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ES8707188A1 - Compounds having antibacterial activity, their preparation and use - Google Patents

Compounds having antibacterial activity, their preparation and use

Info

Publication number
ES8707188A1
ES8707188A1 ES555246A ES555246A ES8707188A1 ES 8707188 A1 ES8707188 A1 ES 8707188A1 ES 555246 A ES555246 A ES 555246A ES 555246 A ES555246 A ES 555246A ES 8707188 A1 ES8707188 A1 ES 8707188A1
Authority
ES
Spain
Prior art keywords
antibacterial activity
compounds
preparation
image
different
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES555246A
Other languages
Spanish (es)
Other versions
ES555246A0 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Schering SpA
Original Assignee
Schering SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering SpA filed Critical Schering SpA
Publication of ES8707188A1 publication Critical patent/ES8707188A1/en
Publication of ES555246A0 publication Critical patent/ES555246A0/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Novel compounds of general formula (I> < IMAGE > wherein R is a C1-C4 alkyl group or a C3-C6 cycloalkyl group R' and R'', which may be the same or different, are selected from hydrogen, halogen atoms, methyl, trifluoromethyl or methoxy groups X and Y, which may be the same or different, are selected from a nitrogen atom, < IMAGE > and pharmaceutically acceptable base addition salts thereof, have a strong antibacterial activity.
ES555246A 1985-05-10 1986-05-09 Compounds having antibacterial activity, their preparation and use Expired ES8707188A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT20653/85A IT1200470B (en) 1985-05-10 1985-05-10 ANTIBACTERIAL ACTIVITY COMPOUNDS, THEIR PREPARATION AND RELATED PHARMACEUTICAL COMPOSITIONS

Publications (2)

Publication Number Publication Date
ES8707188A1 true ES8707188A1 (en) 1987-07-16
ES555246A0 ES555246A0 (en) 1987-07-16

Family

ID=11170084

Family Applications (1)

Application Number Title Priority Date Filing Date
ES555246A Expired ES8707188A1 (en) 1985-05-10 1986-05-09 Compounds having antibacterial activity, their preparation and use

Country Status (6)

Country Link
JP (1) JPS61277668A (en)
DE (1) DE3615303A1 (en)
ES (1) ES8707188A1 (en)
FR (1) FR2583418A1 (en)
GB (1) GB2174704A (en)
IT (1) IT1200470B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8625325D0 (en) * 1986-10-22 1986-11-26 Glaxo Group Ltd Chemical compounds
US5262417A (en) * 1988-12-06 1993-11-16 The Upjohn Company Antibacterial quinolone compounds

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5624671B2 (en) * 1973-07-05 1981-06-08
JPS5824438B2 (en) * 1974-02-12 1983-05-20 大日本製薬株式会社 2-(1-piperazinyl) pyrido (2,3-D) pyrimidine
DE2903850A1 (en) * 1979-02-01 1980-08-07 Bayer Ag 2-AMINO-8-CYCLOPROPYL-5-OXO-5,8- DIHYDRO-PYRIDO CORNER CLAMP ON 2,3-D CORNER CLAMP FOR -PYRIMIDINE-6-CARNONIC ACIDS, METHOD FOR THE PRODUCTION AND USE THEREOF
DE3033157A1 (en) * 1980-09-03 1982-04-01 Bayer Ag, 5090 Leverkusen 7-AMINO-1-CYCLOPROPYL-4-OXO-1,4-DIHYDRO-NAPHTHYRIDINE-3-CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THE ANTIBACTERIAL AGENTS CONTAINING THEM
DE3306772A1 (en) * 1983-02-25 1984-08-30 Bayer Ag, 5090 Leverkusen CHINOLONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THE ANTIBACTERIAL AGENTS CONTAINING THEM
DE3308908A1 (en) * 1983-03-12 1984-09-13 Bayer Ag, 5090 Leverkusen BACTERICIDAL AGENTS
NZ208470A (en) * 1983-07-18 1988-06-30 Abbott Lab 6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid derivatives and antibacterial compositions containing such

Also Published As

Publication number Publication date
IT1200470B (en) 1989-01-18
DE3615303A1 (en) 1986-11-13
GB8610985D0 (en) 1986-06-11
IT8520653A0 (en) 1985-05-10
ES555246A0 (en) 1987-07-16
FR2583418A1 (en) 1986-12-19
JPS61277668A (en) 1986-12-08
GB2174704A (en) 1986-11-12

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