvulsivante, procédé de préparation et composition pharmaceutique
FR2662692A1 (fr) *	1990-05-30	1991-12-06	Novapharme	Derives heterocycliques doues d'activite anticonvulsivante, procede de preparation et composition pharmaceutique.

Also Published As

Publication number	Publication date
JPS51146465A (en)	1976-12-16
DK243576A (da)	1976-12-06
DE2625227A1 (de)	1976-12-23
AU1461876A (en)	1977-12-08
PT65180A (en)	1976-07-01
SU648094A3 (ru)	1979-02-15
US4089962A (en)	1978-05-16
IE43579B1 (en)	1981-04-08
ZA763210B (en)	1978-01-25
CA1081219A (fr)	1980-07-08
AR217662A1 (es)	1980-04-15
BE842578A (fr)	1976-12-03
RO70771B (ro)	1983-07-30
FR2313046B1 (fr)	1982-09-24
CH622254A5 (fr)	1981-03-31
IE43579L (en)	1976-12-05
IL49691A0 (en)	1976-07-30
AT355562B (de)	1980-03-10
AR219280A1 (es)	1980-08-15
NZ181010A (en)	1978-04-28
SE7606225L (sv)	1976-12-06
SE431646B (sv)	1984-02-20
PH14627A (en)	1981-10-12
GB1547564A (en)	1979-06-20
ES460711A1 (es)	1978-04-16
DD125206A5 (fr)	1977-04-06
ES448477A1 (es)	1977-11-01
YU137276A (en)	1982-10-31
BG25211A3 (en)	1978-08-10
YU123376A (en)	1982-10-31
AU506564B2 (en)	1980-01-10
PL101468B1 (pl)	1978-12-30
PT65180B (en)	1978-11-06
IL49691A (en)	1980-09-16
NL7606179A (nl)	1976-12-07
GR60336B (en)	1978-05-09
ATA412376A (de)	1979-08-15
BG26515A3 (bg)	1979-04-12
MX3638E (es)	1981-04-13
CS219320B2 (en)	1983-03-25
RO70771A (fr)	1983-08-03
US4166123A (en)	1979-08-28
PL101455B1 (pl)	1978-12-30
CH618972A5 (fr)	1980-08-29
SU654168A3 (ru)	1979-03-25
HU174190B (hu)	1979-11-28

Publication	Publication Date	Title
FR2313046A1 (fr)	1976-12-31	Derives acylamino de composes heterocycliques
BE868532A (fr)	1978-10-16	Nouveaux derives de la thiazolidine
SE7606224L (sv)	1976-12-06	Forfarande for framstellning av heterocykliska acylaminoderivat
FI773640A (fi)	1978-06-04	Derivat av tiazolidinkarboxylsyror och naerliggande syror
FR2298332A1 (fr)	1976-08-20	Nouveaux derives de 5-fluorouraciles
FR2316926A1 (fr)	1977-02-04	Nouveaux derives de bicycloheptenes
FR2301253A1 (fr)	1976-09-17	Derives de la
FR2319348A1 (fr)	1977-02-25	Derives de n-alkyl-imidazoles substitues
FR2301571A1 (fr)	1976-09-17	Colorants azoiques derivant de diazos de composes heterocycliques
SE7606226L (sv)	1976-12-06	Acylaminoderivat
NO770959L (no)	1977-09-20	Heterocykliske derivater av guanidiner.
BE838128A (fr)	1976-07-30	Composes heterocycliques
BE853578A (fr)	1977-10-14	Derives de thiouree
SE7707407L (sv)	1977-12-29	Forfarande for framstellning av cefamderivat
BE850245A (fr)	1977-07-11	Derives acylamino(alkyl)-benzeniques
PL190247A1 (pl)	1978-03-13	Sposob wytwarzania nowych podstawionych heterocyklicznych n-alkanoloamin
BE859567A (fr)	1978-04-11	Derives piperidylideniques de benzo-xanthenes
FR2313074A1 (fr)	1976-12-31	Diastereoisomeres de derives phenylaminoethanol
FR2306694A1 (fr)	1976-11-05	Derives de la piperazine
RO73050A (fr)	1981-08-30	Procede pour la preparation des derives d'aminoquinazoline
ZA771644B (en)	1978-10-25	Heterocyclic derivatives of guanidine
DK243376A (da)	1976-12-08	Acylaminoderivater
FR2306701A1 (fr)	1976-11-05	Derives de nucleotides
BE861155A (fr)	1978-03-16	Derives sulfamoyles de la 8beta-aminomethylergoline
BE829785A (fr)	1975-10-01	Nouveaux derives de pyrazole

Legal Events

Date	Code	Title	Description
1987-04-24	ST	Notification of lapse